Quantifying ERK activity in response to inhibition of the BRAFV600E-MEK-ERK cascade using mathematical modelling
Hamis, Sara J., Kapelyukh, Yury, McLaren, Aileen, Henderson, Colin J., Roland Wolf, C., Chaplain, Mark A. J.
Published in British journal of cancer (23.11.2021)
Published in British journal of cancer (23.11.2021)
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Journal Article
Improving the predictive power of xenograft and syngeneic anti-tumour studies using mice humanised for pathways of drug metabolism [version 2; peer review: 2 approved]
Henderson, Colin J., McLaren, Aileen W., Kapelyukh, Yury, Wolf, C. Roland
Published in F1000 research (01.01.2022)
Published in F1000 research (01.01.2022)
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Journal Article
Quantitative prediction of human pregnane X receptor and cytochrome P450 3A4 mediated drug-drug interaction in a novel multiple humanized mouse line
Hasegawa, Maki, Kapelyukh, Yury, Tahara, Harunobu, Seibler, Jost, Rode, Anja, Krueger, Sylvia, Lee, Dongtao N, Wolf, C Roland, Scheer, Nico
Published in Molecular pharmacology (01.09.2011)
Published in Molecular pharmacology (01.09.2011)
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Journal Article
Modeling human cytochrome P450 2D6 metabolism and drug-drug interaction by a novel panel of knockout and humanized mouse lines
Scheer, Nico, Kapelyukh, Yury, McEwan, Jillian, Beuger, Vincent, Stanley, Lesley A, Rode, Anja, Wolf, C Roland
Published in Molecular pharmacology (01.01.2012)
Published in Molecular pharmacology (01.01.2012)
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Journal Article
Defining Human Pathways of Drug Metabolism In Vivo through the Development of a Multiple Humanized Mouse Model
Scheer, Nico, Kapelyukh, Yury, Rode, Anja, Oswald, Stefan, Busch, Diana, McLaughlin, Lesley A, Lin, De, Henderson, Colin J, Wolf, C Roland
Published in Drug metabolism and disposition (01.11.2015)
Published in Drug metabolism and disposition (01.11.2015)
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Journal Article
In Vivo Responses of the Human and Murine Pregnane X Receptor to Dexamethasone in Mice
SCHEER, Nico, ROSS, Jillian, KAPELYUKH, Yury, RODE, Anja, WOLF, C. Roland
Published in Drug metabolism and disposition (01.07.2010)
Published in Drug metabolism and disposition (01.07.2010)
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Journal Article
Multiple Substrate Binding by Cytochrome P450 3A4: Estimation of the Number of Bound Substrate Molecules
KAPELYUKH, Yury, PAINE, Mark J. I, MARECHAL, Jean-Didier, SUTCLIFFE, Michael J, WOLF, C. Roland, ROBERTS, Gordon C. K
Published in Drug metabolism and disposition (01.10.2008)
Published in Drug metabolism and disposition (01.10.2008)
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Journal Article
Abstract 2933: Application of a mouse model humanized for the major pathways of drug disposition in anticancer drug development and use
Henderson, Colin J., Scheer, Nico, Kapelyukh, Yury, McLaren, Aileen, MacLeod, Kenneth, Rode, Anja, Lin, De, Wolf, C Roland
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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Journal Article
Investigations with a humanised CYP3A4/3A7 mouse model
Doyle, Eddie, Coutant, Anne-Laure, Kapelyukh, Yury, Boulenc, Xavier
Published in Toxicology letters (10.09.2014)
Published in Toxicology letters (10.09.2014)
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Journal Article
Improving the predictive power of xenograft and syngeneic anti-tumour studies using mice humanised for pathways of drug metabolism [version 1; peer review: 2 approved with reservations]
Henderson, Colin J., McLaren, Aileen W., Kapelyukh, Yury, Wolf, C. Roland
Published in F1000 research (2022)
Published in F1000 research (2022)
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Journal Article
A role for cytochrome b5 in the In vivo disposition of anticancer and cytochrome P450 probe drugs in mice
Henderson, Colin J, McLaughlin, Lesley A, Finn, Robert D, Ronseaux, Sebastien, Kapelyukh, Yury, Wolf, C Roland
Published in Drug metabolism and disposition (01.01.2014)
Published in Drug metabolism and disposition (01.01.2014)
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Journal Article
A Role for Cytochrome b 5 in the In Vivo Disposition of Anticancer and Cytochrome P450 Probe Drugs in Mice
Henderson, Colin J., McLaughlin, Lesley A., Finn, Robert D., Ronseaux, Sebastien, Kapelyukh, Yury, Wolf, C. Roland
Published in Drug metabolism and disposition (01.01.2014)
Published in Drug metabolism and disposition (01.01.2014)
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Journal Article
A role for cytochrome b5 in the in vivo disposition of anti-cancer and cytochrome P450 probe drugs in mice
Henderson, Colin J., McLaughlin, Lesley A., Finn, Robert D., Ronseaux, Sebastien, Kapelyukh, Yury, Wolf, C. Roland
Published in Drug metabolism and disposition (10.10.2013)
Published in Drug metabolism and disposition (10.10.2013)
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