Chemical proteomic profiles of the BCR-ABL inhibitors imatinib, nilotinib, and dasatinib reveal novel kinase and nonkinase targets
Rix, Uwe, Hantschel, Oliver, Dürnberger, Gerhard, Remsing Rix, Lily L., Planyavsky, Melanie, Fernbach, Nora V., Kaupe, Ines, Bennett, Keiryn L., Valent, Peter, Colinge, Jacques, Köcher, Thomas, Superti-Furga, Giulio
Published in Blood (01.12.2007)
Published in Blood (01.12.2007)
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Journal Article
A potent and highly specific FN3 monobody inhibitor of the Abl SH2 domain
Wojcik, John, Hantschel, Oliver, Grebien, Florian, Kaupe, Ines, Bennett, Keiryn L, Barkinge, John, Jones, Richard B, Koide, Akiko, Superti-Furga, Giulio, Koide, Shohei
Published in Nature structural & molecular biology (01.04.2010)
Published in Nature structural & molecular biology (01.04.2010)
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Journal Article
Charting the molecular network of the drug target Bcr-Abl
Brehme, Marc, Hantschel, Oliver, Colinge, Jacques, Kaupe, Ines, Planyavsky, Melanie, Köcher, Thomas, Mechtler, Karl, Bennett, Keiryn L, Superti-Furga, Giulio
Published in Proceedings of the National Academy of Sciences - PNAS (05.05.2009)
Published in Proceedings of the National Academy of Sciences - PNAS (05.05.2009)
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Journal Article
The chemokine interleukin-8 and the surface activation protein CD69 are markers for Bcr–Abl activity in chronic myeloid leukemia
Hantschel, Oliver, Gstoettenbauer, Agnes, Colinge, Jacques, Kaupe, Ines, Bilban, Martin, Burkard, Thomas R., Valent, Peter, Superti-Furga, Giulio
Published in Molecular oncology (01.10.2008)
Published in Molecular oncology (01.10.2008)
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Journal Article
BCR-ABL uncouples canonical JAK2-STAT5 signaling in chronic myeloid leukemia
Hantschel, Oliver, Warsch, Wolfgang, Eckelhart, Eva, Kaupe, Ines, Grebien, Florian, Wagner, Kay-Uwe, Superti-Furga, Giulio, Sexl, Veronika
Published in Nature chemical biology (29.01.2012)
Published in Nature chemical biology (29.01.2012)
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Journal Article
Targeting the SH2-Kinase Interface in Bcr-Abl Inhibits Leukemogenesis
Grebien, Florian, Hantschel, Oliver, Wojcik, John, Kaupe, Ines, Kovacic, Boris, Wyrzucki, Arkadiusz M., Gish, Gerald D., Cerny-Reiterer, Sabine, Koide, Akiko, Beug, Hartmut, Pawson, Tony, Valent, Peter, Koide, Shohei, Superti-Furga, Giulio
Published in Cell (14.10.2011)
Published in Cell (14.10.2011)
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Journal Article
BCR-ABL SH3-SH2 domain mutations in chronic myeloid leukemia patients on imatinib
Sherbenou, Daniel W., Hantschel, Oliver, Kaupe, Ines, Willis, Stephanie, Bumm, Thomas, Turaga, Lalita P., Lange, Thoralf, Dao, Kim-Hien, Press, Richard D., Druker, Brian J., Superti-Furga, Giulio, Deininger, Michael W.
Published in Blood (28.10.2010)
Published in Blood (28.10.2010)
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Initial characterization of the human central proteome
Burkard, Thomas R, Planyavsky, Melanie, Kaupe, Ines, Breitwieser, Florian P, Bürckstümmer, Tilmann, Bennett, Keiryn L, Superti-Furga, Giulio, Colinge, Jacques
Published in BMC systems biology (26.01.2011)
Published in BMC systems biology (26.01.2011)
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Bcr-Abl Directly Activates Stat5 Independent of Jak2
Hantschel, Oliver D., Eckelhart, Eva, Kaupe, Ines, Grebien, Florian, Wagner, Kay-Uwe, Sexl, Veronika, Superti-Furga, Giulio
Published in Blood (19.11.2010)
Published in Blood (19.11.2010)
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Abstract 5128: Physical EGFR network mapping and dynamic regulation in lung cancer cells
Li, Jiannong, Bennett, Keiryn, Song, Lanxi, Bai, Yun, Yoshida, Takeshi, Edwards, Arthur, Kinose, Fumi, Fang, Bin, Zhang, Guolin, Kaupe, Ines, Greben, Florian, Superti-Furga, Giulio, Haura, Eric
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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Targeting the SH2-Kinase Interface in Bcr-Abl Inhibits Leukemogenesis
Grebien, Florian, Hantschel, Oliver, Wojcik, John, Kaupe, Ines, Kovacic, Boris, Wyrzucki, Arkadiusz M., Gish, Gerald D., Cerny-Reiterer, Sabine, Koide, Akiko, Beug, Hartmut, Pawson, Tony, Valent, Peter, Koide, Shohei, Superti-Furga, Giulio
Published in Cell (01.10.2011)
Published in Cell (01.10.2011)
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Journal Article
The Bcr-Abl SH2-Kinase Domain Interface Is Critical for Leukemogenesis and An Additional Therapeutic Target in CML
Hantschel, Oliver D., Grebien, Florian, Kaupe, Ines, Kovacic, Boris, Wojcik, John, Gish, Gerald D, Koide, Shohei, Beug, Hartmut, Pawson, Tony, Superti-Furga, Giulio
Published in Blood (20.11.2009)
Published in Blood (20.11.2009)
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Journal Article
Characterization of BCR-ABL Deletion Mutants from Patients with Chronic Myeloid Leukemia
Sherbenou, Daniel W., Hantschel, Oliver J., Turaga, Lalita, Mag, Ines Kaupe, Willis, Stephanie, Bumm, Thomas, Press, Richard D., Superti-Furga, Giulio, Druker, Brian J., Deininger, Michael W.
Published in Blood (16.11.2007)
Published in Blood (16.11.2007)
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Journal Article
Systematic Profiling and Novel Targets of the Bcr-Abl Kinase Inhibitors Imatinib, Nilotinib and Dasatinib
Hantschel, Oliver, Rix, Uwe, Buerckstuemmer, Tilmann, Schmidt, Uwe, Kneidinger, Michael, Bennett, Keiryn L., Kaupe, Ines, Ellmeier, Wilfried, Valent, Peter, Superti-Furga, Giulio
Published in Blood (16.11.2007)
Published in Blood (16.11.2007)
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Experimental characterization of the human non-sequence-specific nucleic acid interactome
Dürnberger, Gerhard, Bürckstümmer, Tilmann, Huber, Kilian, Giambruno, Roberto, Doerks, Tobias, Karayel, Evren, Burkard, Thomas R, Kaupe, Ines, Müller, André C, Schönegger, Andreas, Ecker, Gerhard F, Lohninger, Hans, Bork, Peer, Bennett, Keiryn L, Superti-Furga, Giulio, Colinge, Jacques
Published in Genome biology (31.07.2013)
Published in Genome biology (31.07.2013)
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