Serum thymidine kinase 1 activity as a pharmacodynamic marker of cyclin-dependent kinase 4/6 inhibition in patients with early-stage breast cancer receiving neoadjuvant palbociclib
Bagegni, Nusayba, Thomas, Shana, Liu, Ning, Luo, Jingqin, Hoog, Jeremy, Northfelt, Donald W, Goetz, Matthew P, Forero, Andres, Bergqvist, Mattias, Karen, Jakob, Neumüller, Magnus, Suh, Edward M, Guo, Zhanfang, Vij, Kiran, Sanati, Souzan, Ellis, Matthew, Ma, Cynthia X
Published in Breast cancer research : BCR (21.11.2017)
Published in Breast cancer research : BCR (21.11.2017)
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Integrin α 1 β 1 is involved in the differentiation into myofibroblasts in adult reactive tissues in vivo
Rodriguez, Alejandro, Karen, Jakob, Gardner, Humphrey, Gerdin, Bengt, Rubin, Kristofer, Sundberg, Christian
Published in Journal of cellular and molecular medicine (01.09.2009)
Published in Journal of cellular and molecular medicine (01.09.2009)
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Discovery and Characterization of the Potent and Highly Selective 1,7-Naphthyridine-Based Inhibitors BAY-091 and BAY-297 of the Kinase PIP4K2A
Wortmann, Lars, Bräuer, Nico, Holton, Simon J, Irlbacher, Horst, Weiske, Jörg, Lechner, Christian, Meier, Robin, Karén, Jakob, Siöberg, Catrine Berthold, Pütter, Vera, Christ, Clara D, ter Laak, Antonius, Lienau, Philip, Lesche, Ralf, Nicke, Barbara, Cheung, Shing-Hu, Bauser, Marcus, Haegebarth, Andrea, von Nussbaum, Franz, Mumberg, Dominik, Lemos, Clara
Published in Journal of medicinal chemistry (11.11.2021)
Published in Journal of medicinal chemistry (11.11.2021)
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Determining direct binders of the Androgen Receptor using a high-throughput Cellular Thermal Shift Assay
Shaw, Joseph, Leveridge, Mathew, Norling, Charlotta, Karén, Jakob, Molina, Daniel Martinez, O'Neill, Daniel, Dowling, James E, Davey, Paul, Cowan, Suzanna, Dabrowski, Michael, Main, Martin, Gianni, Davide
Published in Scientific reports (09.01.2018)
Published in Scientific reports (09.01.2018)
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Journal Article
Effects of the histone deacetylase inhibitor valproic acid on human pericytes in vitro
Karén, Jakob, Rodriguez, Alejandro, Friman, Tomas, Dencker, Lennart, Sundberg, Christian, Scholz, Birger
Published in PloS one (22.09.2011)
Published in PloS one (22.09.2011)
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Journal Article
Effects of tiotropium bromide on airway hyperresponsiveness and inflammation in mice exposed to organic dust
Gregory, Joshua A., Kemi, Cecilia, Ji, Jie, Karén, Jakob, Delin, Ingrid, Gerde, Per, Pieper, Michael P., Adner, Mikael, Larsson, Kjell
Published in Pulmonary pharmacology & therapeutics (01.02.2018)
Published in Pulmonary pharmacology & therapeutics (01.02.2018)
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Abstract PO3-26-04: Discovery of novel inhibitors of the epigenetic regulatory KAT6A histone acetyl transferase and their anti-tumor activity in breast cancer cells
Holsinger, Leslie, RaI, Roopa, Nagawade, Rahul R., Pal, Benoy, Pawar, Samir, Singh, Pankaj, Putta, Krishna, Jaleel, Mahaboobi, Bostrom, Tove, Karen, Jakob, Huang, Qianyang, Hannah, Alison
Published in Cancer research (Chicago, Ill.) (02.05.2024)
Published in Cancer research (Chicago, Ill.) (02.05.2024)
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Journal Article
Integrin α1β1 is involved in the differentiation into myofibroblasts in adult reactive tissues in vivo
Rodriguez, Alejandro, Karen, Jakob, Gardner, Humphrey, Gerdin, Bengt, Rubin, Kristofer, Sundberg, Christian
Published in Journal of cellular and molecular medicine (01.09.2009)
Published in Journal of cellular and molecular medicine (01.09.2009)
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Journal Article
Integrin [alpha]^sub 1^[beta]^sub 1^ is involved in the differentiation into myofibroblasts in adult reactive tissues in vivo
Rodriguez, Alejandro, Karen, Jakob, Gardner, Humphrey, Gerdin, Bengt, Rubin, Kristofer, Sundberg, Christian
Published in Journal of cellular and molecular medicine (01.09.2009)
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Published in Journal of cellular and molecular medicine (01.09.2009)
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Abstract 354: Physiologically relevant target engagement using CETSA
Karén, Jakob, Sioberg, Catrine, Niekrasz, Pawel, Neumuller, Magnus, Martinez Molina, Daniel
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Journal Article
Integrin alpha1beta1 is involved in the differentiation into myofibroblasts in adult reactive tissues in vivo
Rodriguez, Alejandro, Karen, Jakob, Gardner, Humphrey, Gerdin, Bengt, Rubin, Kristofer, Sundberg, Christian
Published in Journal of cellular and molecular medicine (01.09.2009)
Published in Journal of cellular and molecular medicine (01.09.2009)
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