Optimization of Chemical Functionalities of Indole-2-carboxamides To Improve Allosteric Parameters for the Cannabinoid Receptor 1 (CB1)
Khurana, Leepakshi, Ali, Hamed I, Olszewska, Teresa, Ahn, Kwang H, Damaraju, Aparna, Kendall, Debra A, Lu, Dai
Published in Journal of medicinal chemistry (10.04.2014)
Published in Journal of medicinal chemistry (10.04.2014)
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Journal Article
Modulation of CB1 cannabinoid receptor by allosteric ligands: Pharmacology and therapeutic opportunities
Khurana, Leepakshi, Mackie, Ken, Piomelli, Daniele, Kendall, Debra A.
Published in Neuropharmacology (15.09.2017)
Published in Neuropharmacology (15.09.2017)
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Journal Article
Regulation of MIF Enzymatic Activity by an Allosteric Site at the Central Solvent Channel
Pantouris, Georgios, Khurana, Leepakshi, Ma, Anthony, Skeens, Erin, Reiss, Krystle, Batista, Victor S., Lisi, George P., Lolis, Elias J.
Published in Cell chemical biology (18.06.2020)
Published in Cell chemical biology (18.06.2020)
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Journal Article
Pyrimidinyl Biphenylureas: Identification of New Lead Compounds as Allosteric Modulators of the Cannabinoid Receptor CB1
Khurana, Leepakshi, Fu, Bo-Qiao, Duddupudi, Anantha L, Liao, Yu-Hsien, Immadi, Sri Sujana, Kendall, Debra A, Lu, Dai
Published in Journal of medicinal chemistry (09.02.2017)
Published in Journal of medicinal chemistry (09.02.2017)
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Journal Article
Computational analysis of the CB1 carboxyl-terminus in the receptor-G protein complex: Computational Analysis of the CB1 Carboxyl-Terminus
Shim, Joong-Youn, Khurana, Leepakshi, Kendall, Debra A.
Published in Proteins, structure, function, and bioinformatics (01.04.2016)
Published in Proteins, structure, function, and bioinformatics (01.04.2016)
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Journal Article
Structure–Activity Relationship in the Leucettine Family of Kinase Inhibitors
Tahtouh, Tania, Durieu, Emilie, Villiers, Benoît, Bruyère, Céline, Nguyen, Thu Lan, Fant, Xavier, Ahn, Kwang H, Khurana, Leepakshi, Deau, Emmanuel, Lindberg, Mattias F, Sévère, Elodie, Miege, Frédéric, Roche, Didier, Limanton, Emmanuelle, L’Helgoual’ch, Jean-Martial, Burgy, Guillaume, Guiheneuf, Solène, Herault, Yann, Kendall, Debra A, Carreaux, François, Bazureau, Jean-Pierre, Meijer, Laurent
Published in Journal of medicinal chemistry (27.01.2022)
Published in Journal of medicinal chemistry (27.01.2022)
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Journal Article
Pyrimidinyl Biphenylureas: Identification of New Lead Compounds as Allosteric Modulators of the Cannabinoid Receptor CB 1
Khurana, Leepakshi, Fu, Bo-Qiao, Duddupudi, Anantha L, Liao, Yu-Hsien, Immadi, Sri Sujana, Kendall, Debra A, Lu, Dai
Published in Journal of medicinal chemistry (09.02.2017)
Published in Journal of medicinal chemistry (09.02.2017)
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Journal Article