Rapid Synthesis of Highly Substituted 1,6-Naphthyridines Via Heteroaryl Ditriflates
Shimkin, Kirk W., Compton, Jordan S., Diccianni, Justin B., Waldo, Jesse P., Jones, William M., Krawczuk, Paul J., Rosano, Robert J.
Published in Journal of organic chemistry (02.08.2024)
Published in Journal of organic chemistry (02.08.2024)
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Structural Basis of Small-Molecule Aggregate Induced Inhibition of a Protein–Protein Interaction
Blevitt, Jonathan M, Hack, Michael D, Herman, Krystal L, Jackson, Paul F, Krawczuk, Paul J, Lebsack, Alec D, Liu, Annie X, Mirzadegan, Taraneh, Nelen, Marina I, Patrick, Aaron N, Steinbacher, Stefan, Milla, Marcos E, Lumb, Kevin J
Published in Journal of medicinal chemistry (27.04.2017)
Published in Journal of medicinal chemistry (27.04.2017)
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Discovery of a Gut-Restricted JAK Inhibitor for the Treatment of Inflammatory Bowel Disease
Leonard, Kristi A, Madge, Lisa A, Krawczuk, Paul J, Wang, Aihua, Kreutter, Kevin D, Bacani, Genesis M, Chai, Wenying, Smith, Russell C, Tichenor, Mark S, Harris, Michael C, Malaviya, Ravi, Seierstad, Mark, Johnson, Marguerite E, Venable, Jennifer D, Kim, Suzie, Hirst, Gavin C, Mathur, Ashok S, Rao, Tadimeti S, Edwards, James P, Rizzolio, Michele C, Koudriakova, Tatiana
Published in Journal of medicinal chemistry (26.03.2020)
Published in Journal of medicinal chemistry (26.03.2020)
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Energy and Electron Transfer in Polyacetylene-Linked Zinc-Porphyrin-[60]Fullerene Molecular Wires
Vail, Sean A., Krawczuk, Paul J., Guldi, Dirk M., Palkar, Amit, Echegoyen, Luis, Tomé, Joao P. C., Fazio, Michael A., Schuster, David I.
Published in Chemistry : a European journal (20.05.2005)
Published in Chemistry : a European journal (20.05.2005)
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Identification of Two Non-Peptidergic Small Molecule Inhibitors of CBX2 Binding to K27 Trimethylated Oligonucleosomes
Lercher, Lukas, Simon, Nina, Bergmann, Andreas, Tauchert, Marcel, Bochmann, David, Bashir, Tarig, Neuefeind, Torsten, Riley, Daniel, Danna, Ben, Krawczuk, Paul, Pande, Vineet, Patrick, Aaron, Steele, Ruth, Wang, Weixue, Rupnow, Brent, Tummino, Peter, Sharma, Sujata, Finley, Michael
Published in SLAS discovery (01.07.2022)
Published in SLAS discovery (01.07.2022)
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Polypharmacology of Small-Molecule Modulators of the 5-Lipoxygenase Activating Protein (FLAP) Observed via a High-throughput Lipidomics Platform
Song, Jiao, Liu, Xuejun, Zhu, Jian, Tootoonchi, Mandana, Keith, John M, Meduna, Steven P, Dvorak, Curt A, Eccles, Wendy, Krawczuk, Paul J, Blevitt, Jonathan M, Wu, Jiejun, Rao, Navin L, Lebsack, Alec D, Milla, Marcos E
Published in Journal of biomolecular screening (01.02.2016)
Published in Journal of biomolecular screening (01.02.2016)
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Journal Article
NF-kB 유도 키나아제의 소분자 억제제
KREUTTER KEVIN D, CHAI WENYING, LEBSACK ALEC D, PIPPEL DANIEL J, HERRMANN AARON T, ROVIRA ALEXANDER R, HACK MICHAEL D, BARBAY J. KENT, ECCLES WENDY, JONES WILLIAM M, KRAWCZUK PAUL J, WOLIN RONALD L
Year of Publication 08.03.2022
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Year of Publication 08.03.2022
Patent
JAK 패밀리의 키나제의 억제제로서의 이미다조피롤로피리딘
LEONARD KRISTI, KREUTTER KEVIN D, CHAI WENYING, SEIERSTAD MARK, BACANI GENESIS M, KOUDRIAKOVA TATIANA, TICHENOR MARK S, VENABLE JENNIFER D, RIZZOLIO MICHELE C, SMITH RUSSEL C, KRAWCZUK PAUL J, WANG AIHUA
Year of Publication 07.08.2019
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Year of Publication 07.08.2019
Patent
FLAP MODULATORS
KEITH JOHN M, HACK MICHAEL D, JONES WILLIAM M, ECCLES WENDY, MCCLURE KELLY J, ROSEN MARK D, HAWRYLUK NATALIE A, LEBSACK ALEC D, MANI NEELAKANDHA S, KRAWCZUK PAUL, FITZGERALD ANNE E, LIU JING, MEDUNA STEVEN P
Year of Publication 12.01.2016
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Year of Publication 12.01.2016
Patent
SMALL MOLECULAR INHIBITORS OF NF-kB INDUCING KINASE
Jones, William M, Krawczuk, Paul J, Eccles, Wendy, Hack, Michael D, Lebsack, Alec D, Pippel, Daniel J, Rovira, Alexander R, Wolin, Ronald L
Year of Publication 20.06.2024
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Year of Publication 20.06.2024
Patent