Enantioselective Synthesis of 4′-Ethynyl-2-fluoro-2′-deoxyadenosine (EFdA) via Enzymatic Desymmetrization
McLaughlin, Mark, Kong, Jongrock, Belyk, Kevin M, Chen, Billy, Gibson, Andrew W, Keen, Stephen P, Lieberman, David R, Milczek, Erika M, Moore, Jeffrey C, Murray, David, Peng, Feng, Qi, Ji, Reamer, Robert A, Song, Zhiguo J, Tan, Lushi, Wang, Lin, Williams, Michael J
Published in Organic letters (17.02.2017)
Published in Organic letters (17.02.2017)
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Enantioselective Synthesis of β‑Aryloxycarboxylic Esters via Asymmetric Hydrogenation of β‑Aryloxy-α,β-Unsaturated Esters
Stewart, Gavin W, Shevlin, Michael, Yamagata, Adam D. Gammack, Gibson, Andrew W, Keen, Stephen P, Scott, Jeremy P
Published in Organic letters (02.11.2012)
Published in Organic letters (02.11.2012)
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Process Development of the HCV NS5B Site D Inhibitor MK-8876
Williams, Michael J, Chen, Qinghao, Codan, Lorenzo, Dermenjian, Renee K, Dreher, Spencer, Gibson, Andrew W, He, Xianliang, Jin, Yan, Keen, Stephen P, Lee, Alfred Y, Lieberman, David R, Lin, Wei, Liu, Guiquan, McLaughlin, Mark, Reibarkh, Mikhail, Scott, Jeremy P, Strickfuss, Sophie, Tan, Lushi, Varsolona, Richard J, Wen, Feng
Published in Organic process research & development (15.07.2016)
Published in Organic process research & development (15.07.2016)
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Development of a Fit-for-Purpose Large-Scale Synthesis of an Oral PARP Inhibitor
Wallace, Debra J, Baxter, Carl A, Brands, Karel J. M, Bremeyer, Nadine, Brewer, Sarah E, Desmond, Richard, Emerson, Khateeta M, Foley, Jennifer, Fernandez, Paul, Hu, Weifeng, Keen, Stephen P, Mullens, Peter, Muzzio, Daniel, Sajonz, Peter, Tan, Lushi, Wilson, Robert D, Zhou, George, Zhou, Guoyue
Published in Organic process research & development (15.07.2011)
Published in Organic process research & development (15.07.2011)
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Process Development and Large-Scale Synthesis of a c-Met Kinase Inhibitor
Stewart, Gavin W, Brands, Karel M. J, Brewer, Sarah E, Cowden, Cameron J, Davies, Antony J, Edwards, John S, Gibson, Andrew W, Hamilton, Simon E, Katz, Jason D, Keen, Stephen P, Mullens, Peter R, Scott, Jeremy P, Wallace, Debra J, Wise, Christopher S
Published in Organic process research & development (16.07.2010)
Published in Organic process research & development (16.07.2010)
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Practical Asymmetric Synthesis of a γ-Secretase Inhibitor Exploiting Substrate-Controlled Intramolecular Nitrile Oxide−Olefin Cycloaddition
Scott, Jeremy P, Oliver, Steven F, Brands, Karel M. J, Brewer, Sarah E, Davies, Antony J, Gibb, Andrew D, Hands, David, Keen, Stephen P, Sheen, Faye J, Reamer, Robert A, Wilson, Robert D, Dolling, Ulf-H
Published in Journal of organic chemistry (14.04.2006)
Published in Journal of organic chemistry (14.04.2006)
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Stereoselective Total Syntheses and Reassignment of Stereochemistry of the Freshwater Cyanobacterial Hepatotoxins Cylindrospermopsin and 7-Epicylindrospermopsin
Heintzelman, Geoffrey R, Fang, Wen-Kui, Keen, Stephen P, Wallace, Grier A, Weinreb, Steven M
Published in Journal of the American Chemical Society (17.04.2002)
Published in Journal of the American Chemical Society (17.04.2002)
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Stereoselective Total Synthesis of the Cyanobacterial Hepatotoxin 7-Epicylindrospermopsin: Revision of the Stereochemistry of Cylindrospermopsin
Heintzelman, Geoffrey R, Fang, Wen-Kui, Keen, Stephen P, Wallace, Grier A, Weinreb, Steven M
Published in Journal of the American Chemical Society (12.09.2001)
Published in Journal of the American Chemical Society (12.09.2001)
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Practical Asymmetric Synthesis of a Non-Peptidic αvβ3 Antagonist
Keen, Stephen P, Cowden, Cameron J, Bishop, Brian C, Brands, Karel M. J, Davies, Antony J, Dolling, Ulf H, Lieberman, David R, Stewart, Gavin W
Published in Journal of organic chemistry (04.03.2005)
Published in Journal of organic chemistry (04.03.2005)
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Process Development of a Tricyclic Diazepine-Based IDH1 Mutant Inhibitor
Maddess, Matthew L., Cleator, Ed, Morimoto, Mariko, Goodyear, Adrian, Dieguez-Vazquez, Alejandro, Gibb, Andrew, Kirtley, Andy, Christensen, Melodie, Song, Chaohui, Peng, Feng, Alam, Mahbub, Keen, Stephen P., Oliver, Steven F.
Published in Organic process research & development (21.06.2024)
Published in Organic process research & development (21.06.2024)
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Practical Asymmetric Synthesis of a Non-Peptidic α v β 3 Antagonist
Keen, Stephen P., Cowden, Cameron J., Bishop, Brian C., Brands, Karel M. J., Davies, Antony J., Dolling, Ulf H., Lieberman, David R., Stewart, Gavin W.
Published in Journal of organic chemistry (04.03.2005)
Published in Journal of organic chemistry (04.03.2005)
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Cross-metathesis of unsaturated alpha-amino acid derivatives
Biagini, SCG, Gibson, SE, Keen, SP
Published in Journal of the Chemical Society, Perkin Transactions 1 (21.08.1998)
Published in Journal of the Chemical Society, Perkin Transactions 1 (21.08.1998)
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ChemInform Abstract: Enantioselective Synthesis of [beta]-Aryloxycarboxylic Esters via Asymmetric Hydrogenation of [beta]-Aryloxy-[alpha],[beta]-unsaturated Esters
Stewart, Gavin W, Shevlin, Michael, Yamagata, Adam D. Gammack, Gibson, Andrew W, Keen, Stephen P, Scott, Jeremy P
Published in ChemInform (12.03.2013)
Published in ChemInform (12.03.2013)
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ChemInform Abstract: Enantioselective Synthesis of β-Aryloxycarboxylic Esters via Asymmetric Hydrogenation of β-Aryloxy-α,β-unsaturated Esters
Stewart, Gavin W., Shevlin, Michael, Yamagata, Adam D. Gammack, Gibson, Andrew W., Keen, Stephen P., Scott, Jeremy P.
Published in ChemInform (12.03.2013)
Published in ChemInform (12.03.2013)
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