Innovative Randomized Phase I Study and Dosing Regimen Selection to Accelerate and Inform Pivotal COVID‐19 Trial of Nirmatrelvir
Singh, Ravi Shankar P., Toussi, Sima S., Hackman, Frances, Chan, Phylinda L., Rao, Rohit, Allen, Richard, Van Eyck, Lien, Pawlak, Sylvester, Kadar, Eugene P., Clark, Frances, Shi, Haihong, Anderson, Annaliesa S., Binks, Michael, Menon, Sandeep, Nucci, Gianluca, Bergman, Arthur
Published in Clinical pharmacology and therapeutics (01.07.2022)
Published in Clinical pharmacology and therapeutics (01.07.2022)
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Journal Article
Disposition of Nirmatrelvir, an Orally Bioavailable Inhibitor of SARS-CoV-2 3C-Like Protease, across Animals and Humans
Eng, Heather, Dantonio, Alyssa L, Kadar, Eugene P, Obach, R Scott, Di, Li, Lin, Jian, Patel, Nandini C, Boras, Britton, Walker, Gregory S, Novak, Jonathan J, Kimoto, Emi, Singh, Ravi Shankar P, Kalgutkar, Amit S
Published in Drug metabolism and disposition (01.05.2022)
Published in Drug metabolism and disposition (01.05.2022)
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Journal Article
Reduction of in-source collision-induced dissociation and thermolysis of sulopenem prodrugs for quantitative liquid chromatography/electrospray ionization mass spectrometric analysis by promoting sodium adduct formation
Wujcik, Chad E., Kadar, Eugene P.
Published in Rapid communications in mass spectrometry (30.10.2008)
Published in Rapid communications in mass spectrometry (30.10.2008)
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Journal Article
Remediation of undesirable secondary interactions encountered in hydrophilic interaction chromatography during development of a quantitative LC–MS/MS assay for a dipeptidyl peptidase IV (DPP-IV) inhibitor in monkey serum
Kadar, Eugene P., Wujcik, Chad E.
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (15.02.2009)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (15.02.2009)
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Journal Article
Rapid determination of the applicability of hydrophilic interaction chromatography utilizing ACD Labs Log D Suite: A bioanalytical application
Kadar, Eugene P., Wujcik, Chad E., Wolford, David P., Kavetskaia, Olga
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (15.02.2008)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (15.02.2008)
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Journal Article
Metabolism and Excretion of Nirmatrelvir in Humans Using Quantitative Fluorine Nuclear Magnetic Resonance Spectroscopy: A Novel Approach for Accelerating Drug Development
Singh, Ravi Shankar P, Walker, Gregory S, Kadar, Eugene P, Cox, Loretta M, Eng, Heather, Sharma, Raman, Bergman, Arthur J, Van Eyck, Lien, Hackman, Frances, Toussi, Sima S, Kalgutkar, Amit S, Obach, R Scott
Published in Clinical pharmacology and therapeutics (01.12.2022)
Published in Clinical pharmacology and therapeutics (01.12.2022)
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Journal Article
A Novel Milli-fluidic Liver Tissue Chip with Continuous Recirculation for Predictive Pharmacokinetics Applications
Rajan, Shiny Amala Priya, Sherfey, Jason, Ohri, Shivam, Nichols, Lauren, Smith, J. Tyler, Parekh, Paarth, Kadar, Eugene P., Clark, Frances, George, Billy T., Gregory, Lauren, Tess, David, Gosset, James R., Liras, Jennifer, Geishecker, Emily, Obach, R. Scott, Cirit, Murat
Published in The AAPS journal (01.11.2023)
Published in The AAPS journal (01.11.2023)
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Journal Article
Scheduling distributed energy resources in an isolated grid - An artificial neural network approach
Vale, Z A, Faria, P, Morais, H, Khodr, H M, Silva, M, Kadar, P
Published in IEEE PES General Meeting (01.07.2010)
Published in IEEE PES General Meeting (01.07.2010)
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Conference Proceeding
Correction: A Novel Milli-fluidic Liver Tissue Chip with Continuous Recirculation for Predictive Pharmacokinetics Applications
