Stapled α−helical peptide drug development: A potent dual inhibitor of MDM2 and MDMX for p53-dependent cancer therapy
Chang, Yong S, Graves, Bradford, Guerlavais, Vincent, Tovar, Christian, Packman, Kathryn, To, Kwong-Him, Olson, Karen A, Kesavan, Kamala, Gangurde, Pranoti, Mukherjee, Aditi, Baker, Theresa, Darlak, Krzysztof, Elkin, Carl, Filipovic, Zoran, Qureshi, Farooq Z, Cai, Hongliang, Berry, Pamela, Feyfant, Eric, Shi, Xiangguo E, Horstick, James, Annis, D Allen, Manning, Anthony M, Fotouhi, Nader, Nash, Huw, Vassilev, Lyubomir T, Sawyer, Tomi K
Published in Proceedings of the National Academy of Sciences - PNAS (03.09.2013)
Published in Proceedings of the National Academy of Sciences - PNAS (03.09.2013)
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Journal Article
Annexin A2 Is a Molecular Target for TM601, a Peptide with Tumor-targeting and Anti-angiogenic Effects
Kesavan, Kamala, Ratliff, Judson, Johnson, Eric W., Dahlberg, William, Asara, John M., Misra, Preeti, Frangioni, John V., Jacoby, Douglas B.
Published in The Journal of biological chemistry (12.02.2010)
Published in The Journal of biological chemistry (12.02.2010)
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Journal Article
MEKK2 regulates the coordinate activation of ERK5 and JNK in response to FGF-2 in fibroblasts
Kesavan, Kamala, Lobel-Rice, Katherine, Sun, Weiyong, Lapadat, Razvan, Webb, Saiphone, Johnson, Gary L., Garrington, Timothy P.
Published in Journal of cellular physiology (01.04.2004)
Published in Journal of cellular physiology (01.04.2004)
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Journal Article
MEKK2 Associates with the Adapter Protein Lad/RIBP and Regulates the MEK5-BMK1/ERK5 Pathway
Sun, Weiyong, Kesavan, Kamala, Schaefer, Brian C., Garrington, Timothy P., Ware, Margaret, Johnson, Nancy Lassignal, Gelfand, Erwin W., Johnson, Gary L.
Published in The Journal of biological chemistry (16.02.2001)
Published in The Journal of biological chemistry (16.02.2001)
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Journal Article
MEK Kinase 2 and the Adaptor Protein Lad Regulate Extracellular Signal-Regulated Kinase 5 Activation by Epidermal Growth Factor via Src
Sun, Weiyong, Wei, Xudong, Kesavan, Kamala, Garrington, Timothy P., Fan, Ruihua, Mei, Junjie, Anderson, Steven M., Gelfand, Erwin W., Johnson, Gary L.
Published in Molecular and Cellular Biology (01.04.2003)
Published in Molecular and Cellular Biology (01.04.2003)
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Journal Article
Characterization of the in Vivo Sites of Serine Phosphorylation on Lck Identifying Serine 59 as a Site of Mitotic Phosphorylation
Kesavan, Kamala P., Isaacson, Christina C., Ashendel, Curtis L., Geahlen, Robert L., Harrison, Marietta L.
Published in The Journal of biological chemistry (26.04.2002)
Published in The Journal of biological chemistry (26.04.2002)
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Journal Article
Discovery of Sulanemadlin (ALRN-6924), the First Cell-Permeating, Stabilized α‑Helical Peptide in Clinical Development
Guerlavais, Vincent, Sawyer, Tomi K., Carvajal, Luis, Chang, Yong S., Graves, Bradford, Ren, Jian-Guo, Sutton, David, Olson, Karen A., Packman, Kathryn, Darlak, Krzysztof, Elkin, Carl, Feyfant, Eric, Kesavan, Kamala, Gangurde, Pranoti, Vassilev, Lyubomir T., Nash, Huw M., Vukovic, Vojislav, Aivado, Manuel, Annis, D. Allen
Published in Journal of medicinal chemistry (27.07.2023)
Published in Journal of medicinal chemistry (27.07.2023)
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Journal Article
Analysis of Notch1 Function by In Vitro T Cell Differentiation of Pax5 Mutant Lymphoid Progenitors
Hoflinger, Sonja, Kesavan, Kamala, Fuxa, Martin, Hutter, Caroline, Heavey, Barry, Radtke, Freddy, Busslinger, Meinrad
Published in The Journal of immunology (1950) (15.09.2004)
Published in The Journal of immunology (1950) (15.09.2004)
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Journal Article
Agents that bind annexin A2 suppress ocular neovascularization
Lima e Silva, Raquel, Shen, Jikui, Gong, Yuan Yuan, Seidel, Christopher P., Hackett, Sean F., Kesavan, Kamala, Jacoby, Douglas B., Campochiaro, Peter A.
