Search Results - "KRAUSE, James E." :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Characterization of N-(Adamantan-1-ylmethyl)-5-[(3R-aminopyrrolidin-1-yl)methyl]-2-chloro-benzamide, a P2X7 Antagonist in Animal Models of Pain and Inflammation

Characterization of N-(Adamantan-1-ylmethyl)-5-[(3R-aminopyrrolidin-1-yl)methyl]-2-chloro-benzamide, a P2X7 Antagonist in Animal Models of Pain and Inflammation

by Broom, Daniel C, Matson, David J, Bradshaw, Elizabeth, Buck, Marianne E, Meade, Robin, Coombs, Susan, Matchett, Michele, Ford, Kristen K, Yu, Weifeng, Yuan, Jun, Sun, Synthia H, Ochoa, Ricardo, Krause, James E, Wustrow, David J, Cortright, Daniel N
Published in The Journal of pharmacology and experimental therapeutics (01.12.2008)

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Discovery of N-(1-Ethylpropyl)-[3-methoxy-5-(2-methoxy-4-trifluoromethoxyphenyl)-6-methyl-pyrazin-2-yl]amine 59 (NGD 98−2): An Orally Active Corticotropin Releasing Factor-1 (CRF-1) Receptor Antagonist

Discovery of N-(1-Ethylpropyl)-[3-methoxy-5-(2-methoxy-4-trifluoromethoxyphenyl)-6-methyl-pyrazin-2-yl]amine 59 (NGD 98−2): An Orally Active Corticotropin Releasing Factor-1 (CRF-1) Receptor Antagonist

by Hodgetts, Kevin J, Ge, Ping, Yoon, Taeyoung, Lombaert, Stéphane De, Brodbeck, Robbin, Gulianello, Michael, Kieltyka, Andrzej, Horvath, Raymond F, Kehne, John H, Krause, James E, Maynard, George D, Hoffman, Diane, Lee, Younglim, Fung, Laurence, Doller, Dario
Published in Journal of medicinal chemistry (23.06.2011)

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Identification and Characterization of NDT 9513727 [N,N-bis(1,3-Benzodioxol-5-ylmethyl)-1-butyl-2,4-diphenyl-1H-imidazole-5-methanamine], a Novel, Orally Bioavailable C5a Receptor Inverse Agonist

Identification and Characterization of NDT 9513727 [N,N-bis(1,3-Benzodioxol-5-ylmethyl)-1-butyl-2,4-diphenyl-1H-imidazole-5-methanamine], a Novel, Orally Bioavailable C5a Receptor Inverse Agonist

by Brodbeck, Robbin M, Cortright, Daniel N, Kieltyka, Andrzej P, Yu, Jianying, Baltazar, Carolyn O, Buck, Marianne E, Meade, Robin, Maynard, George D, Thurkauf, Andrew, Chien, Du-Shieng, Hutchison, Alan J, Krause, James E
Published in The Journal of pharmacology and experimental therapeutics (01.12.2008)

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The design, synthesis and structure–activity relationships of 1-aryl-4-aminoalkylisoquinolines: A novel series of CRF-1 receptor antagonists

The design, synthesis and structure–activity relationships of 1-aryl-4-aminoalkylisoquinolines: A novel series of CRF-1 receptor antagonists

by Yoon, Taeyoung, De Lombaert, Stéphane, Brodbeck, Robbin, Gulianello, Michael, Chandrasekhar, Jayaraman, Horvath, Raymond F., Ge, Ping, Kershaw, Mark T., Krause, James E., Kehne, John, Hoffman, Diane, Doller, Darío, Hodgetts, Kevin J.
Published in Bioorganic & medicinal chemistry (01.02.2008)

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Leukocyte Effects of C5a-Receptor Blockade During Simulated Extracorporeal Circulation

