Discovery of Ledipasvir (GS-5885): A Potent, Once-Daily Oral NS5A Inhibitor for the Treatment of Hepatitis C Virus Infection
Link, John O., Taylor, James G., Xu, Lianhong, Mitchell, Michael, Guo, Hongyan, Liu, Hongtao, Kato, Darryl, Kirschberg, Thorsten, Sun, Jianyu, Squires, Neil, Parrish, Jay, Keller, Terry, Yang, Zheng-Yu, Yang, Chris, Matles, Mike, Wang, Yujin, Wang, Kelly, Cheng, Guofeng, Tian, Yang, Mogalian, Erik, Mondou, Elsa, Cornpropst, Melanie, Perry, Jason, Desai, Manoj C.
Published in Journal of medicinal chemistry (13.03.2014)
Published in Journal of medicinal chemistry (13.03.2014)
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Journal Article
Discovery of the pan-genotypic hepatitis C virus NS3/4A protease inhibitor voxilaprevir (GS-9857): A component of Vosevi
Taylor, James G., Zipfel, Sheila, Ramey, Kyla, Vivian, Randy, Schrier, Adam, Karki, Kapil K., Katana, Ashley, Kato, Darryl, Kobayashi, Tetsuya, Martinez, Ruben, Sangi, Michael, Siegel, Dustin, Tran, Chinh V., Yang, Zheng-Yu, Zablocki, Jeff, Yang, Cheng Y., Wang, Yujin, Wang, Kelly, Chan, Katie, Barauskas, Ona, Cheng, Guofeng, Jin, Debi, Schultz, Brian E., Appleby, Todd, Villaseñor, Armando G., Link, John O.
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
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Enantioselective Synthesis of (+)-Cephalostatin 1
Fortner, Kevin C, Kato, Darryl, Tanaka, Yoshiki, Shair, Matthew D
Published in Journal of the American Chemical Society (13.01.2010)
Published in Journal of the American Chemical Society (13.01.2010)
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Journal Article
Discovery of velpatasvir (GS-5816): A potent pan-genotypic HCV NS5A inhibitor in the single-tablet regimens Vosevi® and Epclusa
Link, John O., Taylor, James G., Trejo-Martin, Alejandra, Kato, Darryl, Katana, Ashley A., Krygowski, Evan S., Yang, Zheng-Yu, Zipfel, Sheila, Cottell, Jeromy J., Bacon, Elizabeth M., Tran, Chinh V., Yang, Cheng Y., Wang, Yujin, Wang, Kelly W., Zhao, Guangyu, Cheng, Guofeng, Tian, Yang, Gong, Ruoyu, Lee, Yu-Jen, Yu, Mei, Gorman, Eric, Mogalian, Erik, Perry, Jason K.
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
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Journal Article
Direct binding of ledipasvir to HCV NS5A: mechanism of resistance to an HCV antiviral agent
Kwon, Hyock Joo, Xing, Weimei, Chan, Katie, Niedziela-Majka, Anita, Brendza, Katherine M, Kirschberg, Thorsten, Kato, Darryl, Link, John O, Cheng, Guofeng, Liu, Xiaohong, Sakowicz, Roman
Published in PloS one (09.04.2015)
Published in PloS one (09.04.2015)
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Journal Article
Correction to Discovery of Ledipasvir (GS-5885): A Potent, Once-Daily Oral NS5A Inhibitor for the Treatment of Hepatitis C Virus Infection
Link, John O, Taylor, James G, Xu, Lianhong, Mitchell, Michael, Guo, Hongyan, Liu, Hongtao, Kato, Darryl, Kirschberg, Thorsten, Sun, Jianyu, Squires, Neil, Parrish, Jay, Kellar, Terry, Yang, Zheng-Yu, Yang, Chris, Matles, Mike, Wang, Yujin, Wang, Kelly, Cheng, Guofeng, Tian, Yang, Mogalian, Erik, Mondou, Elsa, Cornpropst, Melanie, Perry, Jason, Desai, Manoj C
Published in Journal of medicinal chemistry (25.08.2016)
Published in Journal of medicinal chemistry (25.08.2016)
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Long-acting capsid inhibitor protects macaques from repeat SHIV challenges
Vidal, Samuel J, Bekerman, Elena, Hansen, Derek, Lu, Bing, Wang, Kelly, Mwangi, Judy, Rowe, William, Campigotto, Federico, Zheng, Jim, Kato, Darryl, Chandrashekar, Abishek, Barrett, Julia, Patel, Shivani, Wan, Huahua, Anioke, Tochi, Mercado, Noe B, Nkolola, Joseph P, Ferguson, Melissa J, Rinaldi, William J, Callebaut, Christian, Blair, Wade, Cihlar, Tomas, Geleziunas, Romas, Yant, Stephen R, Barouch, Dan H
