First Scale-Up to Production Scale of a Ring Closing Metathesis Reaction Forming a 15-Membered Macrocycle as a Precursor of an Active Pharmaceutical Ingredient
Nicola, Thomas, Brenner, Michael, Donsbach, Kai, Kreye, Paul
Published in Organic process research & development (01.07.2005)
Published in Organic process research & development (01.07.2005)
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Efficient Large-Scale Synthesis of BILN 2061, a Potent HCV Protease Inhibitor, by a Convergent Approach Based on Ring-Closing Metathesis
Yee, Nathan K, Farina, Vittorio, Houpis, Ioannis N, Haddad, Nizar, Frutos, Rogelio P, Gallou, Fabrice, Wang, Xiao-jun, Wei, Xudong, Simpson, Robert D, Feng, Xuwu, Fuchs, Victor, Xu, Yibo, Tan, Jonathan, Zhang, Li, Xu, Jinghua, Smith-Keenan, Lana L, Vitous, Jana, Ridges, Michael D, Spinelli, Earl M, Johnson, Michael, Donsbach, Kai, Nicola, Thomas, Brenner, Michael, Winter, Eric, Kreye, Paul, Samstag, Wendelin
Published in Journal of organic chemistry (15.09.2006)
Published in Journal of organic chemistry (15.09.2006)
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Synthesis and biological evaluation of leucine enkephalin turn mimetics
Blomberg, D, Kreye, P, Fowler, C, Brickmann, K, Kihlberg, J
Published in Organic & biomolecular chemistry (07.02.2006)
Published in Organic & biomolecular chemistry (07.02.2006)
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Synthesis and Conformational Studies of a β-Turn Mimetic Incorporated in Leu-enkephalin
Blomberg, David, Hedenström, Mattias, Kreye, Paul, Sethson, Ingmar, Brickmann, Kay, Kihlberg, Jan
Published in Journal of organic chemistry (14.05.2004)
Published in Journal of organic chemistry (14.05.2004)
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Stereoselective Synthesis of Steroids and Related Compounds. Part 7. 3-Substituted and 2,3-Disubstituted Cyclopentanones via an Asymmetric Tandem 1,4-Addition/Dieckmann Cyclization
Groth, Ulrich, Halfbrodt, Wolfgang, Kalogerakis, Aris, Koehler, Thomas, Kreye, Paul
Published in ChemInform (15.06.2004)
Published in ChemInform (15.06.2004)
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