ORY-1001, a Potent and Selective Covalent KDM1A Inhibitor, for the Treatment of Acute Leukemia
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Published in The Journal of biological chemistry (09.10.2009)
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Fragment-hopping-based discovery of a novel chemical series of proto-oncogene PIM-1 kinase inhibitors
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Published in PloS one (24.10.2012)
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Martín-Sánchez, Esperanza, Rodríguez-Pinilla, Socorro M, Sánchez-Beato, Margarita, Lombardía, Luis, Domínguez-González, Beatriz, Romero, Diana, Odqvist, Lina, García-Sanz, Pablo, Wozniak, Magdalena B, Kurz, Guido, Blanco-Aparicio, Carmen, Mollejo, Manuela, Alves, F Javier, Menárguez, Javier, González-Palacios, Fernando, Rodríguez-Peralto, José Luis, Ortiz-Romero, Pablo L, García, Juan F, Bischoff, James R, Piris, Miguel A
Published in Haematologica (Roma) (01.01.2013)
Published in Haematologica (Roma) (01.01.2013)
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항종양 아스코르브산 에스테르
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Year of Publication 20.06.2023
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Year of Publication 20.06.2023
Patent
Preclinical characterization of a potent and selective inhibitor of the histone demethylase KDM1A for MLL leukemia
Maes, Tamara, Tirapu, Iñigo, Mascaró, Cristina, Ortega, Alberto, Estiarte, Angels, Valls, Nuria, Castro-Palomino, Julio, Buesa Arjol, Carlos, Kurz, Guido
Published in Journal of clinical oncology (20.05.2013)
Published in Journal of clinical oncology (20.05.2013)
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Arylsulfonamidothiazoles as a New Class of Potential Antidiabetic Drugs. Discovery of Potent and Selective Inhibitors of the 11β-Hydroxysteroid Dehydrogenase Type 1
Barf, Tjeerd, Vallgårda, Jerk, Emond, Rikard, Häggström, Charlotta, Kurz, Guido, Nygren, Alf, Larwood, Vivienne, Mosialou, Erifili, Axelsson, Kent, Olsson, Rolf, Engblom, Lars, Edling, Naimie, Rönquist-Nii, Yuko, Öhman, Birgitta, Alberts, Peteris, Abrahmsén, Lars
Published in Journal of medicinal chemistry (29.08.2002)
Published in Journal of medicinal chemistry (29.08.2002)
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