Total Synthesis of Isokidamycin
O’Keefe, B. Michael, Mans, Douglas M, Kaelin, David E, Martin, Stephen F
Published in Journal of the American Chemical Society (10.11.2010)
Published in Journal of the American Chemical Society (10.11.2010)
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Studies toward the syntheses of pluramycin natural products. The first total synthesis of isokidamycin
O’Keefe, B. Michael, Mans, Douglas M., Kaelin, David E., Martin, Stephen F.
Published in Tetrahedron (02.09.2011)
Published in Tetrahedron (02.09.2011)
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Journal Article
Oxabicyclooctane-Linked Novel Bacterial Topoisomerase Inhibitors as Broad Spectrum Antibacterial Agents
Singh, Sheo B, Kaelin, David E, Wu, Jin, Miesel, Lynn, Tan, Christopher M, Meinke, Peter T, Olsen, David, Lagrutta, Armando, Bradley, Prudence, Lu, Jun, Patel, Sangita, Rickert, Keith W, Smith, Robert F, Soisson, Stephen, Wei, Changqing, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Fukuda, Yasumichi
Published in ACS medicinal chemistry letters (08.05.2014)
Published in ACS medicinal chemistry letters (08.05.2014)
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Journal Article
Tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of left-hand-side moiety (Part-2)
Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Black, Todd, Nargund, Ravi, Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Lu, Jun, Patel, Sangita, Rickert, Keith W., Smith, Robert F., Soisson, Stephen, Sherer, Edward, Joyce, Leo A., Wei, Changqing, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Takano, Hisashi, Shibasaki, Mitsuhito, Yajima, Masanobu, Nishimura, Akinori, Shibata, Takeshi, Fukuda, Yasumichi
Published in Bioorganic & medicinal chemistry letters (01.05.2015)
Published in Bioorganic & medicinal chemistry letters (01.05.2015)
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Journal Article
Hydroxy tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of RHS moiety (Part-3)
Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Gill, Charles, Black, Todd, Nargund, Ravi, Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Wei, Changqing, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Takeuchi, Tomoko, Shibue, Taku, Ohata, Kohei, Takano, Hisashi, Ban, Shizuka, Nishimura, Akinori, Fukuda, Yasumichi
Published in Bioorganic & medicinal chemistry letters (15.06.2015)
Published in Bioorganic & medicinal chemistry letters (15.06.2015)
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Journal Article
Structure activity relationship of C-2 ether substituted 1,5-naphthyridine analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-5)
Singh, Sheo B., Kaelin, David E., Meinke, Peter T., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Olsen, David B., Lagrutta, Armando, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Takeuchi, Tomoko, Takano, Hisashi, Ohata, Kohei, Kurasaki, Haruaki, Nishimura, Akinori, Shibata, Takeshi, Fukuda, Yasumichi
Published in Bioorganic & medicinal chemistry letters (01.09.2015)
Published in Bioorganic & medicinal chemistry letters (01.09.2015)
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Journal Article
Structure activity relationship of pyridoxazinone substituted RHS analogs of oxabicyclooctane-linked 1,5-naphthyridinyl novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-6)
Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Wei, Changqing, Liao, Yonggang, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Yajima, Masanobu, Shibue, Taku, Shibata, Takeshi, Ohata, Kohei, Nishimura, Akinori, Fukuda, Yasumichi
Published in Bioorganic & medicinal chemistry letters (01.09.2015)
Published in Bioorganic & medicinal chemistry letters (01.09.2015)
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Journal Article
Structure activity relationship of substituted 1,5-naphthyridine analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-4)
Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Wei, Changqing, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Shibata, Takeshi, Ohata, Kohei, Takano, Hisashi, Kurasaki, Haruaki, Takeuchi, Tomoko, Nishimura, Akinori, Fukuda, Yasumichi
Published in Bioorganic & medicinal chemistry letters (01.06.2015)
Published in Bioorganic & medicinal chemistry letters (01.06.2015)
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Journal Article
General Strategies for the Synthesis of the Major Classes of C-Aryl Glycosides
Kaelin, David E, Lopez, Omar D, Martin, Stephen F
Published in Journal of the American Chemical Society (18.07.2001)
Published in Journal of the American Chemical Society (18.07.2001)
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Journal Article
C1–C2-linker substituted 1,5-naphthyridine analogues of oxabicyclooctane-linked NBTIs as broad-spectrum antibacterial agents (part 7)
Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Wei, Changqing, Liao, Yonggang, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Shibata, Takeshi, Takeuchi, Tomoko, Ohata, Kohei, Nishimura, Akinori, Fukuda, Yasumichi
Published in MedChemComm (01.01.2015)
Published in MedChemComm (01.01.2015)
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Journal Article
Application of Ring-Closing Metathesis to the Formal Total Synthesis of (+)−FR900482
Fellows, Ingrid M, Kaelin, David E, Martin, Stephen F
Published in Journal of the American Chemical Society (08.11.2000)
Published in Journal of the American Chemical Society (08.11.2000)
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Journal Article
General entries to C-aryl glycosides. Formal synthesis of galtamycinone
Apsel, Beth, Bender, John A, Escobar, Maya, Kaelin, David E, Lopez, Omar D, Martin, Stephen F
Published in Tetrahedron letters (27.01.2003)
Published in Tetrahedron letters (27.01.2003)
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Journal Article
4-Arylcyclohexylalanine analogs as potent, selective, and orally active inhibitors of dipeptidyl peptidase IV
Kaelin, David E., Smenton, Abigail L., Eiermann, George J., He, Huaibing, Leiting, Barbara, Lyons, Kathryn A., Patel, Reshma A., Patel, Sangita B., Petrov, Alexsandr, Scapin, Giovanna, Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E., Duffy, Joseph L.
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
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Journal Article
Total Synthesis of (+)-Ambruticin S
Kirkland, Thomas A, Colucci, John, Geraci, Leo S, Marx, Matthew A, Schneider, Matthias, Kaelin, David E, Martin, Stephen F
Published in Journal of the American Chemical Society (12.12.2001)
Published in Journal of the American Chemical Society (12.12.2001)
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Journal Article
Extension of ASM3 for two-step nitrification and denitrification and its calibration and validation with batch tests and pilot scale data
Kaelin, David, Manser, Reto, Rieger, Leiv, Eugster, Jack, Rottermann, Karin, Siegrist, Hansruedi
Published in Water research (Oxford) (01.04.2009)
Published in Water research (Oxford) (01.04.2009)
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Journal Article
Structure activity relationship of N-1 substituted 1,5-naphthyrid-2-one analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents (Part-9)
Singh, Sheo B., Tan, Christopher M., Kaelin, David, Meinke, Peter T., Miesel, Lynn, Olsen, David B., Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Ohata, Kohei, Takeuchi, Tomoko, Shibue, Taku, Takano, Hisashi, Nishimura, Akinori, Fukuda, Yasumichi
Published in Bioorganic & medicinal chemistry letters (01.11.2022)
Published in Bioorganic & medicinal chemistry letters (01.11.2022)
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