Ricolinostat (ACY‐1215) induced inhibition of aggresome formation accelerates carfilzomib‐induced multiple myeloma cell death
Mishima, Yuko, Santo, Loredana, Eda, Homare, Cirstea, Diana, Nemani, Neeharika, Yee, Andrew J., O'Donnell, Elizabeth, Selig, Martin Karl, Quayle, Steven N., Arastu‐Kapur, Shirin, Kirk, Christopher, Boise, Lawrence H., Jones, Simon S., Raje, Noopur
Published in British journal of haematology (01.05.2015)
Published in British journal of haematology (01.05.2015)
Get full text
Journal Article
Immunoproteasome functions explained by divergence in cleavage specificity and regulation
Winter, Michael B, La Greca, Florencia, Arastu-Kapur, Shirin, Caiazza, Francesco, Cimermancic, Peter, Buchholz, Tonia J, Anderl, Janet L, Ravalin, Matthew, Bohn, Markus F, Sali, Andrej, O'Donoghue, Anthony J, Craik, Charles S
Published in eLife (28.11.2017)
Published in eLife (28.11.2017)
Get full text
Journal Article
Characterization of P. falciparum dipeptidyl aminopeptidase 3 specificity identifies differences in amino acid preferences between peptide‐based substrates and covalent inhibitors
Vries, Laura E., Sanchez, Mateo I., Groborz, Katarzyna, Kuppens, Laurie, Poreba, Marcin, Lehmann, Christine, Nevins, Neysa, Withers‐Martinez, Chrislaine, Hirst, David J., Yuan, Fang, Arastu‐Kapur, Shirin, Horn, Martin, Mares, Michael, Bogyo, Matthew, Drag, Marcin, Deu, Edgar
Published in The FEBS journal (01.10.2019)
Published in The FEBS journal (01.10.2019)
Get full text
Journal Article
Clinical activity of carfilzomib correlates with inhibition of multiple proteasome subunits: application of a novel pharmacodynamic assay
Lee, Susan J., Levitsky, Konstantin, Parlati, Francesco, Bennett, Mark K., Arastu‐Kapur, Shirin, Kellerman, Lois, Woo, Tina F., Wong, Alvin F., Papadopoulos, Kyriakos P., Niesvizky, Ruben, Badros, Ashraf Z., Vij, Ravi, Jagannath, Sundar, Siegel, David, Wang, Michael, Ahmann, Gregory J., Kirk, Christopher J.
Published in British journal of haematology (01.06.2016)
Published in British journal of haematology (01.06.2016)
Get full text
Journal Article
Nonproteasomal Targets of the Proteasome Inhibitors Bortezomib and Carfilzomib: a Link to Clinical Adverse Events
ARASTU-KAPUR, Shirin, ANDERL, Janet L, KIRK, Christopher J, KRAUS, Marianne, PARLATI, Francesco, SHENK, Kevin D, LEE, Susan J, MUCHAMUEL, Tony, BENNETT, Mark K, DRIESSEN, Christoph, BALL, Andrew J
Published in Clinical cancer research (01.05.2011)
Published in Clinical cancer research (01.05.2011)
Get full text
Journal Article
Treatment of Porphyromonas gulae infection and downstream pathology in the aged dog by lysine‐gingipain inhibitor COR388
Arastu‐Kapur, Shirin, Nguyen, Mai, Raha, Debasish, Ermini, Florian, Haditsch, Ursula, Araujo, Joseph, De Lannoy, Ines A. M., Ryder, Mark I., Dominy, Stephen S., Lynch, Casey, Holsinger, Leslie J.
