Combining BH3-mimetics to target both BCL-2 and MCL1 has potent activity in pre-clinical models of acute myeloid leukemia
Moujalled, Donia M, Pomilio, Giovanna, Ghiurau, Corina, Ivey, Adam, Salmon, Jessica, Rijal, Sewa, Macraild, Sarah, Zhang, Lan, Teh, Tse-Chieh, Tiong, Ing-Soo, Lan, Ping, Chanrion, Maia, Claperon, Audrey, Rocchetti, Francesca, Zichi, Adrien, Kraus-Berthier, Laurence, Wang, Youzhen, Halilovic, Ensar, Morris, Erick, Colland, Frédéric, Segal, David, Huang, David, Roberts, Andrew W, Maragno, Ana Leticia, Lessene, Guillaume, Geneste, Olivier, Wei, Andrew H
Published in Leukemia (01.04.2019)
Published in Leukemia (01.04.2019)
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Preclinical evaluation of the simultaneous inhibition of MCL-1 and BCL-2 with the combination of S63845 and venetoclax in multiple myeloma
Algarín, Esperanza M, Díaz-Tejedor, Andrea, Mogollón, Pedro, Hernández-García, Susana, Corchete, Luis A, San-Segundo, Laura, Martín-Sánchez, Montserrat, González-Méndez, Lorena, Schoumacher, Marie, Banquet, Sebastien, Kraus-Berthier, Laurence, Kloos, Ioana, Derreal, Alix, Halilovic, Ensar, Maacke, Heiko, Gutiérrez, Norma C, Mateos, María-Victoria, Paíno, Teresa, Garayoa, Mercedes, Ocio, Enrique M
Published in Haematologica (Roma) (01.03.2020)
Published in Haematologica (Roma) (01.03.2020)
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Treatment of nasopharyngeal carcinoma cells with the histone-deacetylase inhibitor abexinostat: cooperative effects with cis-platin and radiotherapy on patient-derived xenografts
Gressette, Mélanie, Vérillaud, Benjamin, Jimenez-Pailhès, Anne-Sophie, Lelièvre, Hélène, Lo, Kwok-Wai, Ferrand, François-Régis, Gattolliat, Charles-Henry, Jacquet-Bescond, Anne, Kraus-Berthier, Laurence, Depil, Stéphane, Busson, Pierre
Published in PloS one (11.03.2014)
Published in PloS one (11.03.2014)
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Synthesis and Cytotoxic and Antitumor Activity of 1,2-Dihydroxy-1,2-dihydrobenzo[b]acronycine Diacid Hemiesters and Carbamates
Mai, Huong Doan Thi, Gaslonde, Thomas, Michel, Sylvie, Koch, Michel, Tillequin, François, Pfeiffer, Bruno, Renard, Pierre, Kraus-Berthier, Laurence, Léonce, Stéphane, Pierré, Alain
Published in Chemical & pharmaceutical bulletin (01.03.2004)
Published in Chemical & pharmaceutical bulletin (01.03.2004)
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Targeting Bcl-2/Bcl-XL induces antitumor activity in uveal melanoma patient-derived xenografts
Némati, Fariba, de Montrion, Catherine, Lang, Guillaume, Kraus-Berthier, Laurence, Carita, Guillaume, Sastre-Garau, Xavier, Berniard, Aurélie, Vallerand, David, Geneste, Olivier, de Plater, Ludmilla, Pierré, Alain, Lockhart, Brian, Desjardins, Laurence, Piperno-Neumann, Sophie, Depil, Stéphane, Decaudin, Didier
Published in PloS one (2014)
Published in PloS one (2014)
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Novel Stable Camptothecin Derivatives Replacing the E-Ring Lactone by a Ketone Function Are Potent Inhibitors of Topoisomerase I and Promising Antitumor Drugs
Lansiaux, Amélie, Léonce, Stéphane, Kraus-Berthier, Laurence, Bal-Mahieu, Christine, Mazinghien, Romain, Didier, Sébastien, David-Cordonnier, Marie-Hélène, Hautefaye, Patrick, Lavielle, Gilbert, Bailly, Christian, Hickman, John A, Pierré, Alain
Published in Molecular pharmacology (01.08.2007)
Published in Molecular pharmacology (01.08.2007)
