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Published in Journal of medicinal chemistry (27.02.2020)
Published in Journal of medicinal chemistry (27.02.2020)
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Published in Bioorganic & medicinal chemistry (01.02.2008)
Published in Bioorganic & medicinal chemistry (01.02.2008)
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Estuaries and Coasts as an Outlet for Research in Coastal Ecosystems: A Bibliometric Study
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1-Benzylbenzimidazoles : The discovery of a novel series of bradykinin B1 receptor antagonists
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Published in Bioorganic & medicinal chemistry letters (15.09.2008)
Published in Bioorganic & medicinal chemistry letters (15.09.2008)
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Near real-time monitoring of the Biscayne Bay Watershed (South Florida, USA) and major tributaries by water quality research buoys
Troxell, Kassidy, Schonhoff, Bradley, Kershaw, Mark, Ceccopieri, Milena, Crowl, Todd, Gardinali, Piero
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Discovery and Optimization of Quinolinone Derivatives as Potent, Selective, and Orally Bioavailable Mutant Isocitrate Dehydrogenase 1 (mIDH1) Inhibitors
Lin, Jian, Lu, Wei, Caravella, Justin A, Campbell, Ann Marie, Diebold, R. Bruce, Ericsson, Anna, Fritzen, Edward, Gustafson, Gary R, Lancia, David R, Shelekhin, Tatiana, Wang, Zhongguo, Castro, Jennifer, Clarke, Andrea, Gotur, Deepali, Josephine, Helen R, Katz, Marie, Diep, Hien, Kershaw, Mark, Yao, Lili, Kauffman, Goss, Hubbs, Stephen E, Luke, George P, Toms, Angela V, Wang, Liann, Bair, Kenneth W, Barr, Kenneth J, Dinsmore, Christopher, Walker, Duncan, Ashwell, Susan
Published in Journal of medicinal chemistry (25.07.2019)
Published in Journal of medicinal chemistry (25.07.2019)
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Discovery and optimization of novel piperazines as potent inhibitors of fatty acid synthase (FASN)
Martin, Matthew W., Lancia, David R., Li, Hongbin, Schiller, Shawn E.R., Toms, Angela V., Wang, Zhongguo, Bair, Kenneth W., Castro, Jennifer, Fessler, Shawn, Gotur, Deepali, Hubbs, Stephen E., Kauffman, Goss S., Kershaw, Mark, Luke, George P., McKinnon, Crystal, Yao, Lili, Lu, Wei, Millan, David S.
Published in Bioorganic & medicinal chemistry letters (15.04.2019)
Published in Bioorganic & medicinal chemistry letters (15.04.2019)
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FT-1101: A Structurally Distinct Pan-BET Bromodomain Inhibitor with Activity in Preclinical Models of Hematologic Malignancies
Millan, David S, Alvarez Morales, Monica A, Barr, Kenneth J, Cardillo, Daniel, Collis, Alan, Dinsmore, Christopher J, Escobedo, Jaime A, Foley, Kevin P, Herbertz, Torsten, Hubbs, Stephen, Kauffman, Goss S, Kayser-Bricker, Katherine J, Kershaw, Mark T, Luke, George P, Martin, Matthew W, McKinnon, Crystal, Mendes, Rachel L, Muskiewicz, Kristina R, Schiller, Shawn ER, Soulard, Patricia, Talbot, Adam C, Walker, Duncan, Yao, Lili, Williams, Grace L
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1-Benzylbenzimidazoles: The discovery of a novel series of bradykinin B 1 receptor antagonists
Guo, Qin, Chandrasekhar, Jayaraman, Ihle, David, Wustrow, David J., Chenard, Bertrand L., Krause, James E., Hutchison, Alan, Alderman, Dawn, Cheng, Charles, Cortright, Daniel, Broom, Daniel, Kershaw, Mark T., Simmermacher-Mayer, Jean, Peng, Yao, Hodgetts, Kevin J.
Published in Bioorganic & medicinal chemistry letters (15.09.2008)
Published in Bioorganic & medicinal chemistry letters (15.09.2008)
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Aminoquinazolines as TRPV1 antagonists: Modulation of drug-like properties through the exploration of 2-position substitution
Blum, Charles A., Zheng, Xiaozhang, Brielmann, Harry, Hodgetts, Kevin J., Bakthavatchalam, Rajagopal, Chandrasekhar, Jayaraman, Krause, James E., Cortright, Daniel, Matson, David, Crandall, Marci, Ngo, Chu K., Fung, Lawrence, Day, Marta, Kershaw, Mark, De Lombaert, Stéphane, Chenard, Bertrand L.
Published in Bioorganic & medicinal chemistry (15.08.2008)
Published in Bioorganic & medicinal chemistry (15.08.2008)
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1-Benzylbenzimidazoles: The discovery of a novel series of bradykinin B sub(1) receptor antagonists
Guo, Qin, Chandrasekhar, Jayaraman, Ihle, David, Wustrow, David J, Chenard, Bertrand L, Krause, James E, Hutchison, Alan, Alderman, Dawn, Cheng, Charles, Cortright, Daniel, Broom, Daniel, Kershaw, Mark T, Simmermacher-Mayer, Jean, Peng, Yao, Hodgetts, Kevin J
Published in Bioorganic & medicinal chemistry (01.09.2008)
Published in Bioorganic & medicinal chemistry (01.09.2008)
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Aminopyrazine CB1 receptor inverse agonists
Wustrow, David J., Maynard, George D., Yuan, Jun, Zhao, He, Mao, Jianmin, Guo, Qin, Kershaw, Mark, Hammer, Jack, Brodbeck, Robbin M., Near, Kristen E., Zhou, Dan, Beers, David S., Chenard, Bertrand L., Krause, James E., Hutchison, Alan J.
Published in Bioorganic & medicinal chemistry (01.06.2008)
Published in Bioorganic & medicinal chemistry (01.06.2008)
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1-Benzylbenzimidazoles: the discovery of a novel series of bradykinin B(1) receptor antagonists
Guo, Qin, Chandrasekhar, Jayaraman, Ihle, David, Wustrow, David J, Chenard, Bertrand L, Krause, James E, Hutchison, Alan, Alderman, Dawn, Cheng, Charles, Cortright, Daniel, Broom, Daniel, Kershaw, Mark T, Simmermacher-Mayer, Jean, Peng, Yao, Hodgetts, Kevin J
Published in Bioorganic & medicinal chemistry letters (15.09.2008)
Published in Bioorganic & medicinal chemistry letters (15.09.2008)
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