Published in Pharmacology research & perspectives (01.02.2020)
Published in Pharmacology research & perspectives (01.02.2020)
Get full text
Journal Article
Molecular mechanisms of bortezomib resistant adenocarcinoma cells
Suzuki, Erika, Demo, Susan, Deu, Edgar, Keats, Jonathan, Arastu-Kapur, Shirin, Bergsagel, P Leif, Bennett, Mark K, Kirk, Christopher J
Published in PloS one (22.12.2011)
Published in PloS one (22.12.2011)
Get full text
Journal Article
Discovery of Highly Selective Inhibitors of the Immunoproteasome Low Molecular Mass Polypeptide 2 (LMP2) Subunit
Johnson, Henry W. B, Anderl, Janet L, Bradley, Erin K, Bui, John, Jones, Jeffrey, Arastu-Kapur, Shirin, Kelly, Lisa M, Lowe, Eric, Moebius, David C, Muchamuel, Tony, Kirk, Christopher, Wang, Zhengping, McMinn, Dustin
Published in ACS medicinal chemistry letters (13.04.2017)
Published in ACS medicinal chemistry letters (13.04.2017)
Get full text
Journal Article
Porphyromonas gingivalis in Alzheimer's disease brains: Evidence for disease causation and treatment with small-molecule inhibitors
Dominy, Stephen S, Lynch, Casey, Ermini, Florian, Benedyk, Malgorzata, Marczyk, Agata, Konradi, Andrei, Nguyen, Mai, Haditsch, Ursula, Raha, Debasish, Griffin, Christina, Holsinger, Leslie J, Arastu-Kapur, Shirin, Kaba, Samer, Lee, Alexander, Ryder, Mark I, Potempa, Barbara, Mydel, Piotr, Hellvard, Annelie, Adamowicz, Karina, Hasturk, Hatice, Walker, Glenn D, Reynolds, Eric C, Faull, Richard L M, Curtis, Maurice A, Dragunow, Mike, Potempa, Jan
Published in Science advances (01.01.2019)
Published in Science advances (01.01.2019)
Get full text
Journal Article
Alzheimer's Disease-Like Neurodegeneration in Porphyromonas gingivalis Infected Neurons with Persistent Expression of Active Gingipains
Haditsch, Ursula, Roth, Theresa, Rodriguez, Leo, Hancock, Sandy, Cecere, Thomas, Nguyen, Mai, Arastu-Kapur, Shirin, Broce, Sean, Raha, Debasish, Lynch, Casey C, Holsinger, Leslie J, Dominy, Stephen S, Ermini, Florian
Published in Journal of Alzheimer's disease (01.01.2020)
Published in Journal of Alzheimer's disease (01.01.2020)
Get more information
Journal Article
COR388, a novel gingipain inhibitor, decreases fragmentation of APOE in the central nervous system of Alzheimer’s disease patients: Human/Human trials: Other
Raha, Debasish, Broce, Sean, Haditsch, Ursula, Rodriguez, Leo, Ermini, Florian, Detke, Mike, Kapur, Shirin, Hennings, Dave, Roth, Theresa, Nguyen, Mai, Holsinger, Leslie J., Lynch, Casey C., Dominy, Steve
Published in Alzheimer's & dementia (01.12.2020)
Published in Alzheimer's & dementia (01.12.2020)
Get full text
Journal Article
COR388, a novel gingipain inhibitor, decreases fragmentation of APOE in the central nervous system of Alzheimer’s disease patients
Raha, Debasish, Broce, Sean, Haditsch, Ursula, Rodriguez, Leo, Ermini, Florian, Detke, Mike, Kapur, Shirin, Hennings, Dave, Roth, Theresa, Nguyen, Mai, Holsinger, Leslie J., Lynch, Casey C., Dominy, Steve
Published in Alzheimer's & dementia (01.12.2020)
Published in Alzheimer's & dementia (01.12.2020)
Get full text
Journal Article
Identification of proteases that regulate erythrocyte rupture by the malaria parasite Plasmodium falciparum
Bogyo, Matthew, Arastu-Kapur, Shirin, Ponder, Elizabeth L, Fonovi, Urša Pe ar, Yeoh, Sharon, Yuan, Fang, Fonovi, Marko, Grainger, Munira, Phillips, Carolyn I, Powers, James C
Published in Nature chemical biology (01.03.2008)
Published in Nature chemical biology (01.03.2008)
Get full text
Journal Article