Adipocyte P2Y14 receptors play a key role in regulating whole-body glucose and lipid homeostasis
Jain, Shanu, Pydi, Sai P, Jung, Young-Hwan, Scortichini, Mirko, Kesner, Efrat L, Karcz, Tadeusz P, Cook, Donald N, Gavrilova, Oksana, Wess, Jürgen, Jacobson, Kenneth A
Published in JCI insight (24.05.2021)
Published in JCI insight (24.05.2021)
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Journal Article
UDP-glucose and P2Y14 receptor amplify allergen-induced airway eosinophilia
Karcz, Tadeusz P, Whitehead, Gregory S, Nakano, Keiko, Nakano, Hideki, Grimm, Sara A, Williams, Jason G, Deterding, Leesa J, Jacobson, Kenneth A, Cook, Donald N
Published in The Journal of clinical investigation (01.04.2021)
Published in The Journal of clinical investigation (01.04.2021)
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Journal Article
Bridged Piperidine Analogues of a High Affinity Naphthalene-Based P2Y14R Antagonist
Wen, Zhiwei, Salmaso, Veronica, Jung, Young-Hwan, Phung, Ngan B, Gopinatth, Varun, Shah, Qasim, Patterson, Alexandra T, Randle, John C. R, Chen, Zhoumou, Salvemini, Daniela, Lieberman, David I, Whitehead, Gregory S, Karcz, Tadeusz P, Cook, Donald N, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (24.02.2022)
Published in Journal of medicinal chemistry (24.02.2022)
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Journal Article
Bridged Piperidine Analogues of a High Affinity Naphthalene-Based P2Y 14 R Antagonist
Wen, Zhiwei, Salmaso, Veronica, Jung, Young-Hwan, Phung, Ngan B, Gopinatth, Varun, Shah, Qasim, Patterson, Alexandra T, Randle, John C R, Chen, Zhoumou, Salvemini, Daniela, Lieberman, David I, Whitehead, Gregory S, Karcz, Tadeusz P, Cook, Donald N, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (24.02.2022)
Published in Journal of medicinal chemistry (24.02.2022)
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Journal Article
Structure–Activity Relationship of Heterocyclic P2Y14 Receptor Antagonists: Removal of the Zwitterionic Character with Piperidine Bioisosteres
Jung, Young-Hwan, Salmaso, Veronica, Wen, Zhiwei, Bennett, John M, Phung, Ngan B, Lieberman, David I, Gopinatth, Varun, Randle, John C. R, Chen, Zhoumou, Salvemini, Daniela, Karcz, Tadeusz P, Cook, Donald N, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (22.04.2021)
Published in Journal of medicinal chemistry (22.04.2021)
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Journal Article
Structure-Activity Relationship of Heterocyclic P2Y 14 Receptor Antagonists: Removal of the Zwitterionic Character with Piperidine Bioisosteres
Jung, Young-Hwan, Salmaso, Veronica, Wen, Zhiwei, Bennett, John M, Phung, Ngan B, Lieberman, David I, Gopinatth, Varun, Randle, John C R, Chen, Zhoumou, Salvemini, Daniela, Karcz, Tadeusz P, Cook, Donald N, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (22.04.2021)
Published in Journal of medicinal chemistry (22.04.2021)
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Journal Article
Exploration of Alternative Scaffolds for P2Y14 Receptor Antagonists Containing a Biaryl Core
Jung, Young-Hwan, Yu, Jinha, Wen, Zhiwei, Salmaso, Veronica, Karcz, Tadeusz P, Phung, Ngan B, Chen, Zhoumou, Duca, Sierra, Bennett, John M, Dudas, Steven, Salvemini, Daniela, Gao, Zhan-Guo, Cook, Donald N, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (10.09.2020)
Published in Journal of medicinal chemistry (10.09.2020)
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Journal Article
Exploration of Alternative Scaffolds for P2Y 14 Receptor Antagonists Containing a Biaryl Core
Jung, Young-Hwan, Yu, Jinha, Wen, Zhiwei, Salmaso, Veronica, Karcz, Tadeusz P, Phung, Ngan B, Chen, Zhoumou, Duca, Sierra, Bennett, John M, Dudas, Steven, Salvemini, Daniela, Gao, Zhan-Guo, Cook, Donald N, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (10.09.2020)
Published in Journal of medicinal chemistry (10.09.2020)
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Journal Article
Effects of Purinergic Receptor Deletion or Pharmacologic Modulation on Pulmonary Inflammation in Mice
Whitehead, Gregory S., Karcz, Tadeusz P., Tosh, Dilip K., Jung, Young-Hwan, Wen, Zhiwei, Campbell, Ryan G., Gopinatth, Varun, Gao, Zhan-Guo, Jacobson, Kenneth A., Cook, Donald N.
Published in ACS pharmacology & translational science (14.10.2022)
Published in ACS pharmacology & translational science (14.10.2022)
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Journal Article
Therapeutic suppression of pulmonary neutrophilia and allergic airway hyperresponsiveness by a RORγt inverse agonist
Whitehead, Gregory S, Kang, Hong Soon, Thomas, Seddon Y, Medvedev, Alexander, Karcz, Tadeusz P, Izumi, Gentaro, Nakano, Keiko, Makarov, Sergei S, Nakano, Hideki, Jetten, Anton M, Cook, Donald N
Published in JCI insight (25.07.2019)
Published in JCI insight (25.07.2019)
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Journal Article
Exploration of Alternative Scaffolds for P2Y(14) Receptor Antagonists Containing a Biaryl Core
Jung, Young-Hwan, Yu, Jinha, Wen, Zhiwei, Salmaso, Veronica, Karcz, Tadeusz P., Phung, Ngan B., Chen, Zhoumou, Duca, Sierra, Bennett, John M., Dudas, Steven, Salvemini, Daniela, Gao, Zhan-Guo, Cook, Donald N., Jacobson, Kenneth A.
Published in Journal of medicinal chemistry (10.09.2020)
Published in Journal of medicinal chemistry (10.09.2020)
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Journal Article
Structure-Activity Relationship of Heterocyclic P2Y(14) Receptor Antagonists: Removal of the Zwitterionic Character with Piperidine Bioisosteres
Jung, Young-Hwan, Salmaso, Veronica, Wen, Zhiwei, Bennett, John M., Phung, Ngan B., Lieberman, David, Gopinatth, Varun, Randle, John C. R., Chen, Zhoumou, Salvemini, Daniela, Karcz, Tadeusz P., Cook, Donald N., Jacobson, Kenneth A.
Published in Journal of medicinal chemistry (22.04.2021)
Published in Journal of medicinal chemistry (22.04.2021)
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Journal Article
UDP-glucose and P2Y14 receptor amplify allergen-induced airway eosinophilia
Karcz, Tadeusz P, Whitehead, Gregory S, Nakano, Keiko, Nakano, Hideki, Grimm, Sara A, Williams, Jason G, Deterding, Leesa J, Jacobson, Kenneth A, Cook, Donald N
Published in The Journal of clinical investigation (01.04.2021)
Published in The Journal of clinical investigation (01.04.2021)
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Journal Article
UDP-glucose and [P2Y.sub.14] receptor amplify allergen-induced airway eosinophilia
Karcz, Tadeusz P, Whitehead, Gregory S, Nakano, Keiko, Nakano, Hideki, Grimm, Sara A, Williams, Jason G, Deterding, Leesa J, Jacobson, Kenneth A, Cook, Donald N
Published in The Journal of clinical investigation (01.04.2021)
Published in The Journal of clinical investigation (01.04.2021)
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Journal Article