Cyclocondensation of o -phenylenediamines with α-ketothioesters: a novel approach for the synthesis of 2-acylbenzimidazoles
Kavya, Kumar, Honnabandar, Kanaka Vijayashankar, Sridhar, Bilagumba T., Swaroop, Toreshettahally R., Shivakumar, Anantharaman, Mantelingu, Kempegowda
Published in New journal of chemistry (21.10.2024)
Published in New journal of chemistry (21.10.2024)
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Journal Article
Identification and characterization of mercaptopyrimidine‐based small molecules as inhibitors of nonhomologous DNA end joining
Ray, Ujjayinee, Gopinatha, Vindya K., Sharma, Shivangi, Goyary, Laijau, Choudhary, Bibha, Mantelingu, Kempegowda, Rangappa, Kanchugarakoppal S., Raghavan, Sathees C.
Published in The FEBS journal (01.02.2023)
Published in The FEBS journal (01.02.2023)
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Journal Article
A panoramic view on synthetic applications of α-oxothioamides: a highly regioselective synthesis of 2-acyl-4-(het)arylthiazoles and thioethers
Suresh, Rajaghatta N, Swaroop, Toreshettahally R, Gowda, Darshini, Mantelingu, Kempegowda, Rangappa, Kanchugarakoppal S
Published in RSC advances (06.02.2023)
Published in RSC advances (06.02.2023)
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Journal Article
Identification and characterization of novel SCR7‐based small‐molecule inhibitor of DNA end‐joining, SCR130 and its relevance in cancer therapeutics
Ray, Ujjayinee, Raul, Sanjay Kumar, Gopinatha, Vindya K., Ghosh, Dipayan, Rangappa, Kanchugarakoppal S., Mantelingu, Kempegowda, Raghavan, Sathees C.
Published in Molecular carcinogenesis (01.06.2020)
Published in Molecular carcinogenesis (01.06.2020)
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Journal Article
An expedient, efficient and solvent-free synthesis of T3P®-mediated amidation of benzhydrols with poorly reactive N-nucleophiles under MW irradiation
Cheruku, Srinivas, Nagarakere, Sandhya C., Sunilkumar, Makanahalli P., Narayana, Yatheesh, Manikyanally, Kumara N., Rangappa, Kanchugarakoppal S., Mantelingu, Kempegowda
Published in New journal of chemistry (28.02.2022)
Published in New journal of chemistry (28.02.2022)
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Journal Article
Acute toxicity analysis of Disarib, an inhibitor of BCL2
Sharma, Shivangi, Varsha, Kontham Kulangara, Kumari, Susmita, Gopalakrishnan, Vidya, Jose, Anjana Elizabeth, Choudhary, Bibha, Mantelingu, Kempegowda, Raghavan, Sathees C.
Published in Scientific reports (16.09.2020)
Published in Scientific reports (16.09.2020)
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Journal Article
Autocyclized and oxidized forms of SCR7 induce cancer cell death by inhibiting nonhomologous DNA end joining in a Ligase IV dependent manner
Vartak, Supriya V., Swarup, Hassan A., Gopalakrishnan, Vidya, Gopinatha, Vindya K., Ropars, Virginie, Nambiar, Mridula, John, Franklin, Kothanahally, Sharath Kumar S., Kumari, Rupa, Kumari, Nitu, Ray, Ujjayinee, Radha, Gudapureddy, Dinesh, Depina, Pandey, Monica, Ananda, Hanumappa, Karki, Subhas S., Srivastava, Mrinal, Charbonnier, Jean Baptiste, Choudhary, Bibha, Mantelingu, Kempegowda, Raghavan, Sathees C.
Published in The FEBS journal (01.11.2018)
Published in The FEBS journal (01.11.2018)
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Journal Article
Innovative approach for the synthesis of N-substituted amides from nitriles and alcohols using propylphosphonic anhydride (T3P®) under solvent-free conditions
Swarup, Hassan A., Chaithra, Nagaraju, Sandhya, Nagarakere C., Rangappa, Shobith, Mantelingu, Kempegowda, Rangappa, Kanchugarakoppal S.
Published in Synthetic communications (18.08.2019)
Published in Synthetic communications (18.08.2019)
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Journal Article
Electrochemical Synthesis of 3,5-Bis(acyl)-1,2,4-thiadiazoles through n-Bu4NI-mediated Oxidative Dimerization of α-Oxothioamides
SHIVARAJ, Mahadev, SURESH, Rajaghatta N, SWAROOP, Toreshettahally R, KUMARA, Manikyanahally N, RANGAPPA, Kanchugarakoppal S, MANTELINGU, Kempegowda, DEVI, Adaganahalli Boregowda MAMATHA, MANASA, Madihalli Prasanna, UMASHANKARA, Muddegowda
Published in Denki kagaku oyobi kōgyō butsuri kagaku (28.12.2023)
Published in Denki kagaku oyobi kōgyō butsuri kagaku (28.12.2023)
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Journal Article
Synthesis and biological evaluation of theophylline acetohydrazide hydrazone derivatives as antituberculosis agents
Gopinatha, Vindya K., Dukanya, Mantelingu, Kempegowda, Rangappa, Kanchugarakoppal S.
