Search Results - "KUANG RONGZE" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Discovery of a Novel Class of Orally Active Antifungal β-1,3-d-Glucan Synthase Inhibitors

Discovery of a Novel Class of Orally Active Antifungal β-1,3-d-Glucan Synthase Inhibitors

by WALKER, Scott S, YIMING XU, NORRIS, Christine, ANTONACCI, Barry, GURNANI, Maya, CACCIAPUOTI, Anthony, MCNICHOLAS, Paul M, WAINHAUS, Samuel, JASON HERR, R, KUANG, Rongze, ASLANIAN, Robert G, TING, Pauline C, TRIANTAFYLLOU, Ilias, BLACK, Todd A, WALDMAN, Michelle F, MENDRICK, Cara, BROWN, Nathaniel, MANN, Paul, CHAU, Andrew, PATEL, Reena, BAUMAN, Nicholas
Published in Antimicrobial Agents and Chemotherapy (01.11.2011)

Get full text

Journal Article

Discovery of oxazole-based PDE4 inhibitors with picomolar potency

Discovery of oxazole-based PDE4 inhibitors with picomolar potency

by Kuang, Rongze, Shue, Ho-Jane, Xiao, Li, Blythin, David J., Shih, Neng-Yang, Chen, Xiao, Gu, Danlin, Schwerdt, John, Lin, Ling, Ting, Pauline C., Cao, Jianhua, Aslanian, Robert, Piwinski, John J., Prelusky, Daniel, Wu, Ping, Zhang, Ji, Zhang, Xiang, Celly, Chander S., Billah, Motasim, Wang, Peng
Published in Bioorganic & medicinal chemistry letters (01.04.2012)

Get full text

Journal Article

SAR studies of pyridazinone derivatives as novel glucan synthase inhibitors

SAR studies of pyridazinone derivatives as novel glucan synthase inhibitors

by Zhou, Gang, Ting, Pauline C., Aslanian, Robert, Cao, Jianhua, Kim, David W., Kuang, Rongze, Lee, Joe F., Schwerdt, John, Wu, Heping, Jason Herr, R., Zych, Andrew J., Yang, Jinhai, Lam, Sang, Wainhaus, Samuel, Black, Todd A., McNicholas, Paul M., Xu, Yiming, Walker, Scott S.
Published in Bioorganic & medicinal chemistry letters (15.05.2011)

Get full text

Journal Article

The synthesis and structure–activity relationship of pyridazinones as glucan synthase inhibitors

The synthesis and structure–activity relationship of pyridazinones as glucan synthase inhibitors

by Ting, Pauline C., Kuang, Rongze, Wu, Heping, Aslanian, Robert G., Cao, Jianhua, Kim, David W., Lee, Joe F., Schwerdt, John, Zhou, Gang, Wainhaus, Samuel, Black, Todd A., Cacciapuoti, Anthony, McNicholas, Paul M., Xu, Yiming, Walker, Scott S.
Published in Bioorganic & medicinal chemistry letters (15.03.2011)

Get full text

Journal Article

Lead optimization of a sulfonylurea-based piperazine pyridazinone series of glucan synthase inhibitors

Lead optimization of a sulfonylurea-based piperazine pyridazinone series of glucan synthase inhibitors

by Zych, Andrew J., Lam, Sang Q., Jenkins, David M., Herr, R. Jason, Ting, Pauline C., Lee, Joe F., Kuang, Rongze, Wu, Heping, Kim, David W., Aslanian, Robert G., Wainhaus, Samuel, Black, Todd A., Cacciapuoti, Anthony, McNicholas, Paul M., Xu, Yiming, Walker, Scott S.
Published in Bioorganic & medicinal chemistry letters (15.07.2012)

Get full text

Journal Article

The optimization of pyridazinone series of glucan synthase inhibitors

The optimization of pyridazinone series of glucan synthase inhibitors

by Kuang, Rongze, Wu, Heping, Ting, Pauline C., Aslanian, Robert G., Cao, Jianhua, Kim, David W., Lee, Joe F., Schwerdt, John, Zhou, Gang, Jason Herr, R., Zych, Andrew J., Yang, Jinhai, Lam, Sang Q., Jenkins, David M., Sakwa, Samuel A., Wainhaus, Samuel, Black, Todd A., Cacciapuoti, Anthony, McNicholas, Paul M., Xu, Yiming, Walker, Scott S.
Published in Bioorganic & medicinal chemistry letters (15.08.2012)

