Bioisosteric approach to the discovery of imidazo[1,2-a]pyrazines as potent Aurora kinase inhibitors
Meng, Zhaoyang, Kulkarni, Bheemashankar A., Kerekes, Angela D., Mandal, Amit K., Esposite, Sara J., Belanger, David B., Reddy, Panduranga Adulla, Basso, Andrea D., Tevar, Seema, Gray, Kimberly, Jones, Jennifer, Smith, Elizabeth B., Doll, Ronald J., Siddiqui, M. Arshad
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Get full text
Journal Article
Exploring Chemical Diversity of Epoxyquinoid Natural Products: Synthesis and Biological Activity of (−)-Jesterone and Related Molecules
Hu, Yongbo, Li, Chaomin, Kulkarni, Bheemashankar A, Strobel, Gary, Lobkovsky, Emil, Torczynski, Richard M, Porco, John A
Published in Organic letters (31.05.2001)
Published in Organic letters (31.05.2001)
Get full text
Journal Article
A selenide linker for "traceless" solid-phase organic synthesis
Li, Zhengong, Kulkarni, Bheemashankar A., Ganesan, A.
Published in Biotechnology and bioengineering (2000)
Published in Biotechnology and bioengineering (2000)
Get full text
Journal Article
A New Series of Orally Bioavailable Chemokine Receptor 9 (CCR9) Antagonists; Possible Agents for the Treatment of Inflammatory Bowel Disease
Kalindjian, S. Barret, Kadnur, Sanjay V, Hewson, Christopher A, Venkateshappa, Chandregowda, Juluri, Suresh, Kristam, Rajendra, Kulkarni, Bheemashankar, Mohammed, Zainuddin, Saxena, Rohit, Viswanadhan, Vellarkad N, Aiyar, Jayashree, McVey, Donna
Published in Journal of medicinal chemistry (14.04.2016)
Published in Journal of medicinal chemistry (14.04.2016)
Get full text
Journal Article
Discovery and pharmacological evaluation of indole derivatives as potent and selective RORγt inverse agonist for multiple autoimmune conditions
Shaikh, Nadim S., Iyer, Jitesh P., Munot, Yogesh S., Mukhopadhyay, Partha P., Raje, Amol A., Nagaraj, Ranganayaki, Jamdar, Vijay, Gavhane, Ravindra, Lohote, Mahendra, Sherkar, Prasad, Bala, Madhu, Petla, Rajkanth, Meru, Ashwinkumar, Umrani, Dhananjay, Rouduri, Sreekanth, Joshi, Sachin, Reddy, Satyanarayan, Kandikere, Vishwottam, Bhuniya, Debnath, Kulkarni, Bheemashankar, Mookhtiar, Kasim A.
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
Get full text
Journal Article
Discovery and evaluation of 1H-pyrrolo[2,3-b]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis
Thakkar, Mahesh, Bhuniya, Debnath, Kaduskar, Rahul, Mengawade, Tanaji, Naik, Keshav, Salunkhe, Videsh, Bhalerao, Amit, Kurhade, Santosh, Mavinahalli, Jagadeesh, Jain, Vaibhav, Petla, Rajkanth, Avaragolla, Satheesh, Ray, Swagatam, Rouduri, Sreekanth, Dhanave, Avinash, De, Siddhartha, Pathade, Vishal, Tambe, Ashwini, Raje, Amol A., Madgula, Vamsi, Joshi, Sachin, Nadeem, Ahmed, bala, Madhu, Umrani, Dhananjay, Hariharan, Narayanan, Kulkarni, Bheemashankar, Mookhtiar, Kasim A.
Published in Bioorganic & medicinal chemistry letters (15.04.2017)
Published in Bioorganic & medicinal chemistry letters (15.04.2017)
Get full text
Journal Article
Discovery and optimization of N-acyl and N-aroylpyrazolines as B-Raf kinase inhibitors
Blackburn, Christopher, Duffey, Matthew O., Gould, Alexandra E., Kulkarni, Bheemashankar, Liu, Jane X., Menon, Saurabh, Nagayoshi, Masayuki, Vos, Tricia J., Williams, Juliet
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
Get full text
Journal Article
Discovery and evaluation of 1 H -pyrrolo[2,3- b ]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis
Thakkar, Mahesh, Bhuniya, Debnath, Kaduskar, Rahul, Mengawade, Tanaji, Naik, Keshav, Salunkhe, Videsh, Bhalerao, Amit, Kurhade, Santosh, Mavinahalli, Jagadeesh, Jain, Vaibhav, Petla, Rajkanth, Avaragolla, Satheesh, Ray, Swagatam, Rouduri, Sreekanth, Dhanave, Avinash, De, Siddhartha, Pathade, Vishal, Tambe, Ashwini, Raje, Amol A., Madgula, Vamsi, Joshi, Sachin, Nadeem, Ahmed, bala, Madhu, Umrani, Dhananjay, Hariharan, Narayanan, Kulkarni, Bheemashankar, Mookhtiar, Kasim A.
