Search Results - "KRASAVIN MIKHAIL" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Pyridazinone-substituted benzenesulfonamides display potent inhibition of membrane-bound human carbonic anhydrase IX and promising antiproliferative activity against cancer cell lines

Pyridazinone-substituted benzenesulfonamides display potent inhibition of membrane-bound human carbonic anhydrase IX and promising antiproliferative activity against cancer cell lines

by Krasavin, Mikhail, Shetnev, Anton, Baykov, Sergey, Kalinin, Stanislav, Nocentini, Alessio, Sharoyko, Vladimir, Poli, Giulio, Tuccinardi, Tiziano, Korsakov, Mikhail, Tennikova, Tatiana B., Supuran, Claudiu T.
Published in European journal of medicinal chemistry (15.04.2019)

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From random to rational: A discovery approach to selective subnanomolar inhibitors of human carbonic anhydrase IV based on the Castagnoli-Cushman multicomponent reaction

From random to rational: A discovery approach to selective subnanomolar inhibitors of human carbonic anhydrase IV based on the Castagnoli-Cushman multicomponent reaction

by Kalinin, Stanislav, Nocentini, Alessio, Kovalenko, Alexander, Sharoyko, Vladimir, Bonardi, Alessandro, Angeli, Andrea, Gratteri, Paola, Tennikova, Tatiana B., Supuran, Claudiu T., Krasavin, Mikhail
Published in European journal of medicinal chemistry (15.11.2019)

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Rare cis-configured 2,4-disubstituted 1-alkylpiperidines: synthesized and tested against trace-amine-associated receptor 1 (TAAR1)

Rare cis-configured 2,4-disubstituted 1-alkylpiperidines: synthesized and tested against trace-amine-associated receptor 1 (TAAR1)

by Levashova, Ekaterina, Firsov, Andrey, Bakulina, Olga, Peshkov, Anatoly, Kanov, Evgeny, Gainetdinov, Raul R., Krasavin, Mikhail
Published in Mendeleev communications (01.07.2021)

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A novel, flexible strategy to construct privileged dibenzo[b,f][1,4,5]oxathiazepine 5,5-dioxides and their heterocyclic isosteres

A novel, flexible strategy to construct privileged dibenzo[b,f][1,4,5]oxathiazepine 5,5-dioxides and their heterocyclic isosteres

by Sapegin, Alexander, Panova, Valeria, Reutskaya, Elena, Smirnov, Alexey V., Krasavin, Mikhail
Published in Tetrahedron (24.11.2016)

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Corrigendum to “Investigation of 3-sulfamoyl coumarins against cancer-related IX and XII isoforms of human carbonic anhydrase as well as cancer cells leads to the discovery of 2-oxo-2H-benzo[h]chromene-3-sulfonamide – A new caspase-activating proapoptotic agent” [J. Med. Chem. 222 (2021) 113589]

Corrigendum to “Investigation of 3-sulfamoyl coumarins against cancer-related IX and XII isoforms of human carbonic anhydrase as well as cancer cells leads to the discovery of 2-oxo-2H-benzo[h]chromene-3-sulfonamide – A new caspase-activating proapoptotic agent” [J. Med. Chem. 222 (2021) 113589]

by Dar'in, Dmitry, Kantin, Grigory, Kalinin, Stanislav, Sharonova, Tatiana, Bunev, Alexander, Ostapenko, Gennady I., Nocentini, Alessio, Sharoyko, Vladimir, Supuran, Claudiu T., Krasavin, Mikhail
Published in European journal of medicinal chemistry (05.12.2021)

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Reaction of [alpha]-tetralone, 1H-tetrazol-5-amine, and aromatic aldehydes upon microwave irradiation - a convenient method for the synthesis of 5,6,7,12-tetrahydrobenzo[h]tetrazolo[5,1-b]quinazolines

Reaction of [alpha]-tetralone, 1H-tetrazol-5-amine, and aromatic aldehydes upon microwave irradiation - a convenient method for the synthesis of 5,6,7,12-tetrahydrobenzo[h]tetrazolo[5,1-b]quinazolines

by Kantin, Grigory P, Krasavin, Mikhail
Published in Chemistry of heterocyclic compounds (New York, N.Y. 1965) (01.11.2016)

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(E)-3-Arylidene-4-diazopyrrolidine-2,5-diones conveniently elaborated into cytotoxic compounds bearing primary sulfonamide and Michael acceptor moieties

