Homozygous MTAP deletion in primary human glioblastoma is not associated with elevation of methylthioadenosine
Barekatain, Yasaman, Ackroyd, Jeffrey J., Yan, Victoria C., Khadka, Sunada, Wang, Lin, Chen, Ko-Chien, Poral, Anton H., Tran, Theresa, Georgiou, Dimitra K., Arthur, Kenisha, Lin, Yu-Hsi, Satani, Nikunj, Ballato, Elliot S., Behr, Eliot I., deCarvalho, Ana C., Verhaak, Roel G. W., de Groot, John, Huse, Jason T., Asara, John M., Kalluri, Raghu, Muller, Florian L.
Published in Nature communications (09.07.2021)
Published in Nature communications (09.07.2021)
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Journal Article
An enolase inhibitor for the targeted treatment of ENO1-deleted cancers
Lin, Yu-Hsi, Satani, Nikunj, Hammoudi, Naima, Yan, Victoria C, Barekatain, Yasaman, Khadka, Sunada, Ackroyd, Jeffrey J, Georgiou, Dimitra K, Pham, Cong-Dat, Arthur, Kenisha, Maxwell, David, Peng, Zhenghong, Leonard, Paul G, Czako, Barbara, Pisaneschi, Federica, Mandal, Pijus, Sun, Yuting, Zielinski, Rafal, Pando, Susana Castro, Wang, Xiaobo, Tran, Theresa, Xu, Quanyu, Wu, Qi, Jiang, Yongying, Kang, Zhijun, Asara, John M, Priebe, Waldemar, Bornmann, William, Marszalek, Joseph R, DePinho, Ronald A, Muller, Florian L
Published in Nature metabolism (01.12.2020)
Published in Nature metabolism (01.12.2020)
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Journal Article
Impaired anaplerosis is a major contributor to glycolysis inhibitor toxicity in glioma
Khadka, Sunada, Arthur, Kenisha, Barekatain, Yasaman, Behr, Eliot, Washington, Mykia, Ackroyd, Jeffrey, Crowley, Kaitlyn, Suriyamongkol, Pornpa, Lin, Yu-Hsi, Pham, Cong-Dat, Zielinski, Rafal, Trujillo, Marissa, Galligan, James, Georgiou, Dimitra K, Asara, John, Muller, Florian
Published in Cancer & metabolism (25.06.2021)
Published in Cancer & metabolism (25.06.2021)
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Journal Article
Robust detection of oncometabolic aberrations by 1H–13C heteronuclear single quantum correlation in intact biological specimens
Barekatain, Yasaman, Yan, Victoria C., Arthur, Kenisha, Ackroyd, Jeffrey J., Khadka, Sunada, De Groot, John, Huse, Jason T., Muller, Florian L.
Published in Communications biology (25.06.2020)
Published in Communications biology (25.06.2020)
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Journal Article
Prodrugs of a 1‑Hydroxy-2-oxopiperidin-3-yl Phosphonate Enolase Inhibitor for the Treatment of ENO1-Deleted Cancers
Yan, Victoria C., Pham, Cong-Dat, Ballato, Elliot S., Yang, Kristine L., Arthur, Kenisha, Khadka, Sunada, Barekatain, Yasaman, Shrestha, Prakriti, Tran, Theresa, Poral, Anton H., Washington, Mykia, Raghavan, Sudhir, Czako, Barbara, Pisaneschi, Federica, Lin, Yu-Hsi, Satani, Nikunj, Hammoudi, Naima, Ackroyd, Jeffrey J., Georgiou, Dimitra K., Millward, Steven W., Muller, Florian L.
Published in Journal of medicinal chemistry (27.10.2022)
Published in Journal of medicinal chemistry (27.10.2022)
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Journal Article
Aliphatic amines are viable pro-drug moieties in phosphonoamidate drugs
Yan, Victoria C., Pham, Cong-Dat, Arthur, Kenisha, Yang, Kristine L., Muller, Florian L.
Published in Bioorganic & medicinal chemistry letters (15.12.2020)
Published in Bioorganic & medicinal chemistry letters (15.12.2020)
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Journal Article
Abstract 984: Synthesis of mixed, hypoxia-activated phosphoramidate esters for the inhibition of Enolase in ENO1- deleted glioblastoma
Muller, Florian, Yan, Victoria C., Ballato, Elliot S., Yang, Kristine L., Georgiou, Dimitra K., Arthur, Kenisha, Shrestha, Pakriti, Khadka, Sunada, Ackroyd, Jeffrey
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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Journal Article
TAMI-62. ANGIOGENESIS INHIBITORS STRONGLY SYNERGIZE WITH THERAPEUTICS TARGETING TUMOR METABOLISM
Khadka, Sunada, Lin, Yu-Hsi, Ackroyd, Jeffrey, Arthur, Kenisha, Barekatain, Yasaman, Poral, Anton, Tran, Theresa, Georgiou, Dimitra, de Groot, John, Huse, Jason, Asara, John, Muller, Florian
Published in Neuro-oncology (Charlottesville, Va.) (09.11.2020)
Published in Neuro-oncology (Charlottesville, Va.) (09.11.2020)
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Journal Article
Abstract 3208: Angiogenesis inhibitors strongly synergize with therapeutics targeting tumor metabolism
Khadka, Sunada, Lin, Yu-Hsi, Ackroyd, Jeffery, Arthur, Kenisha, Barekatain, Yasaman, Poral, Anton, Tran, Theresa, Behr, Eliot, Chen, Yining, Georgiou, Dimitra, Depinho, Ronald, Muller, Florian
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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Journal Article
Comparative Pharmacology of a Bis-Pivaloyloxymethyl Phosphonate Prodrug Inhibitor of Enolase after Oral and Parenteral Administration
Yan, Victoria C., Barekatain, Yasaman, Lin, Yu-Hsi, Satani, Nikunj, Hammoudi, Naima, Arthur, Kenisha, Georgiou, Dimitra K., Jiang, Yongying, Sun, Yuting, Marszalek, Joseph R., Millward, Steven W., Muller, Florian L.