Published in Journal of the Chinese Chemical Society (Taipei) (01.08.2020)
Published in Journal of the Chinese Chemical Society (Taipei) (01.08.2020)
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Journal Article
A new triazolyl‐indolo‐quinoxaline induces apoptosis in gastric cancer cells by abrogating the STAT3/5 pathway through upregulation of PTPεC
Suresh, Rajaghatta N., Jung, Young Y., Mohan, Chakrabhavi D., Gowda, Shalini V., Harsha, Kachigere B., Mantelingu, Kempegowda, Sethi, Gautam, Ahn, Kwang S., Rangappa, Kanchugarakoppal S.
Published in Drug development research (01.12.2023)
Published in Drug development research (01.12.2023)
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Journal Article
I2-Catalyzed transformation of o-aminobenzamide to o-ureidobenzonitrile using isothiocyanates
Sadashivamurthy Shamanth, Nagaraju Chaithra, Gurukiran, Mahesha, Mahesha Mamatha, Lokanath, N K, Rangappa, Kanchugarakoppal S, Kempegowda Mantelingu
Published in Organic & biomolecular chemistry (14.04.2020)
Published in Organic & biomolecular chemistry (14.04.2020)
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Journal Article
One-pot tandem approach for the synthesis of benzimidazoles and benzothiazoles from alcohols
Raghavendra, Goravanahalli M., Ramesha, Ajjahalli B., Revanna, Cigalli N., Nandeesh, Kebbahalli N., Mantelingu, Kempegowda, Rangappa, Kanchugarakoppal S.
Published in Tetrahedron letters (26.10.2011)
Published in Tetrahedron letters (26.10.2011)
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Journal Article
A novel and facile synthesis of 3,5-Disubstituted isothiozoles under metal free conditions using acetophenones and dithioesters
Nagaraju, Chaithra, Ashok, Swarup Hassan, Shamanth, Sadashivamurthy, Nagarakere, Sandhya C., Sunilkumar, Makanahalli P., Subbegowda, Rangappa Kanchugarakoppal, Mantelingu, Kempegowda
Published in Synthetic communications (01.09.2020)
Published in Synthetic communications (01.09.2020)
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Journal Article
Novel Approach for the Synthesis of 2, 5-disubstituted 1, 3, 4-thiadiazoles from Benzothiohydrazides and Ethylbenzimidate
Shobha, S., Kemparajegowda, Girimanchanaika, Swamy Savvemala A., Swarup, Hassan, Mantelingu, Kempegowda
Published in Letters in organic chemistry (01.01.2023)
Published in Letters in organic chemistry (01.01.2023)
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Journal Article
Differential effects of garcinol and curcumin on histone and p53 modifications in tumour cells
Collins, Hilary M, Abdelghany, Magdy K, Messmer, Marie, Yue, Baigong, Deeves, Sian E, Kindle, Karin B, Mantelingu, Kempegowda, Aslam, Akhmed, Winkler, G Sebastiaan, Kundu, Tapas K, Heery, David M
Published in BMC cancer (29.01.2013)
Published in BMC cancer (29.01.2013)
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Journal Article
Microwave-Assisted, Metal-Free, Chemoselective N-Formylation of Amines using 2-Formyl-1,3-dimethyl-1H-imidazol-3-ium Iodide and In Situ Synthesis of Benzimidazole and Isocyanides
Jagadeesha, Gullahalli S., Mantelingu, Kempegowda, Thimmegowda, Naraganahalli R., Rangappa, Kanchugarakoppal S.
Published in SynOpen (2017) (01.06.2022)
Published in SynOpen (2017) (01.06.2022)
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Journal Article
Microwave-Assisted, Metal-Free, Chemoselective N-Formylation of Amines using 2-Formyl-1,3-dimethyl-1H-imidazol-3-ium Iodide and In Situ Synthesis of Benzimidazole and Isocyanides
Jagadeesha, Gullahalli S., Mantelingu, Kempegowda, Thimmegowda, Naraganahalli R., Rangappa, Kanchugarakoppal S.
Published in SynOpen (2017) (01.06.2022)
Published in SynOpen (2017) (01.06.2022)
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Journal Article