Published in Bioorganic & medicinal chemistry letters (01.04.2017)
Published in Bioorganic & medicinal chemistry letters (01.04.2017)
Get full text
Journal Article
삼환식 화합물, 삼환식 화합물을 포함하는 조성물 및 이의 의약적 용도
PATEL MEENA, BONAGIRI RAJESH, MOOKHTIAR KASIM, KULKARNI BHEEMASHANKAR, BASU SUJAY, KHOSE GORAKSHA, BARAWKAR DINESH, SHEJUL YOGESH, THORAT SACHIN, PANMAND ANIL
Year of Publication 11.09.2020
Get full text
Year of Publication 11.09.2020
Patent
Discovery of a Potent and Orally Bioavailable Benzolactam-Derived Inhibitor of Polo-Like Kinase 1 (MLN0905)
Duffey, Matthew O, Vos, Tricia J, Adams, Ruth, Alley, Jennifer, Anthony, Justin, Barrett, Cynthia, Bharathan, Indu, Bowman, Douglas, Bump, Nancy J, Chau, Ryan, Cullis, Courtney, Driscoll, Denise L, Elder, Amy, Forsyth, Nancy, Frazer, Jonathan, Guo, Jianping, Guo, Luyi, Hyer, Marc L, Janowick, David, Kulkarni, Bheemashankar, Lai, Su-Jen, Lasky, Kerri, Li, Gang, Li, Jing, Liao, Debra, Little, Jeremy, Peng, Bo, Qian, Mark G, Reynolds, Dominic J, Rezaei, Mansoureh, Scott, Margaret Porter, Sells, Todd B, Shinde, Vaishali, Shi, Qiuju Judy, Sintchak, Michael D, Soucy, Francois, Sprott, Kevin T, Stroud, Stephen G, Nestor, Michelle, Visiers, Irache, Weatherhead, Gabriel, Ye, Yingchun, D’Amore, Natalie
Published in Journal of medicinal chemistry (12.01.2012)
Published in Journal of medicinal chemistry (12.01.2012)
Get full text
Journal Article
Design and Optimization of Potent and Orally Bioavailable Tetrahydronaphthalene Raf Inhibitors
Gould, Alexandra E, Adams, Ruth, Adhikari, Sharmila, Aertgeerts, Kathleen, Afroze, Roushan, Blackburn, Christopher, Calderwood, Emily F, Chau, Ryan, Chouitar, Jouhara, Duffey, Matthew O, England, Dylan B, Farrer, Cheryl, Forsyth, Nancy, Garcia, Khristofer, Gaulin, Jeffery, Greenspan, Paul D, Guo, Ribo, Harrison, Sean J, Huang, Shih-Chung, Iartchouk, Natalia, Janowick, Dave, Kim, Mi-Sook, Kulkarni, Bheemashankar, Langston, Steven P, Liu, Jane X, Ma, Li-Ting, Menon, Saurabh, Mizutani, Hirotake, Paske, Erin, Renou, Christelle C, Rezaei, Mansoureh, Rowland, R. Scott, Sintchak, Michael D, Smith, Michael D, Stroud, Stephen G, Tregay, Ming, Tian, Yuan, Veiby, Ole P, Vos, Tricia J, Vyskocil, Stepan, Williams, Juliet, Xu, Tianlin, Yang, Johnny J, Yano, Jason, Zeng, Hongbo, Zhang, Dong Mei, Zhang, Qin, Galvin, Katherine M
Published in Journal of medicinal chemistry (24.03.2011)
Published in Journal of medicinal chemistry (24.03.2011)
Get full text
Journal Article
Discovery and optimization of pyrazoline compounds as B-Raf inhibitors
Duffey, Matthew O., Adams, Ruth, Blackburn, Christopher, Chau, Ryan W., Chen, Susan, Galvin, Katherine M., Garcia, Khristofer, Gould, Alexandra E., Greenspan, Paul D., Harrison, Sean, Huang, Shih-Chung, Kim, Mi-Sook, Kulkarni, Bheemashankar, Langston, Steven, Liu, Jane X., Ma, Li-Ting, Menon, Saurabh, Nagayoshi, Masayuki, Rowland, R. Scott, Vos, Tricia J., Xu, Tianlin, Yang, Johnny J., Yu, Shaoxia, Zhang, Qin
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
Get full text
Journal Article