Published in Journal of cellular physiology (01.12.2010)
Published in Journal of cellular physiology (01.12.2010)
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Journal Article
Stapled α-helical peptide drug development: A potent dual inhibitor of MDM2 and MDMX for p53-dependent cancer therapy
Chang, Yong S., Graves, Bradford, Guerlavais, Vincent, Tovar, Christian, Packman, Kathryn, To, Kwong-Him, Olson, Karen A., Kesavan, Kamala, Gangurde, Pranoti, Mukherjee, Aditi, Baker, Theresa, Darlak, Krzysztof, Elkin, Carl, Filipovic, Zoran, Qureshi, Farooq Z., Cai, Hongliang, Berry, Pamela, Feyfant, Eric, Shi, Xiangguo E., Horstick, James, Annis, D. Allen, Manning, Anthony M., Fotouhi, Nader, Nash, Huw, Vassilev, Lyubomir T., Sawyer, Tomi K.
Published in Proceedings of the National Academy of Sciences - PNAS (03.09.2013)
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Published in Proceedings of the National Academy of Sciences - PNAS (03.09.2013)
Journal Article
Stapled [alpha]-helical peptide drug development: A potent dual inhibitor of MDM2 and MDMX for p53-dependent cancer therapy
Chang, Yong S, Graves, Bradford, Guerlavais, Vincent, Tovar, Christian, Packman, Kathryn, To, Kwong-Him, Olson, Karen A, Kesavan, Kamala, Gangurde, Pranoti, Mukherjee, Aditi, Baker, Theresa, Darlak, Krzysztof, Elkin, Carl, Filipovic, Zoran, Qureshi, Farooq Z, Cai, Hongliang, Berry, Pamela, Feyfant, Eric, Shi, Xiangguo E, Horstick, James, Annis, D Allen, Manning, Anthony M, Fotouhi, Nader, Nash, Huw, Vassilev, Lyubomir T, Sawyer, Tomi K
Published in Proceedings of the National Academy of Sciences - PNAS (03.09.2013)
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Published in Proceedings of the National Academy of Sciences - PNAS (03.09.2013)
Journal Article
Abstract B217: Annexin A2 is a novel molecular target for TM601, a peptide with specific tumor targeting and antiangiogenic properties
Kesavan, Kamala, Ratliff, Judson, Johnson, Eric, Dahlberg, William, Jacoby, Douglas B.
Published in Molecular cancer therapeutics (10.12.2009)
Published in Molecular cancer therapeutics (10.12.2009)
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Journal Article
MEKK1 regulates calpain‐dependent proteolysis of focal adhesion proteins for rear‐end detachment of migrating fibroblasts
Cuevas, Bruce D., Abell, Amy N., Witowsky, James A., Yujiri, Toshiaki, Johnson, Nancy Lassignal, Kesavan, Kamala, Ware, Marti, Jones, Peter L., Weed, Scott A., DeBiasi, Roberta L., Oka, Yoshitomo, Tyler, Kenneth L., Johnson, Gary L.
Published in The EMBO journal (01.07.2003)
Published in The EMBO journal (01.07.2003)
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Journal Article
MEKK1 regulates calpain-dependent proteolysis of focal adhesion proteins for rear-end detachment of migrating fibroblasts
Cuevas, Bruce D., Abell, Amy N., Witowsky, James A., Yujiri, Toshiaki, Johnson, Nancy Lassignal, Kesavan, Kamala, Ware, Marti, Jones, Peter L., Weed, Scott A., DeBiasi, Roberta L., Oka, Yoshitomo, Tyler, Kenneth L., Johnson, Gary L.
Published in The EMBO journal (01.07.2003)
Published in The EMBO journal (01.07.2003)
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Journal Article
INHIBITION OF ANGIOGENESIS
JACOBY, DOUGLAS, B, KESAVAN, KAMALA, SENTISSI, ABDELLAH, EGAN, E. MICHAEL
Year of Publication 17.06.2015
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Year of Publication 17.06.2015
Patent
Treatment of metastatic tumors
Sentissi Abdellah, Jacoby Douglas B, Egan E. Michael, Kesavan Kamala, O'Neill Alison
Year of Publication 28.03.2017
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Year of Publication 28.03.2017
Patent
tratamento de tumores metastáticos
ABDELLAH SENTISSI, ALISON O' NEILL, KAMALA KESAVAN, E. MICHAEL EGAN, DOUGLAS B. JACOBY
Year of Publication 26.01.2016
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Year of Publication 26.01.2016
Patent