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Influence of the Stereoisomeric Position of the Reactive Acetate Groups of the Benzo[b]Acronycine derivative S23906-1 on Its DNA Alkylation, Helix-Opening, Cytotoxic, and Antitumor Activities
Sabine Depauw, Thomas Gaslonde, Stéphane Léonce, Laurence Kraus-Berthier, William Laine, Gaëlle Lenglet, Angèle Chiaroni, Bruno Pfeiffer, Christian Bailly, Sylvie Michel, François Tillequin, Alain PierrÃ, Marie-Hélène David-Cordonnier
Published in Molecular pharmacology (01.12.2009)
Published in Molecular pharmacology (01.12.2009)
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Synthesis and Biological Study of a New Series of 4‘-Demethylepipodophyllotoxin Derivatives
Duca, Maria, Guianvarc'h, Dominique, Meresse, Philippe, Bertounesque, Emmanuel, Dauzonne, Daniel, Kraus-Berthier, Laurence, Thirot, Sylvie, Léonce, Stéphane, Pierré, Alain, Pfeiffer, Bruno, Renard, Pierre, Arimondo, Paola B, Monneret, Claude
Published in Journal of medicinal chemistry (27.01.2005)
Published in Journal of medicinal chemistry (27.01.2005)
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Synthesis and Biological Activity of Sulfonamide Derivatives of Epipodophyllotoxin
Guianvarc'h, Dominique, Duca, Maria, Boukarim, Chawki, Kraus-Berthier, Laurence, Léonce, Stéphane, Pierré, Alain, Pfeiffer, Bruno, Renard, Pierre, Arimondo, Paola B, Monneret, Claude, Dauzonne, Daniel
Published in Journal of medicinal chemistry (22.04.2004)
Published in Journal of medicinal chemistry (22.04.2004)
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Marked Antitumor Activity of a New Potent Acronycine Derivative in Orthotopic Models of Human Solid Tumors
GUILBAUD, Nicolas, KRAUS-BERTHIER, Laurence, ATASSI, Ghanem, HICKMAN, John, PIERRE, Alain, MEYER-LOSIC, Florence, MALIVET, Virginie, CHACUN, Christine, JAN, Michel, TILLEQUIN, Francois, MICHEL, Sylvie, KOCH, Michel, PFEIFFER, Bruno
Published in Clinical cancer research (01.08.2001)
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Published in Clinical cancer research (01.08.2001)
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Synthesis and Cytotoxic and Antitumor Activity of Esters in the 1,2-Dihydroxy-1,2-dihydroacronycine Series
Elomri, Abdelhakim, Mitaku, Sofia, Michel, Sylvie, Skaltsounis, Alexios-Léandros, Tillequin, François, Koch, Michel, Pierré, Alain, Guilbaud, Nicolas, Léonce, Stéphane, Kraus-Berthier, Laurence, Rolland, Yves, Atassi, Ghanem
Published in Journal of medicinal chemistry (22.11.1996)
Published in Journal of medicinal chemistry (22.11.1996)
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Up‐regulated expression of the β3 integrin and the 92‐kDa gelatinase in human HT‐144 melanoma cell tumors grown in nude mice
Gouon, Valérie, Tucker, Gordon C., Kraus‐Berthier, Laurence, Atassi, Ghanem, Kieffer, Nelly
Published in International journal of cancer (27.11.1996)
Published in International journal of cancer (27.11.1996)
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The Histone Deacetylase Inhibitor Abexinostat Induces Cancer Stem Cells Differentiation in Breast Cancer with Low Xist Expression
SALVADOR, Marion A, WICINSKI, Julien, COLLETTE, Yves, BIRNBAUM, Daniel, CHARAFE-JAUFFRET, Emmanuelle, GINESTIER, Christophe, CABAUD, Olivier, TOIRON, Yves, FINETTI, Pascal, JOSSELIN, Emmanuelle, LELIEVRE, Hélène, KRAUS-BERTHIER, Laurence, DEPIL, Stéphane, BERTUCCI, François
Published in Clinical cancer research (01.12.2013)
Published in Clinical cancer research (01.12.2013)