Get full text

Journal Article

Effects of structure on inhibitory activity in a series of mechanism-based inhibitors of human neutrophil elastase

Effects of structure on inhibitory activity in a series of mechanism-based inhibitors of human neutrophil elastase

by Dou, Dengfeng, He, Guijia, Kuang, Rongze, Fu, Qingfong, Venkataraman, Radhika, Groutas, William C.
Published in Bioorganic & medicinal chemistry (15.09.2010)

Get full text

Journal Article

Structure-Based Design of a General Class of Mechanism-Based Inhibitors of the Serine Proteinases Employing a Novel Amino Acid-Derived Heterocyclic Scaffold

Structure-Based Design of a General Class of Mechanism-Based Inhibitors of the Serine Proteinases Employing a Novel Amino Acid-Derived Heterocyclic Scaffold

by Groutas, William C, Kuang, Rongze, Venkataraman, Radhika, Epp, Jeffrey B, Ruan, Sumei, Prakash, Om
Published in Biochemistry (Easton) (22.04.1997)

Get full text

Journal Article

Potent inhibition of serine proteases by heterocyclic sulfide derivatives of 1,2,5-thiadiazolidin-3-one 1,1 dioxide

Potent inhibition of serine proteases by heterocyclic sulfide derivatives of 1,2,5-thiadiazolidin-3-one 1,1 dioxide

by SHU HE, RONGZE KUANG, VENKATARAMAN, R, JUAN TU, TRUONG, T. M, CHAN, H.-K, GROUTAS, W. C
Published in Bioorganic & medicinal chemistry (01.07.2000)

Get full text

Journal Article

Inhibition of serine proteases by functionalized sulfonamides coupled to the 1,2,5-thiadiazolidin-3-one 1,1 dioxide scaffold

Inhibition of serine proteases by functionalized sulfonamides coupled to the 1,2,5-thiadiazolidin-3-one 1,1 dioxide scaffold

by Groutas, William C, He, Shu, Kuang, Rongze, Ruan, Sumei, Tu, Juan, Chan, Ho-Kit
Published in Bioorganic & medicinal chemistry (01.06.2001)

Get full text

Journal Article

Utilization of the 1,2,5-thiadiazolidin-3-one 1,1 dioxide scaffold in the design of potent inhibitors of serine proteases: SAR studies using carboxylates

Utilization of the 1,2,5-thiadiazolidin-3-one 1,1 dioxide scaffold in the design of potent inhibitors of serine proteases: SAR studies using carboxylates

by RONGZE KUANG, EPP, J. B, SUMEI RUAN, CHONG, L. S, VENKATARAMAN, R, JUAN TU, SHU HE, TRUONG, T. M, GROUTAS, W. C
Published in Bioorganic & medicinal chemistry (01.05.2000)

Get full text

Journal Article

Inhibition of Escherichia coli by dimethyl fumarate

Inhibition of Escherichia coli by dimethyl fumarate

by Wang, Hai-Hong, Sun, Da-Wen, Kuang, Rongze
Published in International journal of food microbiology (11.04.2001)

Get full text

Journal Article

Use of the 1,2,5-thiadiazolidin-3-one 1,1 dioxide and isothiazolidin-3-one 1,1 dioxide scaffolds in the design of potent inhibitors of serine proteinases

Use of the 1,2,5-thiadiazolidin-3-one 1,1 dioxide and isothiazolidin-3-one 1,1 dioxide scaffolds in the design of potent inhibitors of serine proteinases

by Kuang, Rongze, Venkataraman, Radhika, Ruan, Sumei, Groutas, William C.
Published in Bioorganic & medicinal chemistry letters (03.03.1998)

Get full text

Journal Article

Substituted 3-oxo-1,2,5-Thiadiazolidine 1,1-Dioxides: A New Class of Potential Mechanism-Based Inhibitors of Human Leukocyte Elastase and Cathepsin G

Substituted 3-oxo-1,2,5-Thiadiazolidine 1,1-Dioxides: A New Class of Potential Mechanism-Based Inhibitors of Human Leukocyte Elastase and Cathepsin G

by Groutas, W.C., Kuang, R.Z., Venkataraman, R.
Published in Biochemical and biophysical research communications (14.01.1994)