(E)-3-Arylidene-4-diazopyrrolidine-2,5-diones conveniently elaborated into cytotoxic compounds bearing primary sulfonamide and Michael acceptor moieties

by Paramonova, Polina, Sharonova, Tatiana, Kalinin, Stanislav, Chupakhin, Evgeny, Bunev, Alexander, Krasavin, Mikhail
Published in Mendeleev communications (01.03.2022)

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Highly hydrophilic 1,3-oxazol-5-yl benzenesulfonamide inhibitors of carbonic anhydrase II for reduction of glaucoma-related intraocular pressure

Highly hydrophilic 1,3-oxazol-5-yl benzenesulfonamide inhibitors of carbonic anhydrase II for reduction of glaucoma-related intraocular pressure

by Kalinin, Stanislav, Valtari, Annika, Ruponen, Marika, Toropainen, Elisa, Kovalenko, Alexander, Nocentini, Alessio, Gureev, Maxim, Dar'in, Dmitry, Urtti, Arto, Supuran, Claudiu T., Krasavin, Mikhail
Published in Bioorganic & medicinal chemistry (01.11.2019)

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Imidazo[1,2-a]quinoxalines Accessed via Two Sequential Isocyanide-Based Multicomponent Reactions

Imidazo[1,2-a]quinoxalines Accessed via Two Sequential Isocyanide-Based Multicomponent Reactions

by Krasavin, Mikhail, Shkavrov, Sergey, Parchinsky, Vladislav, Bukhryakov, Konstantin
Published in Journal of organic chemistry (20.03.2009)

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Carnosine protects neurons against oxidative stress and modulates the time profile of MAPK cascade signaling

by Kulebyakin, Konstantin, Karpova, Larisa, Lakonsteva, Ekaterina, Krasavin, Mikhail, Boldyrev, Alexander
Published in Amino acids (01.07.2012)

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A new way of synthesizing heterocyclic primary sulfonamide probes for carbonic anhydrase

A new way of synthesizing heterocyclic primary sulfonamide probes for carbonic anhydrase

by Krivovicheva, Vasilisa, Bubyrev, Andrey, Kalinin, Stanislav, Dar'in, Dmitry, Gureev, Maxim, Vullo, Daniela, Krasavin, Mikhail, Korsakov, Mikhail, Supuran, Claudiu T.
Published in Mendeleev communications (01.05.2023)

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Castagnoli‐Cushman Reaction of 3‐Aryl Glutaric Acids: A Convenient, Diastereoselective Reaction for 6‐Oxo‐2,4‐diarylpiperidine‐3‐carboxylic Acid Scaffold

Castagnoli‐Cushman Reaction of 3‐Aryl Glutaric Acids: A Convenient, Diastereoselective Reaction for 6‐Oxo‐2,4‐diarylpiperidine‐3‐carboxylic Acid Scaffold

by Paramonova, Polina, Bakulina, Olga, Nabiyev, Alem, Dar'in, Dmitry, Krasavin, Mikhail
Published in ChemistrySelect (Weinheim) (21.01.2022)

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Three‐Component Castagnoli‐Cushman Reaction of 3‐Arylglutaconic Acid Anhydrides, Carbonyl Compounds, and Ammonium Acetate: a Quick and Flexible Way to Assemble Polysubstituted NH‐δ‐lactams

Three‐Component Castagnoli‐Cushman Reaction of 3‐Arylglutaconic Acid Anhydrides, Carbonyl Compounds, and Ammonium Acetate: a Quick and Flexible Way to Assemble Polysubstituted NH‐δ‐lactams

by Peshkov, Anatoly A., Bakulina, Olga, Dar'in, Dmitry, Kantin, Grigory, Bannykh, Anton, Peshkov, Vsevolod A., Krasavin, Mikhail
Published in European journal of organic chemistry (19.03.2021)

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Insertion of metal carbenes into the anilinic N–H bond of unprotected aminobenzenesulfonamides delivers low nanomolar inhibitors of human carbonic anhydrase IX and XII isoforms

