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Synthetic Method for 2′-Amino-LNA Bearing Any of the Four Nucleobases via a Transglycosylation Reaction
Sawamoto, Hiroaki, Arai, Yuuki, Yamakoshi, Shuhei, Obika, Satoshi, Kawanishi, Eiji
Published in Organic letters (06.04.2018)
Published in Organic letters (06.04.2018)
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Discovery of Chlorofluoroacetamide-Based Covalent Inhibitors for Severe Acute Respiratory Syndrome Coronavirus 2 3CL Protease
Hirose, Yuya, Shindo, Naoya, Mori, Makiko, Onitsuka, Satsuki, Isogai, Hikaru, Hamada, Rui, Hiramoto, Tadanari, Ochi, Jinta, Takahashi, Daisuke, Ueda, Tadashi, Caaveiro, Jose M. M., Yoshida, Yuya, Ohdo, Shigehiro, Matsunaga, Naoya, Toba, Shinsuke, Sasaki, Michihito, Orba, Yasuko, Sawa, Hirofumi, Sato, Akihiko, Kawanishi, Eiji, Ojida, Akio
Published in Journal of medicinal chemistry (27.10.2022)
Published in Journal of medicinal chemistry (27.10.2022)
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Inhibition of dynamin‐related protein 1‐filamin interaction improves systemic glucose metabolism
Kato, Yuri, Ariyoshi, Kohei, Nohara, Yasunobu, Matsunaga, Naoya, Shimauchi, Tsukasa, Shindo, Naoya, Nishimura, Akiyuki, Mi, Xinya, Kim, Sang Geon, Ide, Tomomi, Kawanishi, Eiji, Ojida, Akio, Nakashima, Naoki, Mori, Yasuo, Nishida, Motohiro
Published in British journal of pharmacology (01.11.2024)
Published in British journal of pharmacology (01.11.2024)
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Synthesis and properties of GuNA purine/pyrimidine nucleosides and oligonucleotides
Kumagai, Shinji, Sawamoto, Hiroaki, Takegawa-Araki, Tomo, Arai, Yuuki, Yamakoshi, Shuhei, Yamada, Katsuya, Ohta, Tetsuya, Kawanishi, Eiji, Horie, Naohiro, Yamaguchi, Takao, Obika, Satoshi
Published in Organic & biomolecular chemistry (07.12.2020)
Published in Organic & biomolecular chemistry (07.12.2020)
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Synthesis and Biological Evaluation of Thiophene-C-glucosides as Sodium-Dependent Glucose Cotransporter 2 Inhibitors
Sakamaki, Shigeki, Kawanishi, Eiji, Koga, Yuichi, Yamamoto, Yasuo, Kuriyama, Chiaki, Matsushita, Yasuaki, Ueta, Kiichiro, Nomura, Sumihiro
Published in Chemical & pharmaceutical bulletin (01.10.2013)
Published in Chemical & pharmaceutical bulletin (01.10.2013)
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Scalable Process Design for a PDE10A Inhibitor Consisting of Pyrazolopyrimidine and Quinoxaline as Key Units
Yamagami, Takafumi, Kobayashi, Ryo, Moriyama, Noriaki, Horiuchi, Hideki, Toyofuku, Eiji, Kadoh, Yoichi, Kawanishi, Eiji, Izumoto, Shinichi, Hiramatsu, Hajime, Nanjo, Takehiro, Sugino, Masuhiro, Utsugi, Masayuki, Moritani, Yasunori
Published in Organic Process Research & Development (19.04.2019)
Published in Organic Process Research & Development (19.04.2019)
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Discovery of 2-[(E)-2-(7-Fluoro-3-methylquinoxalin-2-yl)vinyl]-6-pyrrolidin-1-yl-N-(tetrahydro-2H-pyran-4-yl)pyrimidin-4-amine Hydrochloride as a Highly Selective PDE10A Inhibitor
Kadoh, Yoichi, Miyoshi, Haruko, Matsumura, Takehiko, Tanaka, Yoshihito, Hongu, Mitsuya, Kimura, Mayumi, Takedomi, Kei, Omori, Kenji, Kotera, Jun, Sasaki, Takashi, Kobayashi, Tamaki, Taniguchi, Hiroyuki, Watanabe, Yumi, Kojima, Koki, Sakamoto, Toshiaki, Himiyama, Toshiyuki, Kawanishi, Eiji
Published in Chemical & pharmaceutical bulletin (2018)
Published in Chemical & pharmaceutical bulletin (2018)
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Radiosynthesis and in vivo evaluation of [ 11C]MP-10 as a positron emission tomography radioligand for phosphodiesterase 10A
Plisson, Christophe, Salinas, Cristian, Weinzimmer, David, Labaree, David, Lin, Shu-Fei, Ding, Yu-Shin, Jakobsen, Steen, Smith, Paul W., Eiji, Kawanishi, Carson, Richard E., Gunn, Roger N., Rabiner, Eugenii A.
Published in Nuclear medicine and biology (01.08.2011)
Published in Nuclear medicine and biology (01.08.2011)
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Phosphodiesterase 10A PET Radioligand Development Program: From Pig to Human
Plisson, Christophe, Weinzimmer, David, Jakobsen, Steen, Natesan, Sridhar, Salinas, Cristian, Lin, Shu-Fei, Labaree, David, Zheng, Ming-Qiang, Nabulsi, Nabeel, Marques, Tiago Reis, Kapur, Shitij, Kawanishi, Eiji, Saijo, Takeaki, Gunn, Roger N., Carson, Richard E., Rabiner, Eugenii A.
Published in Journal of Nuclear Medicine (01.04.2014)
Published in Journal of Nuclear Medicine (01.04.2014)
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Selective covalent targeting of SARS-CoV-2 main protease by enantiopure chlorofluoroacetamide
Yamane, Daiki, Onitsuka, Satsuki, Re, Suyong, Isogai, Hikaru, Hamada, Rui, Hiramoto, Tadanari, Kawanishi, Eiji, Mizuguchi, Kenji, Shindo, Naoya, Ojida, Akio
Published in Chemical science (Cambridge) (09.03.2022)
Published in Chemical science (Cambridge) (09.03.2022)
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Discovery of Canagliflozin, a Novel C-Glucoside with Thiophene Ring, as Sodium-Dependent Glucose Cotransporter 2 Inhibitor for the Treatment of Type 2 Diabetes Mellitus
Nomura, Sumihiro, Sakamaki, Shigeki, Hongu, Mitsuya, Kawanishi, Eiji, Koga, Yuichi, Sakamoto, Toshiaki, Yamamoto, Yasuo, Ueta, Kiichiro, Kimata, Hirotaka, Nakayama, Keiko, Tsuda-Tsukimoto, Minoru
Published in Journal of medicinal chemistry (09.09.2010)
Published in Journal of medicinal chemistry (09.09.2010)
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Discovery of Chlorofluoroacetamide-Based Covalent Inhibitors for SARS-CoV-2 3CL Protease
Hirose, Yuya, Shindo, Naoya, Mori, Makiko, Onitsuka, Satsuki, Isogai, Hikaru, Hamada, Rui, Hiramoto, Tadanari, Ochi, Jinta, Takahashi, Daisuke, Ueda, Tadashi, Caaveiro, Jose M.M., Yoshida, Yuya, Ohdo, Shigehiro, Matsunaga, Naoya, Toba, Shinsuke, Sasaki, Michihito, Orba, Yasuko, Sawa, Hirofumi, Sato, Akihiko, Kawanishi, Eiji, Ojida, Akio
Published in bioRxiv (06.06.2022)
Published in bioRxiv (06.06.2022)
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