Factor Xa Inhibitors: S1 Binding Interactions of a Series of N-{(3S)-1-[(1S)-1-Methyl-2-morpholin-4-yl-2-oxoethyl]-2-oxopyrrolidin-3-yl}sulfonamides
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Published in Journal of medicinal chemistry (05.04.2007)
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Reflection in a workplace qualification: challenges and benefits
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Structure- and property-based design of factor Xa inhibitors: Pyrrolidin-2-ones with acyclic alanyl amides as P4 motifs
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Published in Bioorganic & medicinal chemistry letters (01.12.2006)
Published in Bioorganic & medicinal chemistry letters (01.12.2006)
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Structure and property based design of factor Xa inhibitors: Pyrrolidin-2-ones with biaryl P4 motifs
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Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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Structure and property based design of factor Xa inhibitors: Biaryl pyrrolidin-2-ones incorporating basic heterocyclic motifs
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Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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Selective and dual action orally active inhibitors of thrombin and factor Xa
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Published in Bioorganic & medicinal chemistry letters (15.05.2007)
Published in Bioorganic & medicinal chemistry letters (15.05.2007)
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Design and synthesis of orally active pyrrolidin-2-one-based factor Xa inhibitors
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Pass, Martin, Abu-Rabie, Said, Baxter, Andrew, Conroy, Richard, Coote, Steven J, Craven, Andrew P, Finch, Harry, Hindley, Seán, Kelly, Henry A, Lowdon, Andrew W, McDonald, Edward, Mitchell, William L, Pegg, Neil A, Procopiou, Pan A, Ramsden, Nigel G, Thomas, Rhian, Walker, Dawn A, Watson, Nigel S, Jhoti, Harren, Mooney, Christopher J, Tang, Chi-Man, Thomas, Pamela J, Parry, Simon, Patel, Champa
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Eldred, Colin D., Evans, Brian, Hindley, Sean, Judkins, Brian D., Kelly, Henry A., Kitchin, John, Lumley, Philip, Porter, Barry, Ross, Barry C.
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Pyrrolizidine alkaloid biosynthesis. Synthesis of N-([4-14C]-4-aminobutyl)-1,2-didehydropyrrolidinium and its incorporation into different pyrrolizidine bases (necines)
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Evolution of a Novel Series of [(N,N-Dimethylamino)propyl]- and Piperazinylbenzanilides as the First Selective 5-HT1D Antagonists
Clitherow, John W, Scopes, David I. C, Skingle, Malcolm, Jordan, Christopher C, Feniuk, Wasyl, Campbell, Ian B, Carter, Malcolm C, Collington, Eric W, Connor, Helen E
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Published in Journal of medicinal chemistry (01.07.1994)
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Published in Form: pioneering design (01.05.2014)
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Published in Form: pioneering design (01.05.2014)
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