Synthesis and antimalarial properties of 1-imino derivatives of 7-chloro-3-substituted-3,4-dihydro-1,9(2H,10H)-acridinediones and related structures
KESTEN, S. J, DEGNAN, M. J, HUNG, J, MCNAMARA, D. J, ORTWINE, D. F, UHLENDORF, S. E, WERBEL, L. M
Published in Journal of medicinal chemistry (18.09.1992)
Published in Journal of medicinal chemistry (18.09.1992)
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A SIMPLE AND EFFICIENT SYNTHESIS OF 2-(N-PHENYLAMINO)- BENZOIC ACIDS
Chen, M. H., Beylin, V. G., Iakovleva, E., Kesten, S. J., Magano, J., Vrieze, D.
Published in Synthetic communications (01.01.2002)
Published in Synthetic communications (01.01.2002)
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Nonpeptide angiotensin II receptor antagonists. 2. Design, synthesis, and structure-activity relationships of 2-alkyl-4-(1H-pyrrol-l-yl)-1H-imidazole derivatives: profile of 2-propyl-1-[[2'-(1H-tetrazol-5-yl)-[1,1'-biphenyl]-4-yl]-methyl]-4-[2-(trifluoroacetyl)-1H-pyrrol-1-yl]-1H-imidazole-5-carboxylic acid (CI-996)
Sircar, Ila, Hodges, John C, Quin, John, Bunker, Amy M, Winters, R. Thomas, Edmunds, Jeremy J, Kostlan, Catherine R, Connolly, Cleo, Kesten, Stephen J
Published in Journal of medicinal chemistry (06.08.1993)
Published in Journal of medicinal chemistry (06.08.1993)
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Synthesis, antimalarial activity, and quantitative structure-activity relationships of tebuquine and a series of related 5-[(7-chloro-4-quinolinyl)amino]3-[(alkylamino)methyl][1,1'-biphenyl]-2-ols and Nω-oxides
WERBEL, L. M, DAN COOK, P, ELSLAGER, E. F, HUNG, J. H, JOHNSON, J. L, KESTEN, S. J, MCNAMARA, D. J, ORTWINE, D. F, WORTH, D. F
Published in Journal of medicinal chemistry (01.06.1986)
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Published in Journal of medicinal chemistry (01.06.1986)
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Nonpeptide angiotensin II receptor antagonists. II: Design, synthesis, and structure-activity relationships of 2-alkyl-4(1H-pyrrol-1-yl)-1H-imidazole derivatives : profile of 2-propyl-1[[2'-(1H-tetrazol-5-yl)-[1,1'-biphenyl]-4-yl]-methyl]-4-[2-(trifluoroacetyl)-1H-pyrrol-1-yl]-1H-imidazole-5-carboxylic acid (CI-996)
SIRCAR, I, HODGES, J. C, TOPLISS, J. G, KEISER, J. A, PANEK, R. L, QUIN, J. III, BUNKER, A. M, WINTERS, R. T, EDMUNDS, J. J, KOSTLAN, C. R, CONNOLLY, C, KESTEN, S. J, HAMBY, J. M
Published in Journal of medicinal chemistry (1993)
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Published in Journal of medicinal chemistry (1993)
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Antimalarial drugs. 64. Synthesis and antimalarial properties of 1-imino derivatives of 7-chloro-3-substituted-3,4-dihydro-1,9(2H,10H)-acridinediones and related structures
Kesten, Stephen J, Degnan, Margaret J, Hung, Jocelyn, McNamara, Dennis J, Ortwine, Daniel F, Uhlendorf, Susan E, Werbel, Leslie M
Published in Journal of medicinal chemistry (01.09.1992)
Published in Journal of medicinal chemistry (01.09.1992)
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Pyrazolo[5,1-b]quinazolin-9-ones: a new series of antiallergic agents
Sircar, Jagadish C, Capiris, Thomas, Kesten, Stephen J, Herzig, David J
Published in Journal of medicinal chemistry (01.06.1981)
Published in Journal of medicinal chemistry (01.06.1981)
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ANTIMALARIAL-DRUGS .60. SYNTHESIS, ANTIMALARIAL ACTIVITY, AND QUANTITATIVE STRUCTURE-ACTIVITY-RELATIONSHIPS OF TEBUQUINE AND A SERIES OF RELATED 5-[(7-CHLORO-4-QUINOLINYL)AMINO]-3-[(ALKYLAMINO)METHYL][1,1'-BIPHENYL]-2-OLS AND N-OMEGA-OXIDES1,2
WERBEL, LM, COOK, PD, ELSLAGER, EF, HUNG, JH, JOHNSON, JL, KESTEN, SJ, MCNAMARA, DJ, ORTWINE, DF, WORTH, DF
Published in Journal of medicinal chemistry (01.06.1986)
Published in Journal of medicinal chemistry (01.06.1986)
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