Leukocyte Effects of C5a-Receptor Blockade During Simulated Extracorporeal Circulation

by Rinder, Christine S., MD, Smith, Michael J., PhD, Rinder, Henry M., MD, Cortright, Daniel N., PhD, Brodbeck, Robbin M., PhD, Krause, James E., PhD, Smith, Brian R., MD
Published in The Annals of thoracic surgery (2007)

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TRP channels and pain

TRP channels and pain

by Cortright, Daniel N., Krause, James E., Broom, Daniel C.
Published in Biochimica et biophysica acta (01.08.2007)

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Molecular Characterization of the Gerbil C5a Receptor and Identification of a Transmembrane Domain V Amino Acid That Is Crucial for Small Molecule Antagonist Interaction

Molecular Characterization of the Gerbil C5a Receptor and Identification of a Transmembrane Domain V Amino Acid That Is Crucial for Small Molecule Antagonist Interaction

by Waters, Stephen M., Brodbeck, Robbin M., Steflik, Jeremy, Yu, Jianying, Baltazar, Carolyn, Peck, Amy E., Severance, Daniel, Zhang, Lu Yan, Currie, Kevin, Chenard, Bertrand L., Hutchison, Alan J., Maynard, George, Krause, James E.
Published in The Journal of biological chemistry (09.12.2005)

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Molecular Characterization of a Functional cDNA Encoding the Rat Substance P Receptor

Molecular Characterization of a Functional cDNA Encoding the Rat Substance P Receptor

by Hershey, Andrew D., Krause, James E.
Published in Science (American Association for the Advancement of Science) (23.02.1990)

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Distribution of mRNA for vanilloid receptor subtype 1 (VR1), and VR1-like immunoreactivity, in the central nervous system of the rat and human

Distribution of mRNA for vanilloid receptor subtype 1 (VR1), and VR1-like immunoreactivity, in the central nervous system of the rat and human

by Mezey, Éva, Tóth, Zsuzsanna E., Cortright, Daniel N., Arzubi, Michelle K., Krause, James E., Elde, Robert, Guo, Athena, Blumberg, Peter M., Szallasi, Arpad
Published in Proceedings of the National Academy of Sciences - PNAS (28.03.2000)

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C5L2, a Nonsignaling C5A Binding Protein

C5L2, a Nonsignaling C5A Binding Protein

by Okinaga, Shoji, Slattery, Dubhfeasa, Humbles, Alison, Zsengeller, Zsusanna, Morteau, Olivier, Kinrade, Michele Bennett, Brodbeck, Robbin M, Krause, James E, Choe, Hye-Ryun, Gerard, Norma P, Gerard, Craig
Published in Biochemistry (Easton) (12.08.2003)

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Distribution of mRNA for Vanilloid Receptor Subtype 1 (VR1), and VR1-Like Immunoreactivity, in the Central Nervous System of the Rat and Human

Distribution of mRNA for Vanilloid Receptor Subtype 1 (VR1), and VR1-Like Immunoreactivity, in the Central Nervous System of the Rat and Human

by Mezey, Eva, Toth, Zsuzsanna E., Cortright, Daniel N., Arzubi, Michelle K., Krause, James E., Elde, Robert, Guo, Athena, Blumberg, Peter M., Szallasi, Arpad
Published in Proceedings of the National Academy of Sciences - PNAS (28.03.2000)

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Photoaffinity Labeling of Mutant Neurokinin-1 Receptors Reveals Additional Structural Features of the Substance P/NK-1 Receptor Complex

Photoaffinity Labeling of Mutant Neurokinin-1 Receptors Reveals Additional Structural Features of the Substance P/NK-1 Receptor Complex

by Macdonald, Douglas, Mierke, Dale F, Li, Hanzhong, Pellegrini, Maria, Sachais, Bruce, Krause, James E, Leeman, Susan E, Boyd, Norman D
Published in Biochemistry (Easton) (27.02.2001)

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C5a, But Not C3a, Increases VEGF Secretion in ARPE-19 Human Retinal Pigment Epithelial Cells

