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Published in Bioorganic & medicinal chemistry letters (01.04.2012)
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SAR studies of pyridazinone derivatives as novel glucan synthase inhibitors
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Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
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The synthesis and structure–activity relationship of pyridazinones as glucan synthase inhibitors
Ting, Pauline C., Kuang, Rongze, Wu, Heping, Aslanian, Robert G., Cao, Jianhua, Kim, David W., Lee, Joe F., Schwerdt, John, Zhou, Gang, Wainhaus, Samuel, Black, Todd A., Cacciapuoti, Anthony, McNicholas, Paul M., Xu, Yiming, Walker, Scott S.
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
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Lead optimization of a sulfonylurea-based piperazine pyridazinone series of glucan synthase inhibitors
Zych, Andrew J., Lam, Sang Q., Jenkins, David M., Herr, R. Jason, Ting, Pauline C., Lee, Joe F., Kuang, Rongze, Wu, Heping, Kim, David W., Aslanian, Robert G., Wainhaus, Samuel, Black, Todd A., Cacciapuoti, Anthony, McNicholas, Paul M., Xu, Yiming, Walker, Scott S.
Published in Bioorganic & medicinal chemistry letters (15.07.2012)
Published in Bioorganic & medicinal chemistry letters (15.07.2012)
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The optimization of pyridazinone series of glucan synthase inhibitors
Kuang, Rongze, Wu, Heping, Ting, Pauline C., Aslanian, Robert G., Cao, Jianhua, Kim, David W., Lee, Joe F., Schwerdt, John, Zhou, Gang, Jason Herr, R., Zych, Andrew J., Yang, Jinhai, Lam, Sang Q., Jenkins, David M., Sakwa, Samuel A., Wainhaus, Samuel, Black, Todd A., Cacciapuoti, Anthony, McNicholas, Paul M., Xu, Yiming, Walker, Scott S.
Published in Bioorganic & medicinal chemistry letters (15.08.2012)
Published in Bioorganic & medicinal chemistry letters (15.08.2012)
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Effects of structure on inhibitory activity in a series of mechanism-based inhibitors of human neutrophil elastase
Dou, Dengfeng, He, Guijia, Kuang, Rongze, Fu, Qingfong, Venkataraman, Radhika, Groutas, William C.
Published in Bioorganic & medicinal chemistry (15.09.2010)
Published in Bioorganic & medicinal chemistry (15.09.2010)
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Structure-Based Design of a General Class of Mechanism-Based Inhibitors of the Serine Proteinases Employing a Novel Amino Acid-Derived Heterocyclic Scaffold
Groutas, William C, Kuang, Rongze, Venkataraman, Radhika, Epp, Jeffrey B, Ruan, Sumei, Prakash, Om
Published in Biochemistry (Easton) (22.04.1997)
Published in Biochemistry (Easton) (22.04.1997)
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Utilization of the 1,2,5-thiadiazolidin-3-one 1,1 dioxide scaffold in the design of potent inhibitors of serine proteases: SAR studies using carboxylates
RONGZE KUANG, EPP, J. B, SUMEI RUAN, CHONG, L. S, VENKATARAMAN, R, JUAN TU, SHU HE, TRUONG, T. M, GROUTAS, W. C
Published in Bioorganic & medicinal chemistry (01.05.2000)
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Inhibition of Escherichia coli by dimethyl fumarate
Wang, Hai-Hong, Sun, Da-Wen, Kuang, Rongze
Published in International journal of food microbiology (11.04.2001)
Published in International journal of food microbiology (11.04.2001)
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Use of the 1,2,5-thiadiazolidin-3-one 1,1 dioxide and isothiazolidin-3-one 1,1 dioxide scaffolds in the design of potent inhibitors of serine proteinases
Kuang, Rongze, Venkataraman, Radhika, Ruan, Sumei, Groutas, William C.
Published in Bioorganic & medicinal chemistry letters (03.03.1998)
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Substituted 3-oxo-1,2,5-Thiadiazolidine 1,1-Dioxides: A New Class of Potential Mechanism-Based Inhibitors of Human Leukocyte Elastase and Cathepsin G
Groutas, W.C., Kuang, R.Z., Venkataraman, R.
Published in Biochemical and biophysical research communications (14.01.1994)
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Discovery of aminoquinazoline derivatives as human A(2A) adenosine receptor antagonists
Zhou, Gang, Aslanian, Robert, Gallo, Gioconda, Khan, Tanweer, Kuang, Rongze, Purakkattle, Biju, De Ruiz, Manuel, Stamford, Andrew, Ting, Pauline, Wu, Heping, Wang, Hongwu, Xiao, Dong, Yu, Tao, Zhang, Yonglian, Mullins, Deborra, Hodgson, Robert
Published in Bioorganic & medicinal chemistry letters (15.02.2016)
Published in Bioorganic & medicinal chemistry letters (15.02.2016)
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Published in Bioorganic & medicinal chemistry letters (15.02.2016)
Published in Bioorganic & medicinal chemistry letters (15.02.2016)
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Year of Publication 20.03.2023
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Zhou, Gang, Aslanian, Robert, Gallo, Gioconda, Khan, Tanweer, Kuang, Rongze, Purakkattle, Biju, Ruiz, Manuel De, Stamford, Andrew, Ting, Pauline, Wu, Heping, Wang, Hongwu, Xiao, Dong, Yu, Tao, Zhang, Yonglian, Mullins, Deborra, Hodgson, Robert
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Year of Publication 28.07.2021
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