(E)-Alkenes as replacements of amide bonds: Development of novel and potent acyclic CGRP receptor antagonists
Kim, June J., Wood, Michael R., Stachel, Shawn J., de Leon, Pablo, Nomland, Ashley, Stump, Craig A., McWherter, Melody A., Schirripa, Kathy M., Moore, Eric L., Salvatore, Christopher A., Selnick, Harold G.
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
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Journal Article
Development of Orally Bioavailable and CNS Penetrant Biphenylaminocyclopropane Carboxamide Bradykinin B1 Receptor Antagonists
Kuduk, Scott D., Di Marco, Christina N., Chang, Ronald K., Wood, Michael R., Schirripa, Kathy M., Kim, June J., Wai, Jenny M. C., DiPardo, Robert M., Murphy, Kathy L., Ransom, Richard W., Harrell, C. Meacham, Reiss, Duane R., Holahan, Marie A., Cook, Jacquelynn, Hess, J. Fred, Sain, Nova, Urban, Mark O., Tang, Cuyue, Prueksaritanont, Thomayant, Pettibone, Douglas J., Bock, Mark G.
Published in Journal of medicinal chemistry (25.01.2007)
Published in Journal of medicinal chemistry (25.01.2007)
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Journal Article
Novel CGRP receptor antagonists from central amide replacements causing a reversal of preferred chirality
Wood, Michael R., Schirripa, Kathy M., Kim, June J., Bednar, Rodney A., Fay, John F., Bruno, Joseph G., Moore, Eric L., Mosser, Scott D., Roller, Shane, Salvatore, Christopher A., Vacca, Joseph P., Selnick, Harold G.
Published in Bioorganic & medicinal chemistry letters (15.11.2010)
Published in Bioorganic & medicinal chemistry letters (15.11.2010)
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Journal Article
Cyclopropylamino Acid Amide as a Pharmacophoric Replacement for 2,3-Diaminopyridine. Application to the Design of Novel Bradykinin B1 Receptor Antagonists
Wood, Michael R, Schirripa, Kathy M, Kim, June J, Wan, Bang-Lin, Murphy, Kathy L, Ransom, Richard W, Chang, Raymond S. L, Tang, Cuyue, Prueksaritanont, Thomayant, Detwiler, Theodore J, Hettrick, Lisa A, Landis, Elizabeth R, Leonard, Yvonne M, Krueger, Julie A, Lewis, Sidney D, Pettibone, Douglas J, Freidinger, Roger M, Bock, Mark G
Published in Journal of medicinal chemistry (23.02.2006)
Published in Journal of medicinal chemistry (23.02.2006)
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Journal Article
Novel CGRP receptor antagonists through a design strategy of target simplification with addition of molecular flexibility
Wood, Michael R., Schirripa, Kathy M., Kim, June J., Quigley, Amy G., Stump, Craig A., Bell, Ian M., Bednar, Rodney A., Fay, John F., Bruno, Joseph G., Moore, Eric L., Mosser, Scott D., Roller, Shane, Salvatore, Christopher A., Kane, Stefanie A., Vacca, Joseph P., Selnick, Harold G.
