Broadly Applicable and Comprehensive Synthetic Method for N‑Alkyl-Rich Drug-like Cyclic Peptides
Nomura, Kenichi, Hashimoto, Satoshi, Takeyama, Ryuuichi, Tamiya, Minoru, Kato, Tatsuya, Muraoka, Terushige, Kage, Mirai, Nii, Keiji, Kotake, Kenichiro, Iida, Satomi, Emura, Takashi, Tanada, Mikimasa, Iikura, Hitoshi
Published in Journal of medicinal chemistry (13.10.2022)
Published in Journal of medicinal chemistry (13.10.2022)
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Journal Article
Structure-activity relationships of middle-size cyclic peptides, KRAS inhibitors derived from an mRNA display
Kage, Mirai, Hayashi, Ryuji, Matsuo, Atsushi, Tamiya, Minoru, Kuramoto, Shino, Ohara, Kazuhiro, Irie, Machiko, Chiyoda, Aya, Takano, Koji, Ito, Toshiya, Kotake, Tomoya, Takeyama, Ryuuichi, Ishikawa, Shiho, Nomura, Kenichi, Furuichi, Noriyuki, Morita, Yuya, Hashimoto, Satoshi, Kawada, Hatsuo, Nishimura, Yoshikazu, Nii, Keiji, Sase, Hitoshi, Ohta, Atsushi, Kojima, Tetsuo, Iikura, Hitoshi, Tanada, Mikimasa, Shiraishi, Takuya
Published in Bioorganic & medicinal chemistry (01.08.2024)
Published in Bioorganic & medicinal chemistry (01.08.2024)
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Journal Article
HRAS NRAS KRAS PHARMACEUTICAL COMPOSITION COMPRISING CYCLIC COMPOUND HAVING SELECTIVE INHIBITORY ACTION ON KRAS OVER HRAS AND NRAS
KAGE MIRAI, KOTAKE TOMOYA, HASHIMOTO SATOSHI, MORITA YUYA, WAKAMIYA YUMA, HAYASHI RYUJI, TAMIYA MINORU, KAWADA HATSUO, TAKANO KOJI
Year of Publication 10.06.2024
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Year of Publication 10.06.2024
Patent
HRAS 및 NRAS에 대해서 선택적인 KRAS 저해 작용을 갖는 환상 화합물
KAGE MIRAI, KOTAKE TOMOYA, HASHIMOTO SATOSHI, MORITA YUYA, WAKAMIYA YUMA, HAYASHI RYUJI, TAMIYA MINORU, KAWADA HATSUO, TAKANO KOJI
Year of Publication 12.01.2024
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Year of Publication 12.01.2024
Patent
CYCLIC COMPOUND HAVING SELECTIVE KRAS INHIBITORY EFFECT ON HRAS AND NRAS
TAMIYA Minoru, MORITA Yuya, KOTAKE Tomoya, WAKAMIYA Yuma, TAKANO Koji, HASHIMOTO Satoshi, KAGE Mirai, KAWADA Hatsuo, HAYASHI Ryuji
Year of Publication 09.11.2023
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Year of Publication 09.11.2023
Patent
Development of Orally Bioavailable Peptides Targeting an Intracellular Protein: From a Hit to a Clinical KRAS Inhibitor
Tanada, Mikimasa, Tamiya, Minoru, Matsuo, Atsushi, Chiyoda, Aya, Takano, Koji, Ito, Toshiya, Irie, Machiko, Kotake, Tomoya, Takeyama, Ryuuichi, Kawada, Hatsuo, Hayashi, Ryuji, Ishikawa, Shiho, Nomura, Kenichi, Furuichi, Noriyuki, Morita, Yuya, Kage, Mirai, Hashimoto, Satoshi, Nii, Keiji, Sase, Hitoshi, Ohara, Kazuhiro, Ohta, Atsushi, Kuramoto, Shino, Nishimura, Yoshikazu, Iikura, Hitoshi, Shiraishi, Takuya
Published in Journal of the American Chemical Society (02.08.2023)
Published in Journal of the American Chemical Society (02.08.2023)
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Journal Article
CYCLIC COMPOUND HAVING SELECTIVE INHIBITORY ACTION ON KRAS OVER HRAS AND NRAS
WAKAMIYA, Yuma, HAYASHI, Ryuji, HASHIMOTO, Satoshi, TAMIYA, Minoru, KAWADA, Hatsuo, TAKANO, Koji, KAGE, Mirai, KOTAKE, Tomoya, MORITA, Yuya
Year of Publication 16.05.2024
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Year of Publication 16.05.2024
Patent
Cyclic compound having selective inhibitory action on kras over hras and nras
TAMIYA Minoru, MORITA Yuya, KOTAKE Tomoya, WAKAMIYA Yuma, TAKANO Koji, HASHIMOTO Satoshi, KAGE Mirai, KAWADA Hatsuo, HAYASHI Ryuji
Year of Publication 01.12.2023
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Year of Publication 01.12.2023
Patent
CYCLIC COMPOUND HAVING SELECTIVE INHIBITORY ACTION ON KRAS OVER HRAS AND NRAS
KAWADA, HATSUO, MORITA, YUYA, KOTAKE, TOMOYA, WAKAMIYA, YUMA, TAKANO, KOJI, KAGE, MIRAI, HASHIMOTO, SATOSHI, TAMIYA, MINORU, HAYASHI, RYUJI
Year of Publication 10.11.2022
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Year of Publication 10.11.2022
Patent