Published in ACS pharmacology & translational science (10.02.2023)
Published in ACS pharmacology & translational science (10.02.2023)
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Journal Article
Bioreducible Phosphonoamidate Pro-drug Inhibitor of Enolase: Proof of Concept Study
Yan, Victoria C, Yang, Kristine L, Ballato, Elliot S, Khadka, Sunada, Shrestha, Prakriti, Arthur, Kenisha, Georgiou, Dimitra K, Washington, Mykia, Tran, Theresa, Poral, Anton H, Pham, Cong-Dat, Yan, Matthew J, Muller, Florian L
Published in ACS medicinal chemistry letters (09.07.2020)
Published in ACS medicinal chemistry letters (09.07.2020)
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Journal Article
Robust detection of oncometabolic aberrations by 1 H- 13 C heteronuclear single quantum correlation in intact biological specimens
Barekatain, Yasaman, Yan, Victoria C, Arthur, Kenisha, Ackroyd, Jeffrey J, Khadka, Sunada, De Groot, John, Huse, Jason T, Muller, Florian L
Published in Communications biology (25.06.2020)
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Published in Communications biology (25.06.2020)
Journal Article
Author Correction: An enolase inhibitor for the targeted treatment of ENO1-deleted cancers
Lin, Yu-Hsi, Satani, Nikunj, Hammoudi, Naima, Yan, Victoria C, Barekatain, Yasaman, Khadka, Sunada, Ackroyd, Jeffrey J, Georgiou, Dimitra K, Pham, Cong-Dat, Arthur, Kenisha, Maxwell, David, Peng, Zhenghong, Leonard, Paul G, Czako, Barbara, Pisaneschi, Federica, Mandal, Pijus, Sun, Yuting, Zielinski, Rafal, Pando, Susana Castro, Wang, Xiaobo, Tran, Theresa, Xu, Quanyu, Wu, Qi, Jiang, Yongying, Kang, Zhijun, Asara, John M, Priebe, Waldemar, Bornmann, William, Marszalek, Joseph R, DePinho, Ronald A, Muller, Florian L
Published in Nature metabolism (2021)
Published in Nature metabolism (2021)
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Journal Article
Anaplerotic nutrient stress drives synergy of angiogenesis inhibitors with therapeutics targeting tumor metabolism
Khadka, Sunada, Lin, Yu-Hsi, Ackroyd, Jeffrey, Chen, Yi-An, Sheng, Yanghui, Qian, Wubin, Guo, Sheng, Chen, Yining, Behr, Eliot, Barekatain, Yasaman, Uddin, Nasir, Arthur, Kenisha, Yan, Victoria, Hsu, Wen-Hao, Chang, Qing, Poral, Anton, Tran, Theresa, Chaurasia, Surendra, Georgiou, Dimitra K, Asara, John M, Barthel, Floris P, Millward, Steve W, DePinho, Ronald A, Muller, Florian L
Published in bioRxiv (19.10.2023)
Published in bioRxiv (19.10.2023)
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Journal Article
Robust detection of oncometabolic aberrations by 1H-13C heteronuclear single quantum correlation in live cells and intact tumors ex-vivo
Barekatain, Yasaman, Yan, Victoria C, Kenisha Arthur, Ackroyd, Jeffrey J, Sunada Khadka, De Groot, John, Huse, Jason T, Muller, Florian L
Published in bioRxiv (19.12.2019)
Published in bioRxiv (19.12.2019)
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Paper
Methylthioadenosine is Not Dramatically Elevated in MTAP-Homozygous Deleted Primary Glioblastomas
Barekatain, Yasaman, Yan, Victoria C, Ackroyd, Jeffrey J, Poral, Anton H, Tran, Theresa, Georgiou, Dimitra K, Kenisha Arthur, Yu-Hsi, Lin, Satani, Nikunj, Ballato, Elliot S, Decarvalho, Ana, Verhaak, Roel, De Groot, John, Huse, Jason T, Asara, John M, Muller, Florian L
Published in bioRxiv (18.10.2019)
Published in bioRxiv (18.10.2019)
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