Novel Carboxamide-Based Allosteric MEK Inhibitors: Discovery and Optimization Efforts toward XL518 (GDC-0973)
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Published in ACS medicinal chemistry letters (10.05.2012)
Published in ACS medicinal chemistry letters (10.05.2012)
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Discovery of XL888: A novel tropane-derived small molecule inhibitor of HSP90
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Published in Bioorganic & medicinal chemistry letters (01.09.2012)
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
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Use of a Conformational Radical Clock for Evaluating Alkyllithium-Mediated Cyclization Reactions
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Published in Organic letters (22.03.2001)
Published in Organic letters (22.03.2001)
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RECEPTOR-TYPE KINASE MODULATORS AND METHODS OF USE
RICE, Kenneth, D, ANAND, Neel, Kumar, COSTANZO, Simona, KENNEDY, Abigail, R, BUSSENIUS, Joerg, KIM, Angie, I, PETO, Csaba, J, BLAZEY, Charles, M, TSANG, Tsze, H
Year of Publication 05.09.2018
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Year of Publication 05.09.2018
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Process for preparing receptor-type kinase modulators
KIM, ANGIE I, BUSSENIUS, JOERG, KENNEDY, ABIGAIL R, COSTANZA, SIMONA, PETO, CSABA J, RICE, KENNETH D, ANAND, NEEL KUMAR, BLAZEY, CHARLES M, TSANG, TSZE H
Year of Publication 02.04.2014
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Year of Publication 02.04.2014
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RECEPTOR-TYPE KINASE MODULATORS AND METHODS OF USE
KIM, ANGIE I, BUSSENIUS, JOERG, KENNEDY, ABIGAIL R, PETO, CSABA J, RICE, KENNETH D, ANAND, NEEL KUMAR, BLAZEY, CHARLES M, COSTANZO, SIMONA, TSANG, TSZE H
Year of Publication 04.02.2014
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Year of Publication 04.02.2014
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Receptor-type kinase modulators and methods of use
KIM, ANGIE I, BUSSENIUS, JOERG, KENNEDY, ABIGAIL R, PETO, CSABA J, ANAND, NEEL KUMAR, RICE, KENNETH D, BLAZEY, CHARLES M, COSTANZO, SIMONA, TSANG, TSZE H
Year of Publication 16.05.2013
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Year of Publication 16.05.2013
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Anaplastic lymphoma kinase modulators and methods of use
MANALO, JEAN-CLAIRE L, BUSSENIUS, JOERG, KENNEDY, ABIGAIL R, PETO, CSABA J, DUBENKO, LARISA, KHOURY, RICHARD G, CURTIS, JEFFRY KIMO, BLAZEY, CHARLES M, COSTANZO, SIMONA, KIM, ANGIE I, BOWLES, OWEN JOSEPH, ANAND, NEEL KUMAR, RICE, KENNETH D, TSANG, TSZE H
Year of Publication 18.07.2013
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Year of Publication 18.07.2013
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ANAPLASTIC LYMPHOMA KINASE MODULATORS AND METHODS OF USE
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Year of Publication 18.06.2013
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Year of Publication 18.06.2013
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Receptor-type kinase modulators and methods of use
KIM, ANGIE I, BUSSENIUS, JOERG, KENNEDY, ABIGAIL R, PETO, CSABA J, ANAND, NEEL KUMAR, RICE, KENNETH D, BLAZEY, CHARLES M, COSTANZO, SIMONA, TSANG, TSZE H
Year of Publication 27.10.2011
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Year of Publication 27.10.2011
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Raf modulators and methods of use
KIM ANGIE I, DEFINA STEVEN CHARLES, JOSHI ANAGHA ABHIJIT, MANALO JEAN-CLAIRE L, BOWLES OWEN JOSEPH, COSTANZO SIMONA, KENNEDY ABIGAIL R, ANAND NEEL KUMAR, BUSSENIUS JOERG, TSANG TSZE H, BLAZEY CHARLES M, CURTIS JEFFRY KIMO, PETO CSABA J, RICE KENNETH D, DUBENKO LARISA
Year of Publication 15.04.2014
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Year of Publication 15.04.2014
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RAF MODULATORS AND METHODS OF USE
MANALO, JEAN-CLAIRE L, BUSSENIUS, JOERG, KENNEDY, ABIGAIL R, PETO, CSABA J, DUBENKO, LARISA, CURTIS, JEFFRY KIMO, BLAZEY, CHARLES M, COSTANZO, SIMONA, KIM, ANGIE I, JOSHI, ANAGHA ABHIJIT, BOWLES, OWEN JOSEPH, ANAND, NEEL KUMAR, RICE, KENNETH D, TSANG, TSZE H, DEFINA, STEVEN CHARLES
Year of Publication 24.12.2013
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Year of Publication 24.12.2013
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RECEPTOR TYPE KINASE MODULATORS AND METHODS OF USE
KIM ANGIE I, ANAND NEEL KUMAR, BUSSENIUS JOERG, TSANG TSZE H, BLAZEY CHARLES M, RICE KENNETH D, PETO CSABA J, KENNEDY ABIGAIL R, COSTANZA SIMONA
Year of Publication 21.04.2011
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Year of Publication 21.04.2011
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Anaplastic lymphoma kinase modulators and methods of use
MANALO, JEAN-CLAIRE L, BUSSENIUS, JOERG, KENNEDY, ABIGAIL R, PETO, CSABA J, DUBENKO, LARISA, KHOURY, RICHARD G, CURTIS, JEFFRY KIMO, BLAZEY, CHARLES M, COSTANZO, SIMONA, KIM, ANGIE I, BOWLES, OWEN JOSEPH, ANAND, NEEL KUMAR, RICE, KENNETH D, TSANG, TSZE H
Year of Publication 02.08.2012
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Year of Publication 02.08.2012
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Process for preparing receptor-type kinase modulators
KIM, ANGIE I, BUSSENIUS, JOERG, KENNEDY, ABIGAIL R, COSTANZA, SIMONA, PETO, CSABA J, RICE, KENNETH D, ANAND, NEEL KUMAR, BLAZEY, CHARLES M, TSANG, TSZE H
Year of Publication 30.03.2011
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Year of Publication 30.03.2011
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