Carbazole-containing amides and ureas: Discovery of cryptochrome modulators as antihyperglycemic agents
Humphries, Paul S., Bersot, Ross, Kincaid, John, Mabery, Eric, McCluskie, Kerryn, Park, Timothy, Renner, Travis, Riegler, Erin, Steinfeld, Tod, Turtle, Eric D., Wei, Zhi-Liang, Willis, Erik
Published in Bioorganic & medicinal chemistry letters (01.02.2018)
Published in Bioorganic & medicinal chemistry letters (01.02.2018)
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Journal Article
Carbazole-containing sulfonamides and sulfamides: Discovery of cryptochrome modulators as antidiabetic agents
Humphries, Paul S., Bersot, Ross, Kincaid, John, Mabery, Eric, McCluskie, Kerryn, Park, Timothy, Renner, Travis, Riegler, Erin, Steinfeld, Tod, Turtle, Eric D., Wei, Zhi-Liang, Willis, Erik
Published in Bioorganic & medicinal chemistry letters (01.02.2016)
Published in Bioorganic & medicinal chemistry letters (01.02.2016)
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Journal Article
Optimizing human α-galactosidase for treatment of Fabry disease
Hallows, William C., Skvorak, Kristen, Agard, Nick, Kruse, Nikki, Zhang, Xiyun, Zhu, Yu, Botham, Rachel C., Chng, Chinping, Shukla, Charu, Lao, Jessica, Miller, Mathew, Sero, Antoinette, Viduya, Judy, Ismaili, Moulay Hicham Alaoui, McCluskie, Kerryn, Schiffmann, Raphael, Silverman, Adam P., Shen, Jin-Song, Huisman, Gjalt W.
Published in Scientific reports (23.03.2023)
Published in Scientific reports (23.03.2023)
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Journal Article
Novel Role for the Liver X Nuclear Receptor in the Suppression of Lung Inflammatory Responses
Birrell, Mark A., Catley, Matthew C., Hardaker, Elizabeth, Wong, Sissie, Willson, Timothy M., McCluskie, Kerryn, Leonard, Thomas, Farrow, Stuart N., Collins, Jon L., Haj-Yahia, Saleem, Belvisi, Maria G.
Published in The Journal of biological chemistry (02.11.2007)
Published in The Journal of biological chemistry (02.11.2007)
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Journal Article
Nitric Oxide as a Noninvasive Biomarker of Lipopolysaccharide-Induced Airway Inflammation: Possible Role in Lung Neutrophilia
McCluskie, Kerryn, Birrell, Mark A, Wong, Sissie, Belvisi, Maria G
Published in The Journal of pharmacology and experimental therapeutics (01.11.2004)
Published in The Journal of pharmacology and experimental therapeutics (01.11.2004)
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Journal Article
Role of p38 MAP kinase in LPS‐induced airway inflammation in the rat
Haddad, El‐Bdaoui, Birrell, Mark, McCluskie, Kerryn, Ling, Andrea, Webber, Stephen E, Foster, Martyn L, Belvisi, Maria G
Published in British journal of pharmacology (01.04.2001)
Published in British journal of pharmacology (01.04.2001)
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Journal Article
Second-Generation Inhibitors Demonstrate the Involvement of p38 Mitogen-Activated Protein Kinase in Post-Transcriptional Modulation of Inflammatory Mediator Production in Human and Rodent Airways
Mark A. Birrell, Sissie Wong, Kerryn McCluskie, Matthew C. Catley, Elizabeth L. Hardaker, Saleem Haj-Yahia, Maria G. Belvisi
Published in The Journal of pharmacology and experimental therapeutics (01.03.2006)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2006)
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Journal Article
Differential Effects of Ebselen on Neutrophil Recruitment, Chemokine, and Inflammatory Mediator Expression in a Rat Model of Lipopolysaccharide-Induced Pulmonary Inflammation
Haddad, El-Bdaoui, McCluskie, Kerryn, Birrell, Mark A, Dabrowski, Dominika, Pecoraro, Michela, Underwood, Steve, Chen, Bei, De Sanctis, George T, Webber, Steve E, Foster, Martyn L, Belvisi, Maria G
Published in The Journal of immunology (1950) (15.07.2002)
Published in The Journal of immunology (1950) (15.07.2002)
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Journal Article
Characterization of the preclinical and clinical pharmacokinetics of GLM101, A liposome-encapsulated mannose-1-phosphate drug candidate for the treatment of patients with PMM2-CDG
Alaoui, Hicham, Moors, Tristen, McWilliams, Peter, Hird, Geoff, Shirakura, Teppei, McCluskie, Kerryn
Published in Molecular genetics and metabolism (01.04.2024)
Published in Molecular genetics and metabolism (01.04.2024)
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Journal Article
In vitro treatment with liposome-encapsulated Mannose-1-phosphate restores N-glycosylation in PMM2-CDG patient-derived fibroblasts
Shirakura, Teppei, Krishnamoorthy, Lakshmipriya, Paliwal, Preeti, Hird, Geoffrey, McCluskie, Kerryn, McWilliams, Peter, He, Miao, Ismaili, Moulay Hicham Alaoui
Published in Molecular genetics and metabolism (01.09.2024)
Published in Molecular genetics and metabolism (01.09.2024)
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Journal Article
Pharmacological Assessment of the Nitric-Oxide Synthase Isoform Involved in Eosinophilic Inflammation in a Rat Model of Sephadex-Induced Airway Inflammation
Birrell, Mark A, McCluskie, Kerryn, Haddad, El-Bdaoui, Battram, Cliff H, Webber, Stephen E, Foster, Martyn L, Yacoub, Magdi H, Belvisi, Maria G
Published in The Journal of pharmacology and experimental therapeutics (01.03.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2003)
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Journal Article
An orally administered enzyme therapeutic for homocystinuria that suppresses homocysteine by metabolizing methionine in the gastrointestinal tract
Skvorak, Kristen, Mitchell, Vesna, Teadt, Leann, Franklin, Kierra A., Lee, Hyung-Ok, Kruse, Nikki, Huitt-Roehl, Callie, Hang, Julie, Du, Faye, Galanie, Stephanie, Guan, Steven, Aijaz, Hera, Zhang, Nianliu, Rajkovic, Gabriel, Kruger, Warren D., Ismaili, Moulay Hicham Alaoui, Huisman, Gjalt, McCluskie, Kerryn, Silverman, Adam P.
