Pharmacological Properties of ABT-239 [4-(2-{2-[(2R)-2-Methylpyrrolidinyl]ethyl}-benzofuran-5-yl)benzonitrile]: II. Neurophysiological Characterization and Broad Preclinical Efficacy in Cognition and Schizophrenia of a Potent and Selective Histamine H3 Receptor Antagonist
Fox, Gerard B, Esbenshade, Timothy A, Pan, Jia Bao, Radek, Richard J, Krueger, Kathleen M, Yao, Betty B, Browman, Kaitlin E, Buckley, Michael J, Ballard, Michael E, Komater, Victoria A, Miner, Holly, Zhang, Min, Faghih, Ramin, Rueter, Lynne E, Bitner, R Scott, Drescher, Karla U, Wetter, Jill, Marsh, Kennan, Lemaire, Martine, Porsolt, Roger D, Bennani, Youssef L, Sullivan, James P, Cowart, Marlon D, Decker, Michael W, Hancock, Arthur A
Published in The Journal of pharmacology and experimental therapeutics (01.04.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2005)
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An 80-Amino Acid Deletion in the Third Intracellular Loop of a Naturally Occurring Human Histamine H3 Isoform Confers Pharmacological Differences and Constitutive Activity
Bongers, Gerold, Krueger, Kathleen M, Miller, Thomas R, Baranowski, John L, Estvander, Brian R, Witte, David G, Strakhova, Marina I, van Meer, Peter, Bakker, Remko A, Cowart, Marlon D, Hancock, Arthur A, Esbenshade, Timothy A, Leurs, Rob
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Published in The Journal of pharmacology and experimental therapeutics (01.12.2007)
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Two Novel and Selective Nonimidazole Histamine H3 Receptor Antagonists A-304121 and A-317920: I. In Vitro Pharmacological Effects
Esbenshade, Timothy A, Krueger, Kathleen M, Miller, Thomas R, Kang, Chae Hee, Denny, Lynne I, Witte, David G, Yao, Betty B, Fox, Gerard B, Faghih, Ramin, Bennani, Youssef L, Williams, Michael, Hancock, Arthur A
Published in The Journal of pharmacology and experimental therapeutics (01.06.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2003)
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Pharmacological and behavioral properties of A-349821, a selective and potent human histamine H3 receptor antagonist
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Published in Biochemical pharmacology (01.09.2004)
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G Protein-Dependent Pharmacology of Histamine H3 Receptor Ligands: Evidence for Heterogeneous Active State Receptor Conformations
Krueger, Kathleen M, Witte, David G, Ireland-Denny, Lynne, Miller, Thomas R, Baranowski, John L, Buckner, Steve, Milicic, Ivan, Esbenshade, Timothy A, Hancock, Arthur A
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Published in The Journal of pharmacology and experimental therapeutics (01.07.2005)
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Novel heterocyclic-substituted benzofuran histamine H3 receptor antagonists: in vitro properties, drug-likeness, and behavioral activity
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Published in Biochemical pharmacology (15.04.2007)
Published in Biochemical pharmacology (15.04.2007)
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Pharmacological properties and procognitive effects of ABT-288, a potent and selective histamine H3 receptor antagonist
Esbenshade, Timothy A, Browman, Kaitlin E, Miller, Thomas R, Krueger, Kathleen M, Komater-Roderwald, Victoria, Zhang, Min, Fox, Gerard B, Rueter, Lynne, Robb, Holly M, Radek, Richard J, Drescher, Karla U, Fey, Thomas A, Bitner, R Scott, Marsh, Kennan, Polakowski, James S, Zhao, Chen, Cowart, Marlon D, Hancock, Arthur A, Sullivan, James P, Brioni, Jorge D
Published in The Journal of pharmacology and experimental therapeutics (01.10.2012)
Published in The Journal of pharmacology and experimental therapeutics (01.10.2012)
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Genetic and pharmacological aspects of histamine H3 receptor heterogeneity
Hancock, Arthur A, Esbenshade, Timothy A, Krueger, Kathleen M, Yao, Betty Bei
Published in Life sciences (1973) (31.10.2003)
Published in Life sciences (1973) (31.10.2003)
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The Alkaloid Conessine and Analogues as Potent Histamine H3 Receptor Antagonists
Zhao, Chen, Sun, Minghua, Bennani, Youssef L, Gopalakrishnan, Sujatha M, Witte, David G, Miller, Thomas R, Krueger, Kathleen M, Browman, Kaitlin E, Thiffault, Christine, Wetter, Jill, Marsh, Kennan C, Hancock, Arthur A, Esbenshade, Timothy A, Cowart, Marlon D
Published in Journal of medicinal chemistry (11.09.2008)
Published in Journal of medicinal chemistry (11.09.2008)
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Receptor-tyrosine-kinase- and Gβγ-mediated MAP kinase activation by a common signalling pathway
Blesen, Tim van, Hawes, Brian E, Luttrell, Deirdre K, Krueger, Kathleen M, Touhara, Kazushige, Porfflri, Emilio, Sakaue, Motoyoshi, Luttrell, Louis M, Lefkowitz, Robert J
Published in Nature (London) (31.08.1995)
Published in Nature (London) (31.08.1995)
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Antiobesity effects of A-331440, a novel non-imidazole histamine H3 receptor antagonist
HANCOCK, Arthur A, BENNANI, Youssef L, JIA BAO PAN, SHAPIRO, Robin, WITTE, David G, YAO, Betty B, BUSH, Eugene N, ESBENSHADE, Timothy A, FAGHIH, Ramin, FOX, Gerard B, JACOBSON, Peer, KNOUREK-SEGEL, Victoria, KRUEGER, Kathleen M, NUSS, Merrill E
Published in European journal of pharmacology (08.03.2004)
Published in European journal of pharmacology (08.03.2004)
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Detection of multiple H-3 receptor affinity states utilizing [H-3]A-349821, a novel, selective, non-imidazole histamine H-3 receptor inverse agonist radioligand
Witte, David G., Yao, Betty Bei, Miller, Thomas R., Carr, Tracy L., Cassar, Steven, Sharma, Rahul, Faghih, Ramin, Surber, Bruce W., Esbenshade, Timothy A., Hancock, Arthur A., Krueger, Kathleen M.
Published in British journal of pharmacology (29.01.2009)
Published in British journal of pharmacology (29.01.2009)
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Synthesis, Potency, and In Vivo Profiles of Quinoline Containing Histamine H3 Receptor Inverse Agonists
Altenbach, Robert J, Liu, Huaqing, Banfor, Patricia N, Browman, Kaitlin E, Fox, Gerard B, Fryer, Ryan M, Komater, Victoria A, Krueger, Kathleen M, Marsh, Kennan, Miller, Thomas R, Pan, Jia Bao, Pan, Liping, Sun, Minghua, Thiffault, Christine, Wetter, Jill, Zhao, Chen, Zhou, Deliang, Esbenshade, Timothy A, Hancock, Arthur A, Cowart, Marlon D
Published in Journal of medicinal chemistry (01.11.2007)
Published in Journal of medicinal chemistry (01.11.2007)
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In vitro Optimization of Structure Activity Relationships of Analogues of A‐331440 Combining Radioligand Receptor Binding Assays and Micronucleus Assays of Potential Antiobesity Histamine H3 Receptor Antagonists
Hancock, Arthur A., Diehl, Marilyn S., Faghih, Ramin, Bush, Eugene N., Krueger, Kathleen M., Krishna, Gopala, Miller, Thomas R., Wilcox, Nguyen, Phong, Pratt, John K., Cowart, Marlon D., Esbenshade, Timothy A., Jacobson, Peer B.
Published in Basic & clinical pharmacology & toxicology (01.09.2004)
Published in Basic & clinical pharmacology & toxicology (01.09.2004)
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Detection of multiple H3 receptor affinity states utilizing [3H]A‐349821, a novel, selective, non‐imidazole histamine H3 receptor inverse agonist radioligand
Witte, David G, Yao, Betty Bei, Miller, Thomas R, Carr, Tracy L, Cassar, Steven, Sharma, Rahul, Faghih, Ramin, Surber, Bruce W, Esbenshade, Timothy A, Hancock, Arthur A, Krueger, Kathleen M
Published in British journal of pharmacology (01.07.2006)
Published in British journal of pharmacology (01.07.2006)
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Pharmacological Properties of ABT-239 [4-(2-{2-[(2R)-2-Methylpyrrolidinyl]ethyl}-benzofuran-5-yl)benzonitrile]: I. Potent and Selective Histamine H3 Receptor Antagonist with Drug-Like Properties
Esbenshade, Timothy A, Fox, Gerard B, Krueger, Kathleen M, Miller, Thomas R, Kang, Chae Hee, Denny, Lynne I, Witte, David G, Yao, Betty B, Pan, Liping, Wetter, Jill, Marsh, Kennan, Bennani, Youssef L, Cowart, Marlon D, Sullivan, James P, Hancock, Arthur A
Published in The Journal of pharmacology and experimental therapeutics (01.04.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2005)
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Differential activation of dual signaling responses by human H1 and H2 histamine receptors
Esbenshade, Timothy A, Kang, Chae Hee, Krueger, Kathleen M, Miller, Thomas R, Witte, David G, Roch, Jean M, Masters, Jeffrey N, Hancock, Arthur A
Published in Journal of receptors and signal transduction (2003)
Published in Journal of receptors and signal transduction (2003)
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Journal Article
Pharmacological Properties and Procognitive Effects of ABT-288, a Potent and Selective Histamine H 3 Receptor Antagonist
Esbenshade, Timothy A., Browman, Kaitlin E., Miller, Thomas R., Krueger, Kathleen M., Komater-Roderwald, Victoria, Zhang, Min, Fox, Gerard B., Rueter, Lynne, Robb, Holly M., Radek, Richard J., Drescher, Karla U., Fey, Thomas A., Bitner, R. Scott, Marsh, Kennan, Polakowski, James S., Zhao, Chen, Cowart, Marlon D., Hancock, Arthur A., Sullivan, James P., Brioni, Jorge D.
Published in The Journal of pharmacology and experimental therapeutics (01.10.2012)
Published in The Journal of pharmacology and experimental therapeutics (01.10.2012)
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The Role of Sequestration in G Protein-coupled Receptor Resensitization
Krueger, Kathleen M., Daaka, Yehia, Pitcher, Julie A., Lefkowitz, Robert J.
Published in The Journal of biological chemistry (01.01.1997)
Published in The Journal of biological chemistry (01.01.1997)
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Journal Article
Pharmacological Properties of ABT-239 [4-(2-{2-[(2 R )-2-Methylpyrrolidinyl]ethyl}-benzofuran-5-yl)benzonitrile]: II. Neurophysiological Characterization and Broad Preclinical Efficacy in Cognition and Schizophrenia of a Potent and Selective Histamine H 3 Receptor Antagonist
Fox, Gerard B., Esbenshade, Timothy A., Pan, Jia Bao, Radek, Richard J., Krueger, Kathleen M., Yao, Betty B., Browman, Kaitlin E., Buckley, Michael J., Ballard, Michael E., Komater, Victoria A., Miner, Holly, Zhang, Min, Faghih, Ramin, Rueter, Lynne E., Bitner, R. Scott, Drescher, Karla U., Wetter, Jill, Marsh, Kennan, Lemaire, Martine, Porsolt, Roger D., Bennani, Youssef L., Sullivan, James P., Cowart, Marlon D., Decker, Michael W., Hancock, Arthur A.
Published in The Journal of pharmacology and experimental therapeutics (01.04.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2005)
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