Structure Based Discovery of Inhibitors of CYP125 and CYP142 from Mycobacterium tuberculosis
Katariya, Mona M., Snee, Matthew, Tunnicliffe, Richard B., Kavanagh, Madeline E., Boshoff, Helena I. M., Amadi, Cecilia N., Levy, Colin W., Munro, Andrew W., Abell, Chris, Leys, David, Coyne, Anthony G., McLean, Kirsty J.
Published in Chemistry : a European journal (22.05.2023)
Published in Chemistry : a European journal (22.05.2023)
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Non-classical Helices with cis Carbon-Carbon Double Bonds in the Backbone: Structural Features of α,γ-Hybrid Peptide Foldamers
Ganesh Kumar, Mothukuri, Thombare, Varsha J., Katariya, Mona M., Veeresh, Kuruva, Raja, K. Muruga Poopathi, Gopi, Hosahudya N.
Published in Angewandte Chemie (International ed.) (27.06.2016)
Published in Angewandte Chemie (International ed.) (27.06.2016)
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A new strategy for hit generation: Novel in cellulo active inhibitors of CYP121A1 from Mycobacterium tuberculosis via a combined X-ray crystallographic and phenotypic screening approach (XP screen)
Frederickson, Martyn, Selvam, Irwin R., Evangelopoulos, Dimitrios, McLean, Kirsty J., Katariya, Mona M., Tunnicliffe, Richard B., Campbell, Bethany, Kavanagh, Madeline E., Charoensutthivarakul, Sitthivut, Blankley, Richard T., Levy, Colin W., de Carvalho, Luiz Pedro S., Leys, David, Munro, Andrew W., Coyne, Anthony G., Abell, Chris
Published in European journal of medicinal chemistry (15.02.2022)
Published in European journal of medicinal chemistry (15.02.2022)
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HBTU mediated 1-hydroxybenzotriazole (HOBt) conjugate addition: synthesis and stereochemical analysis of beta-benzotriazole N-oxide substituted gamma-amino acids and hybrid peptides
Mali, Sachitanand M., Kumar, Mothukuri Ganesh, Katariya, Mona M., Gopi, Hosahudya N.
Published in Organic & biomolecular chemistry (14.11.2014)
Published in Organic & biomolecular chemistry (14.11.2014)
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Journal Article
Non-classical Helices with cis Carbon-Carbon Double Bonds in the Backbone: Structural Features of α,γ-Hybrid Peptide Foldamers
Ganesh Kumar, Mothukuri, Thombare, Varsha J., Katariya, Mona M., Veeresh, Kuruva, Raja, K. Muruga Poopathi, Gopi, Hosahudya N.
Published in Angewandte Chemie (27.06.2016)
Published in Angewandte Chemie (27.06.2016)
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Journal Article
Non-classical Helices with cis Carbon-Carbon Double Bonds in the Backbone: Structural Features of [alpha],[gamma]-Hybrid Peptide Foldamers
GaneshKumar, Mothukuri, Thombare, Varsha J, Katariya, Mona M, Veeresh, Kuruva, Raja, K Muruga Poopathi, Gopi, Hosahudya N
Published in Angewandte Chemie International Edition (27.06.2016)
Published in Angewandte Chemie International Edition (27.06.2016)
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Journal Article
HBTU mediated 1-hydroxybenzotriazole (HOBt) conjugate addition: synthesis and stereochemical analysis of β-benzotriazole N-oxide substituted γ-amino acids and hybrid peptidesElectronic supplementary information (ESI) available: 1H and 13C NMR spectra of 1a-f, 6a-d, 7a-d, dipeptides, 8 (i, ii)-12(i, ii) and 13, and ORTEP diagrams for 7a, 6a, 6c, 10i and 13. CCDC 1012298-1012302. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c4ob01548g
Mali, Sachitanand M, Ganesh Kumar, Mothukuri, Katariya, Mona M, Gopi, Hosahudya N
Year of Publication 09.10.2014
Year of Publication 09.10.2014
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Journal Article
Non-classical Helices with cis Carbon-Carbon Double Bonds in the Backbone: Structural Features of [alpha],[gamma]-Hybrid Peptide Foldamers
GaneshKumar, Mothukuri, Thombare, Varsha J, Katariya, Mona M, Veeresh, Kuruva, Raja, K Muruga Poopathi, Gopi, Hosahudya N
Published in Angewandte Chemie (27.06.2016)
Published in Angewandte Chemie (27.06.2016)
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Journal Article