Atypical Responsiveness of the Orphan Receptor GPR55 to Cannabinoid Ligands
Kapur, Ankur, Zhao, Pingwei, Sharir, Haleli, Bai, Yushi, Caron, Marc G., Barak, Larry S., Abood, Mary E.
Published in The Journal of biological chemistry (23.10.2009)
Published in The Journal of biological chemistry (23.10.2009)
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Journal Article
FGF21 Normalizes Plasma Glucose in Mouse Models of Type 1 Diabetes and Insulin Receptor Dysfunction
Diener, John L, Mowbray, Sarah, Huang, Waan-Jeng, Yowe, David, Xu, Jian, Caplan, Shari, Misra, Abhay, Kapur, Ankur, Shapiro, Jeffrey, Ke, Xiaoling, Wu, Xiaoping, Bose, Avirup, Panza, Darrell, Chen, Min, Beaulieu, Valerie, Gao, Jiaping
Published in Endocrinology (Philadelphia) (01.09.2021)
Published in Endocrinology (Philadelphia) (01.09.2021)
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Journal Article
The Endocannabinoids Anandamide and Virodhamine Modulate the Activity of the Candidate Cannabinoid Receptor GPR55
Sharir, Haleli, Console-Bram, Linda, Mundy, Christina, Popoff, Steven N., Kapur, Ankur, Abood, Mary E.
Published in Journal of neuroimmune pharmacology (01.12.2012)
Published in Journal of neuroimmune pharmacology (01.12.2012)
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Journal Article
Mutation Studies of Ser7.39 and Ser2.60 in the Human CB1 Cannabinoid Receptor: Evidence for a Serine-Induced Bend in CB1 Transmembrane Helix 7
Kapur, Ankur, Hurst, Dow P, Fleischer, Daniel, Whitnell, Rob, Thakur, Ganesh A, Makriyannis, Alexandros, Reggio, Patricia H, Abood, Mary E
Published in Molecular pharmacology (01.06.2007)
Published in Molecular pharmacology (01.06.2007)
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Journal Article
Mapping the Structural Requirements in the CB1 Cannabinoid Receptor Transmembrane Helix II for Signal Transduction
Kapur, Ankur, Samaniego, Patrick, Thakur, Ganesh A, Makriyannis, Alexandros, Abood, Mary E
Published in The Journal of pharmacology and experimental therapeutics (01.04.2008)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2008)
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Journal Article
Targeting of the orphan receptor GPR35 by pamoic acid: a potent activator of extracellular signal-regulated kinase and β-arrestin2 with antinociceptive activity
Zhao, Pingwei, Sharir, Haleli, Kapur, Ankur, Cowan, Alan, Geller, Ellen B, Adler, Martin W, Seltzman, Herbert H, Reggio, Patricia H, Heynen-Genel, Susanne, Sauer, Michelle, Chung, Thomas D Y, Bai, Yushi, Chen, Wei, Caron, Marc G, Barak, Larry S, Abood, Mary E
Published in Molecular pharmacology (01.10.2010)
Published in Molecular pharmacology (01.10.2010)
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Journal Article
Novel insights into CB1 cannabinoid receptor signaling: a key interaction identified between the extracellular-3 loop and transmembrane helix 2
Marcu, Jahan, Shore, Derek M, Kapur, Ankur, Trznadel, Megan, Makriyannis, Alexandros, Reggio, Patricia H, Abood, Mary E
Published in The Journal of pharmacology and experimental therapeutics (01.05.2013)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2013)
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Journal Article
Novel Insights into CB 1 Cannabinoid Receptor Signaling: A Key Interaction Identified between the Extracellular-3 Loop and Transmembrane Helix 2
Marcu, Jahan, Shore, Derek M., Kapur, Ankur, Trznadel, Megan, Makriyannis, Alexandros, Reggio, Patricia H., Abood, Mary E.