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S55746 is a novel orally active BCL-2 selective and potent inhibitor that impairs hematological tumor growth
Casara, Patrick, Davidson, James, Claperon, Audrey, Le Toumelin-Braizat, Gaëtane, Vogler, Meike, Bruno, Alain, Chanrion, Maïa, Lysiak-Auvity, Gaëlle, Le Diguarher, Thierry, Starck, Jérôme-Benoît, Chen, Ijen, Whitehead, Neil, Graham, Christopher, Matassova, Natalia, Dokurno, Pawel, Pedder, Christopher, Wang, Youzhen, Qiu, Shumei, Girard, Anne-Marie, Schneider, Emilie, Gravé, Fabienne, Studeny, Aurélie, Guasconi, Ghislaine, Rocchetti, Francesca, Maïga, Sophie, Henlin, Jean-Michel, Colland, Frédéric, Kraus-Berthier, Laurence, Le Gouill, Steven, Dyer, Martin J S, Hubbard, Roderick, Wood, Mike, Amiot, Martine, Cohen, Gerald M, Hickman, John A, Morris, Erick, Murray, James, Geneste, Olivier
Published in Oncotarget (13.04.2018)
Published in Oncotarget (13.04.2018)
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Prediction of Human Nonlinear Pharmacokinetics of a New Bcl-2 Inhibitor Using PBPK Modeling and Interspecies Extrapolation Strategy
Pierrillas, Philippe B, Henin, Emilie, Ball, Kathryn, Ogier, Julien, Amiel, Magali, Kraus-Berthier, Laurence, Chenel, Marylore, Bouzom, François, Tod, Michel
Published in Drug metabolism and disposition (01.06.2019)
Published in Drug metabolism and disposition (01.06.2019)
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Tumor Growth Inhibition modelling based on receptor occupancy and biomarker activity of a new Bcl-2 inhibitor in mice
Pierrillas, Philippe B, Henin, Emilie, Ogier, Julien, Kraus-Berthier, Laurence, Chenel, Marylore, Bouzom, Francois, Tod, Michel
Published in The Journal of pharmacology and experimental therapeutics (01.12.2018)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2018)
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Comparison of the pharmacological profile of an olivacine derivative and a potential prodrug
KRAUS-BERTHIER, Laurence, GUILBAUD, Nicolas, LEONCE, Stéphane, PARKER, Tracy, GENISSEL, Patrick, GUILLONNEAU, Claude, GOLDSTEIN, Solo, ATASSI, Ghanem, PIERRE, Alain
Published in Cancer chemotherapy and pharmacology (01.08.2002)
Published in Cancer chemotherapy and pharmacology (01.08.2002)
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Cytokine-like protein 1–induced survival of monocytes suggests a combined strategy targeting MCL1 and MAPK in CMML
Sevin, Margaux, Debeurme, Franck, Laplane, Lucie, Badel, Séverine, Morabito, Margot, Newman, Hanna L., Torres-Martin, Miguel, Yang, Qin, Badaoui, Bouchra, Wagner-Ballon, Orianne, Saada, Véronique, Sélimoglu-Buet, Dorothée, Kraus-Berthier, Laurence, Banquet, Sébastien, Derreal, Alix, Fenaux, Pierre, Itzykson, Raphael, Braun, Thorsten, Etienne, Gabriel, Berthon, Celine, Thépot, Sylvain, Kepp, Oliver, Kroemer, Guido, Padron, Eric, Figueroa, Maria E., Droin, Nathalie, Solary, Eric
Published in Blood (17.06.2021)
Published in Blood (17.06.2021)
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Synthesis, Antitumor Activity, and Mechanism of Action of Benzo[b]chromeno[6,5-g][1,81naphthyridin-7-one Analogs of Acronycine
Tian, Wen, Yougnia, Rodrigue, Depauw, Sabine, Lansiaux, Amelie, David-Cordonnier, Marie-Helene, Pfeiffer, Bruno, Kraus-Berthier, Laurence, Leonce, Stephane, Pierre, Alain, Dufat, Hanh, Michel, Sylvie
Published in Journal of medicinal chemistry (25.12.2014)
Published in Journal of medicinal chemistry (25.12.2014)
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