Modulators of the structural dynamics of the retinoid X receptor to reveal receptor function
Nahoum, Virginie, Pérez, Efrén, Germain, Pierre, Rodríguez-Barrios, Fátima, Manzo, Fabio, Kammerer, Sabrina, Lemaire, Geraldine, Hirsch, Oliver, Royer, Catherine A, Gronemeyer, Hinrich, de Lera, Angel R, Bourguet, William
Published in Proceedings of the National Academy of Sciences - PNAS (30.10.2007)
Published in Proceedings of the National Academy of Sciences - PNAS (30.10.2007)
Get full text
Journal Article
Characterization of the Interaction between Retinoic Acid Receptor/Retinoid X Receptor (RAR/RXR) Heterodimers and Transcriptional Coactivators through Structural and Fluorescence Anisotropy Studies
Pogenberg, Vivian, Guichou, Jean-François, Vivat-Hannah, Valérie, Kammerer, Sabrina, Pérez, Efrén, Germain, Pierre, de Lera, Angel R., Gronemeyer, Hinrich, Royer, Catherine A., Bourguet, William
Published in The Journal of biological chemistry (14.01.2005)
Published in The Journal of biological chemistry (14.01.2005)
Get full text
Journal Article
Rational design of RAR-selective ligands revealed by RARβ crystal stucture
Germain, Pierre, Kammerer, Sabrina, Pérez, Efrén, Peluso-Iltis, Carole, Tortolani, David, Zusi, F Christopher, Starrett, John, Lapointe, Philippe, Daris, Jean-Paul, Marinier, Anne, de Lera, Angel R, Rochel, Natacha, Gronemeyer, Hinrich
Published in EMBO reports (01.09.2004)
Published in EMBO reports (01.09.2004)
Get full text
Journal Article
Silicon Analogues of the Retinoid Agonists TTNPB and 3-Methyl-TTNPB, Disila-TTNPB and Disila-3-methyl-TTNPB: Chemistry and Biology
Büttner, Matthias W., Burschka, Christian, Daiss, Jürgen O., Ivanova, Diana, Rochel, Natacha, Kammerer, Sabrina, Peluso-Iltis, Carole, Bindler, Audrey, Gaudon, Claudine, Germain, Pierre, Moras, Dino, Gronemeyer, Hinrich, Tacke, Reinhold
Published in Chembiochem : a European journal of chemical biology (24.09.2007)
Published in Chembiochem : a European journal of chemical biology (24.09.2007)
Get full text
Journal Article
9- cis-Retinoic acid analogues with bulky hydrophobic rings: new RXR-selective agonists
Alvarez, Rosana, Vega, M. Jesús, Kammerer, Sabrina, Rossin, Aurélie, Germain, Pierre, Gronemeyer, Hinrich, de Lera, Angel R.
Published in Bioorganic & medicinal chemistry letters (20.12.2004)
Published in Bioorganic & medicinal chemistry letters (20.12.2004)
Get full text
Journal Article
RARβ ligand-binding domain bound to an SRC-1 co-activator peptide: purification, crystallization and preliminary X-ray diffraction analysis
Kammerer, Sabrina, Germain, Pierre, Flaig, Ralf, Peluso-Iltis, Carole, Mitschler, André, Rochel, Natacha, Gronemeyer, Hinrich, Moras, Dino
Published in Acta crystallographica. Section D, Biological crystallography. (01.11.2004)
Published in Acta crystallographica. Section D, Biological crystallography. (01.11.2004)
Get full text
Journal Article
Rational design of RAR-selective ligands revealed by RAR[beta] crystal stucture
Germain, Pierre, Kammerer, Sabrina, Pérez, Efrén, Peluso-Iltis, Carole, Tortolani, David, Zusi, F Christopher, Starrett, John, Lapointe, Philippe, Jean-Paul, Daris, Marinier, Anne, de Lera, Angel R, Rochel, Natacha, Gronemeyer, Hinrich
Published in EMBO reports (01.09.2004)
Published in EMBO reports (01.09.2004)
Get full text
Journal Article
Rational design of RAR-selective ligands revealed by RARbeta crystal stucture
Germain, Pierre, Kammerer, Sabrina, Pérez, Efrén, Peluso-Iltis, Carole, Tortolani, David, Zusi, F Christopher, Starrett, John, Lapointe, Philippe, Daris, Jean-Paul, Marinier, Anne, de Lera, Angel R, Rochel, Natacha, Gronemeyer, Hinrich
Published in EMBO reports (01.09.2004)
Published in EMBO reports (01.09.2004)
Get full text
Journal Article
RARbeta ligand-binding domain bound to an SRC-1 co-activator peptide: purification, crystallization and preliminary X-ray diffraction analysis
Kammerer, Sabrina, Germain, Pierre, Flaig, Ralf, Peluso-Iltis, Carole, Mitschler, André, Rochel, Natacha, Gronemeyer, Hinrich, Moras, Dino
Published in Acta crystallographica. Section D, Biological crystallography. (01.11.2004)
Published in Acta crystallographica. Section D, Biological crystallography. (01.11.2004)
Get full text
Journal Article
9-cis-Retinoic Acid Analogues with Bulky Hydrophobic Rings: New RXR-Selective Agonists
Alvarez, Rosana, Vega, M. Jesus, Kammerer, Sabrina, Rossin, Aurelie, Germain, Pierre, Gronemeyer, Hinrich, de Lera, Angel R.
Published in ChemInform (19.04.2005)
Published in ChemInform (19.04.2005)
Get full text
Journal Article