Design, synthesis and identification of novel benzimidazole derivatives as highly potent NPY Y5 receptor antagonists with attractive in vitro ADME profiles
Tamura, Yuusuke, Omori, Naoki, Kouyama, Naoki, Nishiura, Yuji, Hayashi, Kyouhei, Watanabe, Kana, Tanaka, Yukari, Chiba, Takeshi, Yukioka, Hideo, Sato, Hiroki, Okuno, Takayuki
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
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Journal Article
Identification of a novel and orally available benzimidazole derivative as an NPY Y5 receptor antagonist with in vivo efficacy
Tamura, Yuusuke, Omori, Naoki, Kouyama, Naoki, Nishiura, Yuji, Hayashi, Kyouhei, Watanabe, