Discovery of novel histone lysine methyltransferase G9a/GLP (EHMT2/1) inhibitors: Design, synthesis, and structure-activity relationships of 2,4-diamino-6-methylpyrimidines
Katayama, Katsushi, Ishii, Ken, Tsuda, Eisuke, Yotsumoto, Keiichi, Hiramoto, Kumiko, Suzuki, Makoto, Yasumatsu, Isao, Igarashi, Wataru, Torihata, Munefumi, Ishiyama, Takashi, Katagiri, Takahiro
Published in Bioorganic & medicinal chemistry letters (15.10.2020)
Published in Bioorganic & medicinal chemistry letters (15.10.2020)
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Journal Article
Synthesis and Biological Evaluation of Quinaldopeptin
Katayama, Katsushi, Okamura, Takuya, Sunadome, Takuya, Nakagawa, Koji, Takeda, Hiroshi, Shiro, Motoo, Matsuda, Akira, Ichikawa, Satoshi
Published in Journal of organic chemistry (21.03.2014)
Published in Journal of organic chemistry (21.03.2014)
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Journal Article
Total Synthesis of Sandramycin and Its Analogues via a Multicomponent Assemblage
Katayama, Katsushi, Nakagawa, Koji, Takeda, Hiroshi, Matsuda, Akira, Ichikawa, Satoshi
Published in Organic letters (17.01.2014)
Published in Organic letters (17.01.2014)
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Journal Article
Design, synthesis, and biological evaluation of spiroindolines as novel inducers of oligodendrocyte progenitor cell differentiation—Use of a conformation-based hypothesis to facilitate compound design
Katayama, Katsushi, Nagata, Tsutomu, Takashima, Kouhei, Yoshida, Ayako, Okada, Hiroyuki, Oyama, Yoshiaki, Muto, Tsuyoshi
Published in Bioorganic & medicinal chemistry letters (15.08.2020)
Published in Bioorganic & medicinal chemistry letters (15.08.2020)
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Journal Article
Phenotypic-screening generates active novel fetal globin-inducers that downregulate Bcl11a in a monkey model
Makino, Tomohiro, Haruyama, Munetada, Katayama, Katsushi, Terashima, Hideki, Tsunemi, Tomoyuki, Miyazaki, Kazuo, Terakawa, Maki, Yamashiro, Kyoko, Yoshioka, Ryosuke, Maeda, Hiroaki
Published in Biochemical pharmacology (01.01.2020)
Published in Biochemical pharmacology (01.01.2020)
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Journal Article
Discovery and structure-activity relationships of spiroindolines as novel inducers of oligodendrocyte progenitor cell differentiation
Katayama, Katsushi, Arai, Yoshikazu, Murata, Kenji, Saito, Shoichi, Nagata, Tsutomu, Takashima, Kouhei, Yoshida, Ayako, Masumura, Makoto, Koda, Shuichi, Okada, Hiroyuki, Muto, Tsuyoshi
Published in Bioorganic & medicinal chemistry (15.03.2020)
Published in Bioorganic & medicinal chemistry (15.03.2020)
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Journal Article
Design, synthesis, and optimization of a series of 2-azaspiro[3.3]heptane derivatives as orally bioavailable fetal hemoglobin inducers
Katayama, Katsushi, Tsunemi, Tomoyuki, Miyazaki, Kazuo, Uoto, Kouichi, Yoshioka, Ryosuke, Terashima, Hideki, Terakawa, Maki, Yamashiro, Kyoko, Haruyama, Munetada, Maeda, Hiroaki, Makino, Tomohiro
Published in Bioorganic & medicinal chemistry letters (01.10.2020)
Published in Bioorganic & medicinal chemistry letters (01.10.2020)
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Journal Article
Discovery of DS79932728: A Potent, Orally Available G9a/GLP Inhibitor for Treating beta-Thalassemia and Sickle Cell Disease
Katayama, Katsushi, Ishii, Ken, Terashima, Hideki, Tsuda, Eisuke, Suzuki, Makoto, Yotsumoto, Keiichi, Hiramoto, Kumiko, Yasumatsu, Isao, Torihata, Munefumi, Ishiyama, Takashi, Muto, Tsuyoshi, Katagiri, Takahiro
Published in ACS medicinal chemistry letters (14.01.2021)
Published in ACS medicinal chemistry letters (14.01.2021)
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Journal Article
SUBSTITUTED BENZENE COMPOUND
NAKAZAWA Yusuke, INOUE Masahiro, FUJIMOTO Teppei, TSUCHIYA Yuto, MATSUI Satoshi, ISHIBASHI Koutaro, MURAKAMI Keigo, KATAYAMA Katsushi, KAWAI Junya
Year of Publication 02.08.2024
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Year of Publication 02.08.2024
Patent
ChemInform Abstract: Total Synthesis of Sandramycin and Its Analogues via a Multicomponent Assemblage
Katayama, Katsushi, Nakagawa, Koji, Takeda, Hiroshi, Matsuda, Akira, Ichikawa, Satoshi
Published in ChemInform (01.07.2014)
Published in ChemInform (01.07.2014)
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Journal Article
ChemInform Abstract: Synthesis and Biological Evaluation of Quinaldopeptin
Katayama, Katsushi, Okamura, Takuya, Sunadome, Takuya, Nakagawa, Koji, Takeda, Hiroshi, Shiro, Motoo, Matsuda, Akira, Ichikawa, Satoshi
Published in ChemInform (02.09.2014)
Published in ChemInform (02.09.2014)
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Journal Article