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
Published in Bioorganic & medicinal chemistry letters (01.10.2009)
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Journal Article
α-Hydroxy amides as a novel class of bradykinin B1 selective antagonists
WOOD, Michael R, SCHIRRIPA, Kathy M, CHANG, Raymond S. L, HOLAHAN, Marie A, COOK, Jacquelynn J, LEMAIRE, Wei, MOSSER, Scott D, BEDNAR, Rodney A, CUYUE TANG, PRUEKSARITANONT, Thomayant, WALLACE, Audrey A, QIN MEI, KIM, June J, JIAN YU, BOHN, Dennis L, CLAYTON, Frank C, ADARAYN, Emily D, SITKO, Gary R, LEONARD, Yvonne M, FREIDINGER, Roger M, PETTIBONE, Douglas J, BOCK, Mark G, KUDUK, Scott D, CHANG, Ronald K, DI MARCO, Christina N, DIPARDO, Robert M, WAN, Bang-Lin, MURPHY, Kathy L, RANSOM, Richard W
Published in Bioorganic & medicinal chemistry letters (15.01.2008)
Published in Bioorganic & medicinal chemistry letters (15.01.2008)
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Journal Article
5-Piperazinyl pyridine carboxamide bradykinin B1 antagonists
Kuduk, Scott D., Di Marco, Christina Ng, Chang, Ronald K., Wood, Michael R., Kim, June J., Schirripa, Kathy M., Murphy, Kathy L., Ransom, Richard W., Tang, Cuyue, Torrent, Maricel, Ha, Sookhee, Prueksaritanont, Thomayant, Pettibone, Douglas J., Bock, Mark G.
Published in Bioorganic & medicinal chemistry letters (15.05.2006)
Published in Bioorganic & medicinal chemistry letters (15.05.2006)
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Journal Article
Benzodiazepines as Potent and Selective Bradykinin B1 Antagonists
Wood, Michael R, Kim, June J, Han, Wei, Dorsey, Bruce D, Homnick, Carl F, DiPardo, Robert M, Kuduk, Scott D, MacNeil, Tanya, Murphy, Kathy L, Lis, Edward V, Ransom, Richard W, Stump, Gary L, Lynch, Joseph J, O'Malley, Stacey S, Miller, Patricia J, Chen, Tsing-Bau, Harrell, Charles M, Chang, Raymond S. L, Sandhu, Punam, Ellis, Joan D, Bondiskey, Peter J, Pettibone, Douglas J, Freidinger, Roger M, Bock, Mark G
Published in Journal of medicinal chemistry (08.05.2003)
Published in Journal of medicinal chemistry (08.05.2003)
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Journal Article
Development of orally bioavailable and CNS penetrant biphenylaminocyclopropane carboxamide bradykinin B-1 receptor antagonists
Kuduk, Scott D., Di Marco, Christina N., Chang, Ronald K., Wood, Michael R., Schirripa, Kathy M., Kim, June J., Wai, Jenny M. C., DiPardo, Robert M., Murphy, Kathy L., Ransom, Richard W., Harrell, C. Meacham, Reiss, Duane R., Holahan, Marie A., Cook, Jacquelynn, Hess, J. Fred, Sain, Nova, Urban, Mark O., Tang, Cuyue, Prueksaritanont, Thomayant, Pettibone, Douglas J., Bock, Mark G.
Published in Journal of medicinal chemistry (25.01.2007)
Published in Journal of medicinal chemistry (25.01.2007)
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Journal Article
Cyclopropylamino acid amide as a pharmacophoric replacement for 2,3-diaminopyridine. Application to the design of novel bradykinin B-1 receptor antagonists
Wood, MR, Schirripa, KM, Kim, JJ, Wan, BL, Murphy, KL, Ransom, RW, Chang, RSL, Tang, CY, Prueksaritanont, T, Detwiler, TJ, Hettrick, LA, Landis, ER, Leonard, YM, Krueger, JA, Lewis, SD, Pettibone, DJ, Freidinger, RM, Bock, MG
Published in Journal of medicinal chemistry (23.02.2006)
Published in Journal of medicinal chemistry (23.02.2006)
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Journal Article
α-Hydroxy amides as a novel class of bradykinin B 1 selective antagonists
Wood, Michael R., Schirripa, Kathy M., Kim, June J., Kuduk, Scott D., Chang, Ronald K., Di Marco, Christina N., DiPardo, Robert M., Wan, Bang-Lin, Murphy, Kathy L., Ransom, Richard W., Chang, Raymond S.L., Holahan, Marie A., Cook, Jacquelynn J., Lemaire, Wei, Mosser, Scott D., Bednar, Rodney A., Tang, Cuyue, Prueksaritanont, Thomayant, Wallace, Audrey A., Mei, Qin, Yu, Jian, Bohn, Dennis L., Clayton, Frank C., Adarayn, Emily D., Sitko, Gary R., Leonard, Yvonne M., Freidinger, Roger M., Pettibone, Douglas J., Bock, Mark G.
