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Ewers, M, Buerger, K, Teipel, S J, Scheltens, P, Schröder, J, Zinkowski, R P, Bouwman, F H, Schönknecht, P, Schoonenboom, N S M, Andreasen, N, Wallin, A, DeBernardis, J F, Kerkman, D J, Heindl, B, Blennow, K, Hampel, H
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Published in Neurology (11.12.2007)
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Longitudinal CSF and MRI biomarkers improve the diagnosis of mild cognitive impairment
de Leon, M.J., DeSanti, S., Zinkowski, R., Mehta, P.D., Pratico, D., Segal, S., Rusinek, H., Li, J., Tsui, W., Saint Louis, L.A., Clark, C.M., Tarshish, C., Li, Y., Lair, L., Javier, E., Rich, K., Lesbre, P., Mosconi, L., Reisberg, B., Sadowski, M., DeBernadis, J.F., Kerkman, D.J., Hampel, H., Wahlund, L.-O., Davies, P.
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Published in Neurobiology of aging (01.03.2006)
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Discovery of a novel class of orally active, non-peptide angiotensin II antagonists
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Published in Journal of medicinal chemistry (01.10.1992)
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Preclinical pharmacological actions of (+/-)-(1'R,3R)-3-phenyl-1- [1',2',3',4'-tetrahydro-5',6'-methylene-dioxy-1'-naphthalenyl) methyl] pyrrolidine methanesulfonate (ABT-200), a potential antidepressant agent that antagonizes alpha-2 adrenergic receptors and inhibits the neuronal uptake of norepinephrine
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Published in The Journal of pharmacology and experimental therapeutics (01.03.1995)
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Published in The Journal of pharmacology and experimental therapeutics (01.03.1995)
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Characterization of antihypertensive activity of ABBOTT-81988, a nonpeptide angiotensin II antagonist in the renal hypertensive rat
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Published in The Journal of pharmacology and experimental therapeutics (01.01.1994)
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Published in The Journal of pharmacology and experimental therapeutics (01.01.1994)
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Antihypertensive activity of ABBOTT-81282, a nonpeptide angiotensin II antagonist, in the renal hypertensive rat
Lee, J Y, Brune, M E, Warner, R B, Buckner, S B, Winn, M, De, B, Zydowsky, T M, Opgenorth, T J, Kerkman, D J, DeBernardis, J F
Published in Pharmacology (01.09.1993)
Published in Pharmacology (01.09.1993)
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Cardiovascular effects of orally administered ABBOTT-81988, an angiotensin II antagonist, in conscious spontaneously hypertensive rats
Lee, J Y, Warner, R B, Brune, M E, Adler, A L, Winn, M, De, B, Zydowsky, T M, Opgenorth, T J, Kerkman, D J, DeBernardis, J F
Published in American journal of hypertension (01.11.1994)
Published in American journal of hypertension (01.11.1994)
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A-69024: a non-benzazepine antagonist with selectivity for the dopamine D-1 receptor
Kerkman, D J, Ackerman, M, Artman, L D, MacKenzie, R G, Johnson, M C, Bednarz, L, Montana, W, Asin, K E, Stampfli, H, Kebabian, J W
Published in European journal of pharmacology (03.08.1989)
Published in European journal of pharmacology (03.08.1989)
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A new nasal decongestant, A-57219: a comparison with oxymetazoline
DeBernardis, J F, Winn, M, Kerkman, D J, Kyncl, J J, Buckner, S, Horrom, B
Published in Journal of pharmacy and pharmacology (01.09.1987)
Published in Journal of pharmacy and pharmacology (01.09.1987)
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Adrenergic and dopaminergic properties of dopamine sulfoconjugates
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Published in Journal of cardiovascular pharmacology (01.11.1985)
Published in Journal of cardiovascular pharmacology (01.11.1985)
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Pharmacological characterization of abbott-81282, a novel, non-peptide angiotensin-II antagonist selective for type-1 receptors
Hancock, A.A., Buckner, S.A., Lee, J.Y., Brune, M., Morse, P.A., Oheim, K., Warner, R.B., Winn, M., Zydowsky, T.M., De, B., Kerkman, D.J., DeBernardis, J.F.
Published in Life sciences (1973) (1993)
Published in Life sciences (1973) (1993)
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Conformationally defined adrenergic agents. 4. 1-(Aminomethyl)phthalans: synthesis and pharmacological consequences of the phthalan ring oxygen atom
DeBernardis, John F, Arendsen, David L, Kyncl, John J, Kerkman, Daniel J
Published in Journal of medicinal chemistry (01.01.1987)
Published in Journal of medicinal chemistry (01.01.1987)
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Synthesis and in vitro evaluation of fused ring heterocycle-containing angiotensin II antagonists
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Published in Bioorganic & medicinal chemistry letters (06.01.1994)
Published in Bioorganic & medicinal chemistry letters (06.01.1994)
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Conformationally defined adrenergic agents. 1. Design and synthesis of novel alpha 2 selective adrenergic agents: electrostatic repulsion based conformational prototypes
DeBernardis, J F, Kerkman, D J, Winn, M, Bush, E N, Arendsen, D L, McClellan, W J, Kyncl, J J, Basha, F Z
Published in Journal of medicinal chemistry (01.10.1985)
Published in Journal of medicinal chemistry (01.10.1985)
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Conformationally defined adrenergic agents. 5. Resolution, absolute configuration, and pharmacological characterization of the enantiomers of 2-(5,6-dihydroxy-1,2,3,4-tetrahydro-1-naphthyl)imidazoline: a potent agonist at .alpha.-adrenoceptors
DeBernardis, John F, Kerkman, Daniel J, Arendsen, David L, Buckner, Steve A, Kyncl, John J, Hancock, Arthur A
Published in Journal of medicinal chemistry (01.06.1987)
Published in Journal of medicinal chemistry (01.06.1987)
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Conformationally defined adrenergic agents. 2. Catechol imidazoline derivatives: biological effects at alpha 1 and alpha 2 adrenergic receptors
DeBernardis, J F, Kyncl, J J, Basha, F Z, Arendsen, D L, Martin, Y C, Winn, M, Kerkman, D J
Published in Journal of medicinal chemistry (01.04.1986)
Published in Journal of medicinal chemistry (01.04.1986)
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[3H]A-81988, a potent, selective, competitive antagonist radioligand for angiotensin AT1 receptors
Hancock, A A, Surber, B W, Rotert, G, Thomas, S, Tasker, A S, Sorensen, B K, Vodenlich, A D, Opgenorth, T J, Kerkman, D J, DeBernardis, J F
Published in European journal of pharmacology (15.03.1994)
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Published in European journal of pharmacology (15.03.1994)
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Discovery of a novel class of orally active, non-peptide angiotensin II antogonists
DE, B, WINN, M, OPGENORTH, T, MARSH, K, ZYDOWSKY, T. M, KERKMAN, D. J, DEBERNARDIS, J. F, LEE, L, BUCKNER, S, WARNER, R, BRUNE, M, HANCOCK, A
Published in Journal of medicinal chemistry (1992)
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Published in Journal of medicinal chemistry (1992)
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Conformationally defined adrenergic agents. 3. Modifications to the carbocyclic ring of 5,6-dihydroxy-1-(2-imidazolinyl)tetralin: improved separation of alpha 1 and alpha 2 adrenergic activities
DeBernardis, J F, Winn, M, Arendsen, D L, Kerkman, D J, Kyncl, J J
Published in Journal of medicinal chemistry (01.08.1986)
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Published in Journal of medicinal chemistry (01.08.1986)
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