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Published in Journal of medicinal chemistry (06.05.2004)
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Identification of a dual δ OR antagonist/μ OR agonist as a potential therapeutic for diarrhea-predominant Irritable Bowel Syndrome (IBS-d)
Breslin, Henry J., Diamond, Craig J., Kavash, Robert W., Cai, Chaozhong, Dyatkin, Alexey B., Miskowski, Tamara A., Zhang, Sui-Po, Wade, Paul R., Hornby, Pamela J., He, Wei
Published in Bioorganic & medicinal chemistry letters (15.07.2012)
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De Novo Design of Self-Assembling Foldamers That Inhibit Heparin–Protein Interactions
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Evolution of anti-HIV drug candidates. Part 3: diarylpyrimidine (DAPY) analogues
Ludovici, Donald W., De Corte, Bart L., Kukla, Michael J., Ye, Hong, Ho, Chih Y., Lichtenstein, Mark A., Kavash, Robert W., Andries, Koen, de Béthune, Marie-Pierre, Azijn, Hilde, Pauwels, Rudi, Lewi, Paul J., Heeres, Jan, Koymans, Lucien M.H., de Jonge, Marc R., Van Aken, Koen J.A., Daeyaert, Frederik F.D., Das, Kalyan, Arnold, Edward, Janssen, Paul A.J.
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
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Published in Bioorganic & medicinal chemistry letters (03.09.2001)
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
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Tripeptidyl-peptidase II (TPP II) inhibitory activity of (S)-2,3-dihydro-2-(1H-imidazol-2-yl)-1H-indoles, a systematic SAR evaluation. Part 2
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Published in Bioorganic & medicinal chemistry letters (15.12.2003)
Published in Bioorganic & medicinal chemistry letters (15.12.2003)
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Two Interrelated Strategies for Cephalotaxine Synthesis
Lin, Xiaodong, Kavash, Robert W, Mariano, Patrick S
Published in Journal of organic chemistry (18.10.1996)
Published in Journal of organic chemistry (18.10.1996)
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Optimized Fully-Synthetic Salicylamide Heparin Antagonists Have Greater Efficacy Versus LMWHs and Display Improved Hemodynamic Responses as Compared to Protamine
Scott, Richard W., Costanzo, Michael J., Freeman, Katie B., Kavash, Robert W., Young, Trevor M., DeGrado, William F., Jeske, Walter
Published in Blood (19.11.2010)
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Year of Publication 27.09.2012
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Year of Publication 27.09.2012
Patent
On the detection of multiple-binding modes of ligands to proteins, from biological, structural, and modeling data
Lewi, Paul J, de Jonge, Marc, Daeyaert, Frits, Koymans, Luc, Vinkers, Maarten, Heeres, Jan, Janssen, Paul A J, Arnold, Eddy, Das, Kalyan, Clark, Jr, Art D, Hughes, Stephen H, Boyer, Paul L, de Béthune, Marie-Pierre, Pauwels, Rudi, Andries, Koen, Kukla, Mike, Ludovici, Donald, De Corte, Bart, Kavash, Robert, Ho, Chih, Lewis, Paul J
Published in Journal of computer-aided molecular design (01.02.2003)
Published in Journal of computer-aided molecular design (01.02.2003)
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Tripeptidyl-peptidase II (TPP II) inhibitory activity of ( S )-2,3-dihydro-2-(1 H -imidazol-2-yl)-1 H -indoles, a systematic SAR evaluation. Part 2
Breslin, Henry J., Miskowski, Tamara A., Kukla, Michael J., De Winter, Hans L., Somers, Maria V.F., Roevens, Peter W.M., Kavash, Robert W.
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
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