C5a, But Not C3a, Increases VEGF Secretion in ARPE-19 Human Retinal Pigment Epithelial Cells

by Cortright, Daniel N., Meade, Robin, Waters, Stephen M., Chenard, Bertrand L., Krause, James E.
Published in Current eye research (2009)

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Arginine-Vasopressin Neurons in the Rat Hypothalamus Produce Neurokinin B and Co-express the Tachykinin NK-3 Receptor and Angiotensin II Type 1 Receptor

Arginine-Vasopressin Neurons in the Rat Hypothalamus Produce Neurokinin B and Co-express the Tachykinin NK-3 Receptor and Angiotensin II Type 1 Receptor

by HATAE, Takashi, KAWANO, Hitoshi, KARPITSKIY, Vladimir, KRAUSE, James E., MASUKO, Sadahiko
Published in Archives of Histology and Cytology (01.01.2001)

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Discovery of Novel 6,6-Heterocycles as Transient Receptor Potential Vanilloid (TRPV1) Antagonists

Discovery of Novel 6,6-Heterocycles as Transient Receptor Potential Vanilloid (TRPV1) Antagonists

by Blum, Charles A, Caldwell, Timothy, Zheng, Xiaozhang, Bakthavatchalam, Rajagopal, Capitosti, Scott, Brielmann, Harry, De Lombaert, Stéphane, Kershaw, Mark T, Matson, David, Krause, James E, Cortright, Daniel, Crandall, Marci, Martin, William J, Murphy, Beth Ann, Boyce, Susan, Jones, A. Brian, Mason, Glenn, Rycroft, Wayne, Perrett, Helen, Conley, Rachael, Burnaby-Davies, Nicola, Chenard, Bertrand L, Hodgetts, Kevin J
Published in Journal of medicinal chemistry (22.04.2010)

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Opportunities and Challenges in the Discovery of New Central Nervous System Drugs

Opportunities and Challenges in the Discovery of New Central Nervous System Drugs

by Krause, James E., Chenard, Bertrand L.
Published in Annals of the New York Academy of Sciences (01.11.2008)

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Pyrido[2,3-b]pyrazines, discovery of TRPV1 antagonists with reduced potential for the formation of reactive metabolites

Pyrido[2,3-b]pyrazines, discovery of TRPV1 antagonists with reduced potential for the formation of reactive metabolites

by Hodgetts, Kevin J., Blum, Charles A., Caldwell, Timothy, Bakthavatchalam, Rajagopal, Zheng, Xiaozhang, Capitosti, Scott, Krause, James E., Cortright, Daniel, Crandall, Marci, Murphy, Beth Ann, Boyce, Susan, Brian Jones, A., Chenard, Bertrand L.
Published in Bioorganic & medicinal chemistry letters (01.08.2010)

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Aminoquinazolines as TRPV1 antagonists: Modulation of drug-like properties through the exploration of 2-position substitution

Aminoquinazolines as TRPV1 antagonists: Modulation of drug-like properties through the exploration of 2-position substitution

by Blum, Charles A., Zheng, Xiaozhang, Brielmann, Harry, Hodgetts, Kevin J., Bakthavatchalam, Rajagopal, Chandrasekhar, Jayaraman, Krause, James E., Cortright, Daniel, Matson, David, Crandall, Marci, Ngo, Chu K., Fung, Lawrence, Day, Marta, Kershaw, Mark, De Lombaert, Stéphane, Chenard, Bertrand L.
Published in Bioorganic & medicinal chemistry (15.08.2008)

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Hunting for ion channel modulators with herpes simplex virus

Hunting for ion channel modulators with herpes simplex virus

by Cortright, Daniel N, Buck, Marianne E, Krause, James E
Published in Nature methods (01.09.2007)

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Substance P and its receptor neurokinin 1 expression in asthmatic airways

Substance P and its receptor neurokinin 1 expression in asthmatic airways

by Chu, Hong Wei, Kraft, Monica, Krause, James E., Rex, Michael D., Martin, Richard J.
Published in Journal of allergy and clinical immunology (01.10.2000)

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