Realizing the Trifunctional Potential of Alkyl 4-Chloro-2-diazo-3-oxobutanoates: Convenient Assembly of 6,7-Dihydro-4H-[1,2,3]triazolo[5,1-c][1,4]thiazine Core
Dar'in, Dmitrii, Khoroshilova, Olesya, Kantin, Grigory, Krasavin, Mikhail
Published in Synthesis (Stuttgart) (17.04.2020)
Published in Synthesis (Stuttgart) (17.04.2020)
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An Alternative Approach to the Hydrated Imidazoline Ring Expansion (HIRE) of Diarene‐Fused [1.4]Oxazepines
Grintsevich, Sergey, Sapegin, Alexander, Reutskaya, Elena, Peintner, Stefan, Erdélyi, Máté, Krasavin, Mikhail
Published in European journal of organic chemistry (22.09.2020)
Published in European journal of organic chemistry (22.09.2020)
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Further Insight into the Castagnoli–Cushman-type Synthesis of 1,4,6-Trisubstituted 1,6-Dihydropyridin-2-(3H)‑ones from 3‑Arylglutaconic Acid Anhydrides
Firsov, Andrei, Bakulina, Olga, Dar’in, Dmitry, Guranova, Natalia, Krasavin, Mikhail
Published in Journal of organic chemistry (15.05.2020)
Published in Journal of organic chemistry (15.05.2020)
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Synthesis of novel glutarimide ligands for the E3 ligase substrate receptor Cereblon (CRBN): Investigation of their binding mode and antiproliferative effects against myeloma cell lines
Krasavin, Mikhail, Adamchik, Maria, Bubyrev, Andrey, Heim, Christopher, Maiwald, Samuel, Zhukovsky, Daniil, Zhmurov, Petr, Bunev, Alexander, Hartmann, Marcus D.
Published in European journal of medicinal chemistry (15.01.2023)
Published in European journal of medicinal chemistry (15.01.2023)
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Three-Component Castagnoli–Cushman Reaction of 3‑Arylglutaconic Acids with Aromatic Aldehydes and Amines Delivers Rare 4,6-Diaryl-1,6-dihydropyridin-2(3H)‑ones
Firsov, Andrei, Chupakhin, Evgeny, Dar’in, Dmitry, Bakulina, Olga, Krasavin, Mikhail
Published in Organic letters (15.03.2019)
Published in Organic letters (15.03.2019)
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Mucoadhesive properties of nanogels based on stimuli-sensitive glycosaminoglycan-graft-pNIPAAm copolymers
Pilipenko, Iuliia, Korzhikov-Vlakh, Viktor, Valtari, Annika, Anufrikov, Yurii, Kalinin, Stanislav, Ruponen, Marika, Krasavin, Mikhail, Urtti, Arto, Tennikova, Tatiana
Published in International journal of biological macromolecules (01.09.2021)
Published in International journal of biological macromolecules (01.09.2021)
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Rethinking Hydrolytic Imidazoline Ring Expansion: A Common Approach to the Preparation of Medium-Sized Rings via Side-Chain Insertion into [1.4]Oxa- and [1.4]Thiazepinone Scaffolds
Reutskaya, Elena, Osipyan, Angelina, Sapegin, Alexander, Novikov, Alexander S, Krasavin, Mikhail
Published in Journal of organic chemistry (15.02.2019)
Published in Journal of organic chemistry (15.02.2019)
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Synthesis of 1-oxa-9-azaspiro[5.5]undecane-9-sulfonamides bearing a diverse molecular periphery and a rare zinc-binding group for carbonic anhydrase interrogation
Lukin, Alexey, Vinogradova, Lyubov, Komarova, Kristina, Kalinin, Stanislav, Krasavin, Mikhail
Published in Mendeleev communications (01.03.2023)
Published in Mendeleev communications (01.03.2023)
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Unexpected formal [4 + 2]-cycloaddition of chalcone imines and homophthalic anhydrides: preparation of dihydropyridin-2(1)-ones
Guranova, Natalia, Golubev, Pavel, Bakulina, Olga, Dar'in, Dmitry, Kantin, Grigory, Krasavin, Mikhail
Published in Organic & biomolecular chemistry (05.05.2021)
Published in Organic & biomolecular chemistry (05.05.2021)
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Non-chelating p-phenylidene-linked bis-imidazoline analogs of known influenza virus endonuclease inhibitors: Synthesis and anti-influenza activity
Dar'in, Dmitry, Zarubaev, Vladimir, Galochkina, Anastasia, Gureev, Maxim, Krasavin, Mikhail
Published in European journal of medicinal chemistry (01.01.2019)
Published in European journal of medicinal chemistry (01.01.2019)
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Diversity-oriented synthesis of N,N-dimethylamino-substituted azoles employing TBTU
Lukin, Alexey, Kalinchenkova, Natalya, Vedekhina, Tatiana, Zhurilo, Nikolay, Krasavin, Mikhail
Published in Tetrahedron letters (11.07.2018)
Published in Tetrahedron letters (11.07.2018)
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From Rare Reagents to Rare Products: Regiospecific Silver‐Catalyzed [3+2] Cycloaddition of Aryl‐, Alkyl‐ and Aminosulfonyl Diazomethanes with Arenediazonium Tosylates
Levashova, Ekaterina, Bakulina, Olga, Dar'in, Dmitry, Bubyrev, Andrey, Chuprun, Sergey, Krasavin, Mikhail
Published in European journal of organic chemistry (23.07.2020)
Published in European journal of organic chemistry (23.07.2020)
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Probing the ‘bipolar’ nature of the carbonic anhydrase active site: Aromatic sulfonamides containing 1,3-oxazol-5-yl moiety as picomolar inhibitors of cytosolic CA I and CA II isoforms
Krasavin, Mikhail, Korsakov, Mikhail, Dorogov, Mikhail, Tuccinardi, Tiziano, Dedeoglu, Nurcan, Supuran, Claudiu T.
Published in European journal of medicinal chemistry (28.08.2015)
Published in European journal of medicinal chemistry (28.08.2015)
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