Get full text

Journal Article

Discovery of aminoquinazoline derivatives as human A(2A) adenosine receptor antagonists

Discovery of aminoquinazoline derivatives as human A(2A) adenosine receptor antagonists

by Zhou, Gang, Aslanian, Robert, Gallo, Gioconda, Khan, Tanweer, Kuang, Rongze, Purakkattle, Biju, De Ruiz, Manuel, Stamford, Andrew, Ting, Pauline, Wu, Heping, Wang, Hongwu, Xiao, Dong, Yu, Tao, Zhang, Yonglian, Mullins, Deborra, Hodgson, Robert
Published in Bioorganic & medicinal chemistry letters (15.02.2016)

Get full text

Journal Article

Discovery of aminoquinazoline derivatives as human A2A adenosine receptor antagonists

Discovery of aminoquinazoline derivatives as human A2A adenosine receptor antagonists

by Zhou, Gang, Aslanian, Robert, Gallo, Gioconda, Khan, Tanweer, Kuang, Rongze, Purakkattle, Biju, Ruiz, Manuel De, Stamford, Andrew, Ting, Pauline, Wu, Heping, Wang, Hongwu, Xiao, Dong, Yu, Tao, Zhang, Yonglian, Mullins, Deborra, Hodgson, Robert
Published in Bioorganic & medicinal chemistry letters (15.02.2016)

Get full text

Journal Article

혈장 칼리크레인 억제제

혈장 칼리크레인 억제제

by ZHAO ZHIQIANG, MERCHANT ROHAN, SHARP PHILLIP PATRICK, BAO JIANMING, SINZ CHRISTOPHER J, CHENG ALAN C, KUANG RONGZE, SHEARN NANCE GALEN PAUL, HICKS JACQUELINE D, LOMBARDO MATTHEW J, LOPEZ JOVAN ALEXANDER, TIAN MAOQUN, YANG SONG, WU ZHICAI
Year of Publication 20.03.2023

Get full text

Patent

Discovery of aminoquinazoline derivatives as human A sub(2A) adenosine receptor antagonists

Discovery of aminoquinazoline derivatives as human A sub(2A) adenosine receptor antagonists

by Zhou, Gang, Aslanian, Robert, Gallo, Gioconda, Khan, Tanweer, Kuang, Rongze, Purakkattle, Biju, Ruiz, Manuel De, Stamford, Andrew, Ting, Pauline, Wu, Heping, Wang, Hongwu, Xiao, Dong, Yu, Tao, Zhang, Yonglian, Mullins, Deborra, Hodgson, Robert
Published in Bioorganic & medicinal chemistry letters (15.02.2016)

Get full text

Journal Article

혈장 칼리크레인 억제제

혈장 칼리크레인 억제제

by OGAWA ANTHONY KEN, ZHAO ZHIQIANG, BAO JIANMING, LANG SIMON B, JABRI SALMAN, TAOKA BRANDON M, HAYES DONNA A. A. W, SINZ CHRISTOPHER J, CHENG ALAN C, GAO YING DUO, KUANG RONGZE, SHEARN NANCE GALEN PAUL, HICKS JACQUELINE D, LOMBARDO MATTHEW J, TIAN MAOQUN, YANG SONG, WU ZHICAI
Year of Publication 21.02.2023

Get full text

Patent

치환된 아미노 트리아졸로피리미딘 및 아미노 트리아졸로피라진 아데노신 수용체 길항제, 제약 조성물 및 그의 용도

치환된 아미노 트리아졸로피리미딘 및 아미노 트리아졸로피라진 아데노신 수용체 길항제, 제약 조성물 및 그의 용도

by WANG HUIJUN, ALI AMJAD, DENG QIAOLIN, CUMMING JARED, KUANG RONGZE, DEMONG DUANE, RICO DUQUE JENNY LORENA, BRILL ZACHARY G, PLUMMER CHRISTOPHER W, ZHANG YONGLIAN, GRAHAM THOMAS H, LIM YEON HEE, ZHAO KAKE
Year of Publication 28.07.2021

Get full text

Patent

1
2
3
4
5
6
7
8
9
10
11
Next
[16]