Insertion of metal carbenes into the anilinic N–H bond of unprotected aminobenzenesulfonamides delivers low nanomolar inhibitors of human carbonic anhydrase IX and XII isoforms

by Sharonova, Tatiana, Paramonova, Polina, Kalinin, Stanislav, Bunev, Alexander, Gasanov, Rovshan Е., Nocentini, Alessio, Sharoyko, Vladimir, Tennikova, Tatiana B., Dar’in, Dmitry, Supuran, Claudiu T., Krasavin, Mikhail
Published in European journal of medicinal chemistry (05.06.2021)

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1,3-Oxazole-based selective picomolar inhibitors of cytosolic human carbonic anhydrase II alleviate ocular hypertension in rabbits: Potency is supported by X-ray crystallography of two leads

1,3-Oxazole-based selective picomolar inhibitors of cytosolic human carbonic anhydrase II alleviate ocular hypertension in rabbits: Potency is supported by X-ray crystallography of two leads

by Ferraroni, Marta, Lucarini, Laura, Masini, Emanuela, Korsakov, Mikhail, Scozzafava, Andrea, Supuran, Claudiu T., Krasavin, Mikhail
Published in Bioorganic & medicinal chemistry (01.09.2017)

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Dual PTP1B/TC-PTP Inhibitors: Biological Evaluation of 3--Ones

Dual PTP1B/TC-PTP Inhibitors: Biological Evaluation of 3--Ones

by Derkach, Kira V, Gureev, Maxim A, Babushkina, Anastasia A, Mikhaylov, Vladimir N, Zakharova, Irina O, Bakhtyukov, Andrey A, Sorokoumov, Viktor N, Novikov, Alexander S, Krasavin, Mikhail, Shpakov, Alexander O, Balova, Irina A
Published in International journal of molecular sciences (01.02.2023)

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Attachment of a 5-nitrofuroyl moiety to spirocyclic piperidines produces non-toxic nitrofurans that are efficacious in vitro against multidrug-resistant Mycobacterium tuberculosis

Attachment of a 5-nitrofuroyl moiety to spirocyclic piperidines produces non-toxic nitrofurans that are efficacious in vitro against multidrug-resistant Mycobacterium tuberculosis

by Krasavin, Mikhail, Lukin, Alexei, Vedekhina, Tatiana, Manicheva, Olga, Dogonadze, Marine, Vinogradova, Tatiana, Zabolotnykh, Natalia, Rogacheva, Elizaveta, Kraeva, Liudmila, Sharoyko, Vladimir, Tennikova, Tatiana B., Dar'in, Dmitry, Sokolovich, Evgeny
Published in European journal of medicinal chemistry (15.03.2019)

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Exploration of the nitrogen heterocyclic periphery around the core of the advanced FFA1 agonist fasiglifam (TAK‐875)

Exploration of the nitrogen heterocyclic periphery around the core of the advanced FFA1 agonist fasiglifam (TAK‐875)

by Lukin, Alexey, Bakholdina, Anna, Zhurilo, Nikolay, Onopchenko, Oleksandra, Zhuravel, Elena, Zozulya, Sergey, Gureev, Maxim, Safrygin, Alexander, Krasavin, Mikhail
Published in Archiv der Pharmazie (Weinheim) (01.04.2021)

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Novel electrophilic amides amenable by the Ugi reaction perturb thioredoxin system via thioredoxin reductase 1 (TrxR1) inhibition: Identification of DVD-445 as a new lead compound for anticancer therapy

Novel electrophilic amides amenable by the Ugi reaction perturb thioredoxin system via thioredoxin reductase 1 (TrxR1) inhibition: Identification of DVD-445 as a new lead compound for anticancer therapy

by Jovanović, Mirna, Zhukovsky, Daniil, Podolski-Renić, Ana, Domračeva, Ilona, Žalubovskis, Raivis, Senćanski, Milan, Glišić, Sanja, Sharoyko, Vladimir, Tennikova, Tatiana, Dar'in, Dmitry, Pešić, Milica, Krasavin, Mikhail
Published in European journal of medicinal chemistry (01.11.2019)

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Preparation and in situ use of unstable N -alkyl α-diazo-γ-butyrolactams in Rh II -catalyzed X-H insertion reactions

Preparation and in situ use of unstable N -alkyl α-diazo-γ-butyrolactams in Rh II -catalyzed X-H insertion reactions

by Eremeyeva, Maria, Zhukovsky, Daniil, Dar'in, Dmitry, Krasavin, Mikhail
Published in Beilstein journal of organic chemistry (02.04.2020)

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