Published in The Journal of pharmacology and experimental therapeutics (01.05.2013)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2013)
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Journal Article
Novel Insights into CB1 Cannabinoid Receptor Signaling: A Key Interaction Identified between the Extracellular-3 Loop and Transmembrane Helix 2S
Marcu, Jahan, Shore, Derek M., Kapur, Ankur, Trznadel, Megan, Makriyannis, Alexandros, Reggio, Patricia H., Abood, Mary E.
Published in The Journal of pharmacology and experimental therapeutics (01.05.2013)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2013)
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Journal Article
Biarylpyrazole Inverse Agonists at the Cannabinoid CB1 Receptor: Importance of the C-3 Carboxamide Oxygen/Lysine3.28(192) Interaction
Hurst, Dow, Umejiego, Uju, Lynch, Diane, Seltzman, Herbert, Hyatt, Steven, Roche, Michael, McAllister, Sean, Fleischer, Daniel, Kapur, Ankur, Abood, Mary, Shi, Shanping, Jones, Jannie, Lewis, Deborah, Reggio, Patricia
Published in Journal of medicinal chemistry (05.10.2006)
Published in Journal of medicinal chemistry (05.10.2006)
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Journal Article
Mapping the Structural Requirements in the CB 1 Cannabinoid Receptor Transmembrane Helix II for Signal Transduction
Kapur, Ankur, Samaniego, Patrick, Thakur, Ganesh A., Makriyannis, Alexandros, Abood, Mary E.
Published in The Journal of pharmacology and experimental therapeutics (01.04.2008)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2008)
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Journal Article
Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive ActivityS
Zhao, Pingwei, Sharir, Haleli, Kapur, Ankur, Cowan, Alan, Geller, Ellen B., Adler, Martin W., Seltzman, Herbert H., Reggio, Patricia H., Heynen-Genel, Susanne, Sauer, Michelle, Chung, Thomas D.Y., Bai, Yushi, Chen, Wei, Caron, Marc G., Barak, Larry S., Abood, Mary E.
Published in Molecular pharmacology (01.10.2010)
Published in Molecular pharmacology (01.10.2010)
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Journal Article
Mutation Studies of Ser7.39 and Ser2.60 in the Human CB 1 Cannabinoid Receptor: Evidence for a Serine-Induced Bend in CB 1 Transmembrane Helix 7
Kapur, Ankur, Hurst, Dow P., Fleischer, Daniel, Whitnell, Rob, Thakur, Ganesh A., Makriyannis, Alexandros, Reggio, Patricia H., Abood, Mary E.
Published in Molecular pharmacology (01.06.2007)
Published in Molecular pharmacology (01.06.2007)
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Journal Article
Activation of the Torpedo nicotinic acetylcholine receptor
Kapur, Ankur, Davies, Martin, Dryden, William F., Dunn, Susan M.J.
Published in The FEBS journal (01.03.2006)
Published in The FEBS journal (01.03.2006)
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Journal Article
Tryptophan 86 of the α Subunit in the Torpedo Nicotinic Acetylcholine Receptor Is Important for Channel Activation by the Bisquaternary Ligand Suberyldicholine
Kapur, Ankur, Davies, Martin, Dryden, William F, Dunn, Susan M. J
Published in Biochemistry (Easton) (29.08.2006)
Published in Biochemistry (Easton) (29.08.2006)
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Journal Article
Activation of the Torpedo nicotinic acetylcholine receptor: The contribution of residues αArg55 and γGlu93
Kapur, Ankur, Davies, Martin, Dryden, William F., Dunn, Susan M.J.
Published in The FEBS journal (01.03.2006)
Published in The FEBS journal (01.03.2006)
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Journal Article
FGF21 Normalizes Plasma Glucose in Mouse Models of Type 1 Diabetes and Insulin Receptor Dysfunction
Diener, John L, Mowbray, Sarah, Huang, Waan-Jeng, Yowe, David, Xu, Jian, Caplan, Shari, Misra, Abhay, Kapur, Ankur, Shapiro, Jeffrey, Ke, Xiaoling, Wu, Xiaoping, Bose, Avirup, Panza, Darrell, Chen, Min, Beaulieu, Valerie, Gao, Jiaping
Published in bioRxiv (01.02.2021)
Published in bioRxiv (01.02.2021)
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