Identification and Profiling of a Novel Diazaspiro[3.4]octane Chemical Series Active against Multiple Stages of the Human Malaria Parasite Plasmodium falciparum and Optimization Efforts
Le Manach, Claire, Dam, Jean, Woodland, John G, Kaur, Gurminder, Khonde, Lutete P, Brunschwig, Christel, Njoroge, Mathew, Wicht, Kathryn J, Horatscheck, André, Paquet, Tanya, Boyle, Grant A, Gibhard, Liezl, Taylor, Dale, Lawrence, Nina, Yeo, Tomas, Mok, Sachel, Eastman, Richard T, Dorjsuren, Dorjbal, Talley, Daniel C, Guo, Hui, Simeonov, Anton, Reader, Janette, van der Watt, Mariëtte, Erlank, Erica, Venter, Nelius, Zawada, Jacek W, Aswat, Ayesha, Nardini, Luisa, Coetzer, Theresa L, Lauterbach, Sonja B, Bezuidenhout, Belinda C, Theron, Anjo, Mancama, Dalu, Koekemoer, Lizette L, Birkholtz, Lyn-Marie, Wittlin, Sergio, Delves, Michael, Ottilie, Sabine, Winzeler, Elizabeth A, von Geldern, Thomas W, Smith, Dennis, Fidock, David A, Street, Leslie J, Basarab, Gregory S, Duffy, James, Chibale, Kelly
Published in Journal of medicinal chemistry (25.02.2021)
Published in Journal of medicinal chemistry (25.02.2021)
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