Published in Bioorganic & medicinal chemistry letters (15.01.2008)
Published in Bioorganic & medicinal chemistry letters (15.01.2008)
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Journal Article
Benzodiazepines as potent and selective bradykinin B-1 antagonists
Wood, MR, Kim, JJ, Han, W, Dorsey, BD, Homnick, CF, DiPardo, RM, Kuduk, SD, MacNeil, T, Murphy, KL, Lis, EV, Ransom, RW, Stump, GL, Lynch, JJ, O'Malley, SS, Miller, PJ, Chen, TB, Harrell, CM, Chang, RSL, Sandhu, P, Ellis, JD, Bondiskey, PJ, Pettibone, DJ, Freidinger, RM, Bock, MG
Published in Journal of medicinal chemistry (08.05.2003)
Published in Journal of medicinal chemistry (08.05.2003)
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Journal Article
alpha -Hydroxy amides as a novel class of bradykinin B sub(1) selective antagonists
Wood, Michael R, Schirripa, Kathy M, Kim, June J, Kuduk, Scott D, Chang, Ronald K, Di Marco, Christina N, DiPardo, Robert M, Wan, Bang-Lin, Murphy, Kathy L, Ransom, Richard W, Chang, Raymond SL, Holahan, Marie A, Cook, Jacquelynn J, Lemaire, Wei, Mosser, Scott D, Bednar, Rodney A, Tang, Cuyue, Prueksaritanont, Thomayant, Wallace, Audrey A, Mei, Qin, Yu, Jian, Bohn, Dennis L, Clayton, Frank C, Adarayn, Emily D, Sitko, Gary R, Leonard, Yvonne M, Freidinger, Roger M, Pettibone, Douglas J, Bock, Mark G
Published in Bioorganic & medicinal chemistry (01.01.2008)
Published in Bioorganic & medicinal chemistry (01.01.2008)
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Journal Article
5-Piperazinyl pyridine carboxamide bradykinin B sub(1) antagonists
Kuduk, Scott D, Di Marco, Christina Ng, Chang, Ronald K, Wood, Michael R, Kim, June J, Schirripa, Kathy M, Murphy, Kathy L, Ransom, Richard W, Tang, Cuyue, Torrent, Maricel, Ha, Sookhee, Prueksaritanont, Thomayant, Pettibone, Douglas J, Bock, Mark G
Published in Bioorganic & medicinal chemistry letters (01.01.2006)
Published in Bioorganic & medicinal chemistry letters (01.01.2006)
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Journal Article
4-1BB T-cell antigen binds to mature B cells and macrophages, and costimulates anti-mu-primed splenic B cells
Pollok, K E, Kim, Y J, Hurtado, J, Zhou, Z, Kim, K K, Kwon, B S
Published in European journal of immunology (01.02.1994)
Published in European journal of immunology (01.02.1994)
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Journal Article
1,3-SUBSTITUTED AZETIDINE PDE10 INHIBITORS
KIM, JUNE, J, STEEN, JUSTIN, T, BESHORE, DOUGLAS, C, KUDUK, SCOTT, D, REGER, THOMAS, COX, CHRISTOPHER, D, MCVEAN, CAROL
Year of Publication 10.08.2016
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Year of Publication 10.08.2016
Patent
1,3 substituted azetidine PDE10 inhibitors
COX CHRISTOPHER D, BESHORE DOUGLAS C, REGER THOMAS, KIM JUNE J, SHEEN JUSTIN T, MCVEAN CAROL A, KUDUK SCOTT D
Year of Publication 14.06.2016
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Year of Publication 14.06.2016
Patent