Published in Molecular genetics and metabolism (01.08.2023)
Published in Molecular genetics and metabolism (01.08.2023)
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Journal Article
Oral enzyme therapy for maple syrup urine disease ( MSUD ) suppresses plasma leucine levels in intermediate MSUD mice and healthy nonhuman primates
Skvorak, Kristen, Liu, Joyce, Kruse, Nikki, Mehmood, Roasa, Das, Subhamoy, Jenne, Stephan, Chng, Chinping, Lao, U. Loi, Duan, Da, Asfaha, Jonathan, Du, Faye, Teadt, Leann, Sero, Antionette, Ching, Charlene, Riggins, James, Pope, Lianne, Yan, Ping, Mashiana, Harminder, Ismaili, Moulay Hicham Alaoui, McCluskie, Kerryn, Huisman, Gjalt, Silverman, Adam P.
Published in Journal of inherited metabolic disease (01.11.2023)
Published in Journal of inherited metabolic disease (01.11.2023)
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Journal Article
Engineering α-glucosidase to improve protein stability and cellular uptake for the potential treatment of Pompe disease
Botham, Rachel C., Hallows, William C., Reddy, Charu, Dellas, Nikki, Homan, David, Lao, Jessica, Zhu, Cynthia, Chng, Chinping, Sero, Antoinette, Miller, Matt, Choi, Su Jin, Sun, Baodong, McCluskie, Kerryn, Huisman, Gjalt, Silverman, Adam P.
Published in Molecular genetics and metabolism (01.02.2021)
Published in Molecular genetics and metabolism (01.02.2021)
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Journal Article
Engineering α-galactosidase A (GLA) to improve protein stability, efficacy and reduced immune response for the treatment of Fabry disease
Hallows, William Casey, Skvorak, Kristen, Zhu, Cynthia Yu, Sero, Antoinette, Botham, Rachel, Agard, Nicholas, Chng, Chinping, Dellas, Nikki, Miller, Matt, Shin, Jinsong, Viduya, Judy, Zhang, Xiyun, Schiffmann, Raphael, Huisman, Gjalt, McCluskie, Kerryn, Alaoui, Hicham
Published in Molecular genetics and metabolism (01.02.2020)
Published in Molecular genetics and metabolism (01.02.2020)
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Journal Article
Oral enzyme therapy for maple syrup urine disease (MSUD) suppresses plasma leucine levels in intermediate MSUD mice and healthy non-human primates
Skvorak, Kristen, Liu, Joyce, Kruse, Nikki, Mehmood, Roasa, Das, Subhamoy, Jenne, Stephan, Chng, Chinping, Lao, U Loi, Duan, Da, Asfaha, Jonathan, Du, Faye, Teadt, Leann, Sero, Antionette, Ching, Charlene, Riggins, James, Pope, Lianne, Yan, Ping, Mashiana, Harminder, Ismaili, Moulay Hicham Alaoui, McCluskie, Kerryn, Huisman, Gjalt, Silverman, Adam P
Published in Journal of inherited metabolic disease (26.07.2023)
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Published in Journal of inherited metabolic disease (26.07.2023)
Journal Article
IκB Kinase-2-Independent and -Dependent Inflammation in Airway Disease Models: Relevance of IKK-2 Inhibition to the Clinic
Birrell, Mark A., Wong, Sissie, Hardaker, Elizabeth L., Catley, Matthew C., McCluskie, Kerryn, Collins, Michael, Haj-Yahia, Saleem, Belvisi, Maria G.
Published in Molecular pharmacology (01.06.2006)
Published in Molecular pharmacology (01.06.2006)
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Journal Article
Iκ-B kinase-2 inhibitor blocks inflammation in human airway smooth muscle and a rat model of asthma
BIRRELL, Mark A, HARDAKER, Elizabeth, SHAW, Robert J, SAVAGE, Tony J, BELVISI, Maria G, WONG, Sissie, MCCLUSKIE, Kerryn, CATLEY, Matthew, DE ALBA, Jorge, NEWTON, Robert, HAJ-YAHIA, Saleem, TAO PUN, K, WATTS, Clarissa J
Published in American journal of respiratory and critical care medicine (15.10.2005)
Published in American journal of respiratory and critical care medicine (15.10.2005)
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