Rajan, Shiny Amala Priya, Sherfey, Jason, Ohri, Shivam, Nichols, Lauren, Smith, J. Tyler, Parekh, Paarth, Kadar, Eugene P., Clark, Frances, George, Billy T., Gregory, Lauren, Tess, David, Gosset, James R., Liras, Jennifer, Geishecker, Emily, Obach, R. Scott, Cirit, Murat
Published in The AAPS journal (20.11.2023)
Published in The AAPS journal (20.11.2023)
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Journal Article
Estimation of Circulating Drug Metabolite Exposure in Human Using In Vitro Data and Physiologically Based Pharmacokinetic Modeling: Example of a High Metabolite/Parent Drug Ratio
Obach, R Scott, Lin, Jian, Kimoto, Emi, Duvvuri, Sridhar, Nicholas, Timothy, Kadar, Eugene P, Tremaine, Larry M, Sawant-Basak, Aarti
Published in Drug metabolism and disposition (01.02.2018)
Published in Drug metabolism and disposition (01.02.2018)
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Journal Article
An oral SARS-CoV-2 M pro inhibitor clinical candidate for the treatment of COVID-19
Owen, Dafydd R, Allerton, Charlotte M N, Anderson, Annaliesa S, Aschenbrenner, Lisa, Avery, Melissa, Berritt, Simon, Boras, Britton, Cardin, Rhonda D, Carlo, Anthony, Coffman, Karen J, Dantonio, Alyssa, Di, Li, Eng, Heather, Ferre, RoseAnn, Gajiwala, Ketan S, Gibson, Scott A, Greasley, Samantha E, Hurst, Brett L, Kadar, Eugene P, Kalgutkar, Amit S, Lee, Jack C, Lee, Jisun, Liu, Wei, Mason, Stephen W, Noell, Stephen, Novak, Jonathan J, Obach, R Scott, Ogilvie, Kevin, Patel, Nandini C, Pettersson, Martin, Rai, Devendra K, Reese, Matthew R, Sammons, Matthew F, Sathish, Jean G, Singh, Ravi Shankar P, Steppan, Claire M, Stewart, Al E, Tuttle, Jamison B, Updyke, Lawrence, Verhoest, Patrick R, Wei, Liuqing, Yang, Qingyi, Zhu, Yuao
Published in Science (American Association for the Advancement of Science) (24.12.2021)
Published in Science (American Association for the Advancement of Science) (24.12.2021)
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Journal Article
Guidelines for Selecting Surfacing Alternatives for Unsealed Roads
Henning, T. F. P., Bennett, C. R., Kadar, P.
Published in Transportation research record (01.01.2007)
Published in Transportation research record (01.01.2007)
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Journal Article
PhotoVoltaic EV charge station
Kadar, P., Varga, A.
Published in 2013 IEEE 11th International Symposium on Applied Machine Intelligence and Informatics (SAMI) (01.01.2013)
Published in 2013 IEEE 11th International Symposium on Applied Machine Intelligence and Informatics (SAMI) (01.01.2013)
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Conference Proceeding
Journal Article
Accumulation of uranium, transuranium and fission products on stainless steel surfaces II. Sorption studies in a laboratory model system
Kádár, P., Varga, K., Baja, B., Németh, Z., Vajda, N., Stefánka, Zs, Kövér, L., Cserny, I., Tóth, J., Pintér, T., Schunk, J.
Published in Journal of radioanalytical and nuclear chemistry (01.06.2011)
Published in Journal of radioanalytical and nuclear chemistry (01.06.2011)
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Journal Article
Long-term trends in the corrosion state and surface properties of the stainless steel tubes of steam generators decontaminated chemically in VVER-type nuclear reactors
Baja, B., Varga, K., Szabó, N.A., Németh, Z., Kádár, P., Oravetz, D., Homonnay, Z., Kuzmann, E., Schunk, J., Patek, G.
Published in Corrosion science (01.12.2009)
Published in Corrosion science (01.12.2009)
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Journal Article
Accumulation of uranium, transuranium and fission products on stainless steel surfaces. I. A comprehensive view of the experimental parameters influencing the extent and character of the contamination
Kádár, P., Varga, K., Németh, Z., Vajda, N., Pintér, T., Schunk, J.
Published in Journal of radioanalytical and nuclear chemistry (01.05.2010)
Published in Journal of radioanalytical and nuclear chemistry (01.05.2010)
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Journal Article