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Published in Talanta (Oxford) (15.11.2005)
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Structure of HIV-1 reverse transcriptase in a complex with the non-nucleoside inhibitor α-APA R 95845 at 2.8 å resolution
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Published in Structure (London) (15.04.1995)
Published in Structure (London) (15.04.1995)
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Vinkers, H M, de Jonge, M R, Daeyaert, E D, Heeres, J, Koymans, L M H, van Lenthe, J H, Lewi, P J, Timmerman, H, Janssen, P A J
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Koymans, Luc M.H., Moereels, Henri, Bossche, Hugo Vanden
Published in Journal of steroid biochemistry and molecular biology (01.06.1995)
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Published in Protein science (01.10.1995)
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Lisitsa, A. V., Guseva, S. A., Karuzina, I. I., Archakov, A. I., Koymans, L.
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In Search of a Novel Anti-HIV Drug: Multidisciplinary Coordination in the Discovery of 4-[[4-[[4-[(1E)-2-Cyanoethenyl]-2,6-dimethylphenyl]amino]-2- pyrimidinyl]amino]benzonitrile (R278474, Rilpivirine)
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Published in Journal of medicinal chemistry (24.03.2005)
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Published in Antimicrobial Agents and Chemotherapy (01.02.1998)
Published in Antimicrobial Agents and Chemotherapy (01.02.1998)
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P450 superfamily: update on new sequences, gene mapping, accession numbers and nomenclature
Nelson, D R, Koymans, L, Kamataki, T, Stegeman, J J, Feyereisen, R, Waxman, D J, Waterman, M R, Gotoh, O, Coon, M J, Estabrook, R W, Gunsalus, I C, Nebert, D W
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Published in Pharmacogenetics (London) (01.02.1996)
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MARICHAL, P, KOYMANS, L, WILLEMSENS, S, BELLENS, D, VERHASSELT, P, LUYTEN, W, BORGERS, M, RAMAEKERS, F. C. S, ODDS, F. C, BOSSCHE, H. V
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Published in Microbiology (Society for General Microbiology) (01.10.1999)
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Ludovici, Donald W., De Corte, Bart L., Kukla, Michael J., Ye, Hong, Ho, Chih Y., Lichtenstein, Mark A., Kavash, Robert W., Andries, Koen, de Béthune, Marie-Pierre, Azijn, Hilde, Pauwels, Rudi, Lewi, Paul J., Heeres, Jan, Koymans, Lucien M.H., de Jonge, Marc R., Van Aken, Koen J.A., Daeyaert, Frederik F.D., Das, Kalyan, Arnold, Edward, Janssen, Paul A.J.
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
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Structure of HIV-1 RT/TIBO R 86183 complex reveals similarity in the binding of diverse nonnucleoside inhibitors
Ding, J, Das, K, Moereels, H, Koymans, L, Andries, K, Janssen, P A, Hughes, S H, Arnold, E
Published in Nature structural biology (01.05.1995)
Published in Nature structural biology (01.05.1995)
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