A mimetic of the mSin3-binding helix of NRSF/REST ameliorates abnormal pain behavior in chronic pain models
Ueda, Hiroshi, Kurita, Jun-ichi, Neyama, Hiroyuki, Hirao, Yuuka, Kouji, Hiroyuki, Mishina, Tadashi, Kasai, Masaji, Nakano, Hirofumi, Yoshimori, Atsushi, Nishimura, Yoshifumi
Published in Bioorganic & medicinal chemistry letters (15.10.2017)
Published in Bioorganic & medicinal chemistry letters (15.10.2017)
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Development of Low-Molecular-Weight Compounds Targeting the Cancer-Associated KLF5 Transcription Factor
Nakaya, Takeo, Aizawa, Kenichi, Taguchi, Yuki, Tsuji, Kentaro, Sekine, Sachi, Murakami, Kazuhiro, Kasai, Masaji, Nakano, Hirofumi, Kondoh, Yasumitsu, Dan, Shingo, Yoshimori, Atsushi, Kouji, Hiroyuki, Takehara, Dai, Suzuki, Toru, Osada, Hiroyuki, Murata, Masayuki, Tanaka, Akira, Nagai, Ryozo
Published in ACS medicinal chemistry letters (14.04.2022)
Published in ACS medicinal chemistry letters (14.04.2022)
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Visualized and Quantitative Conformational Analysis of Peptidomimetics
Takashima, Hajime, Yoshimori, Atsushi, Honda, Eiji, Taguri, Tomonori, Ozawa, Jun, Kasai, Masaji, Shuto, Satoshi, Takehara, Dai
Published in ACS omega (12.10.2021)
Published in ACS omega (12.10.2021)
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Bioreductive activation of mitomycin C by DT-diaphorase
Siegel, David, Beall, Howard, Senekowitsch, Claudia, Kasai, Masaji, Arai, Hitoshi, Gibson, Neil W, Ross, David
Published in Biochemistry (Easton) (01.09.1992)
Published in Biochemistry (Easton) (01.09.1992)
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Development of a Practical Synthetic Route of a PDE V Inhibitor KF31327
Fujino, Kenji, Takami, Hitoshi, Atsumi, Toshiyuki, Ogasa, Takehiro, Mohri, Shin-ichiro, Kasai, Masaji
Published in Organic process research & development (01.07.2001)
Published in Organic process research & development (01.07.2001)
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ANTICANCER AGENT AND CARDIAC-FUNCTION-IMPROVING AGENT
AIZAWA, Kenichi, NAGAI, Ryozo, NAKAYA, Takeo, NAKANO, Hirofumi, KOUJI, Hiroyuki, KASAI, Masaji
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
Patent
Large scale synthesis of the high quality indoloquinone antitumor agent EO 9 via [bis(trifluoroacetoxy)iodo]benzene oxidation of 4-aminoindole
Kinugawa, M, Masuda, Y, Arai, H, Nishikawa, H, Ogasa, T, Tomioka, S, Kasai, M
Published in Synthesis (Stuttgart) (01.05.1996)
Published in Synthesis (Stuttgart) (01.05.1996)
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Journal Article
NOVEL Sin3 MODULATOR AND MEDICAL APPLICATION THEREOF
MISHINA, Tadashi, HIRAO, Yuka, HASHIMOTO, Hitoshi, KAWASE, Haruki, AGO, Yukio, NISHIMURA, Yoshifumi, KOUJI, Hiroyuki, KURITA, Junichi, KASAI, Masaji, YOSHIMORI, Atsushi
Year of Publication 07.03.2019
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Year of Publication 07.03.2019
Patent
Comparison of uptake of mitomycin C and KW-2149 by murine P388 leukemia cells sensitive or resistant to mitomycin C
Kobayashi, E, Okabe, M, Kono, M, Arai, H, Kasai, M, Gomi, K, Lee, J H, Inaba, M, Tsuruo, T
Published in Cancer chemotherapy and pharmacology (01.01.1993)
Published in Cancer chemotherapy and pharmacology (01.01.1993)
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Journal Article
Synthesis and biological evaluation of quinocarcin derivatives: thioalkyl-substituted quinones and hydroquinones
Saito, Hiromitsu, Hirata, Tadashi, Kasai, Masaji, Fujimoto, Kazuhisa, Ashizawa, Tadashi, Morimoto, Makoto, Sato, Akira
Published in Journal of medicinal chemistry (01.07.1991)
Published in Journal of medicinal chemistry (01.07.1991)
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Journal Article
Microbially mediated enantioselective ester hydrolyses utilizing Rhizopus nigricans. A new method of assigning the absolute stereochemistry of acyclic 1-arylalkanols
Ziffer, Herman, Kawai, Kenichi, Kasai, Masaji, Imuta, Mitsuru, Froussios, Cleanthis
Published in Journal of organic chemistry (01.09.1983)
Published in Journal of organic chemistry (01.09.1983)
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Journal Article
Synthesis and structure-activity relationships of new dimeric mitomycin derivatives; 7-N,7'-N'bis(.OMEGA.-thioalkyl)dimitomycins
KONO, MOTOMICHI, SAITOH, YUTAKA, KASAI, MASAJI, SHIRAHATA, KUNIKATSU, MORIMOTO, MAKOTO, ASHIZAWA, TADASHI
Published in Journal of antibiotics (1993)
Published in Journal of antibiotics (1993)
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Journal Article
THE CONFIGURATION OF MITIROMYCIN AND ITS DERIVATION FROM MITOMYCIN B
KONO, MOTOMICHI, KASAI, MASAJI, SHIRAHATA, KUNIKATSU, HIRAYAMA, NORIAKI
Published in Journal of antibiotics (1991)
Published in Journal of antibiotics (1991)
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Journal Article
Preparation of chiral allylic alcohols using Rhizopusnigricans. Use of the Harada-Nakanishi exciton chirality method for verifying configurational assignments of allylic alcohols
Ito, Satoru, Kasai, Masaji, Ziffer, Herman, Sllverton, J. V
Published in Canadian journal of chemistry (01.03.1987)
Published in Canadian journal of chemistry (01.03.1987)
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