Published in Nature (London) (27.01.2022)
Published in Nature (London) (27.01.2022)
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Neurotoxicity of an Hepatitis B Virus (HBV) Transcript Inhibitor in 13-Week Rat and Monkey Studies
Lake, April D, Holsapple, Kevin, McDonnell, Tanya, Arezzo, Joseph C, Ramirez, Ricardo, Gamelin, Lindsay, Yu, Mei, Glatt, Dylan, Dick, Ryan, Xie, Xiaodong, Choy, Regina, Cheng, Guofeng, Tay, Chin H, Chester, Anne, Kato, Darryl, Burns-Naas, Leigh Ann
Published in Toxicological sciences (28.03.2022)
Published in Toxicological sciences (28.03.2022)
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HIV 치료용 캡시드 저해제
KATO DARRYL, CHOU CHIENHUNG, SCHROEDER SCOTT D, TSE WINSTON C, ZHANG JENNIFER R, LAZERWITH SCOTT E
Year of Publication 27.02.2023
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Year of Publication 27.02.2023
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Year of Publication 01.08.2024
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Year of Publication 01.08.2024
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Discovery of Hepatitis B Virus Surface Antigen Suppressor GS-8873
Kato, Darryl, Choy, Regina Wai-Yan, Canales, Eda, Dick, Ryan A., Lake, April D., Shapiro, Nathan D., Chin, Elbert, Li, Jiayao, Zhang, Jennifer R., Wu, Qiaoyin, Saito, Roland D., Metobo, Sammy, Aktoudianakis, Evangelos, Schroeder, Scott D., Yang, Zheng-Yu, Glatt, Dylan M., Balsitis, Scott, Gamelin, Lindsay, Yu, Mei, Cheng, Guofeng, Delaney, William E., Link, John O.
Published in ACS medicinal chemistry letters (11.04.2024)
Published in ACS medicinal chemistry letters (11.04.2024)
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HIV 바이러스 감염 치료용 화합물
MACK JAMES B.C, WATKINS WILLIAM J, BRIZGYS GEDIMINAS J, GUNEY TEZCAN, LINK JOHN O, SCHROEDER SCOTT D, CHU HANG, MUN DONG MIN, FARAND JULIE, KATO DARRYL, LI JIAYAO, CHOU CHIENHUNG, WU QIAOYIN, ZHANG JENNIFER R, GRAUPE MICHAEL
Year of Publication 23.07.2024
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Year of Publication 23.07.2024
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Year of Publication 22.07.2024
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Year of Publication 22.07.2024
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Year of Publication 30.06.2023
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Year of Publication 30.06.2023
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Year of Publication 22.08.2022
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Year of Publication 22.08.2022
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Year of Publication 27.05.2024
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Year of Publication 27.05.2024
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MCL-1 MCL-1 INHIBITORS
WATKINS WILLIAM J, HWANG TAE H, HURTLEY ANNA E, SQUIRES NEIL H, TSUI VICKIE H, CHU HANG, NEWBY ZACHARY, KOBAYASHI TETSUYA, LI XIAOFEN, LIN DAVID W, VENKATARAMANI CHANDRASEKAR, LAZERWITH SCOTT E, KATO DARRYL, MITCHELL MICHAEL L, YANG HONG, GUERRERO JUAN A, JIANG LAN, MEDLEY JONATHAN W, KNOX JOHN E, NADUTHAMBI DEVAN
Year of Publication 18.07.2023
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Year of Publication 18.07.2023
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WATKINS WILLIAM J, MEDLEY JONATHAN WILLIAM, HURTLEY ANNA E, TSUI VICKIE H, CHU HANG, KOBAYASHI TETSUYA, LIN DAVID W, VENKATARAMANI CHANDRASEKAR, KATO DARRYL, YANG HONG, GUERRERO JUAN A, JIANG LAN, ZHU QINGMING, NADUTHAMBI DEVAN
Year of Publication 19.07.2022
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Year of Publication 19.07.2022
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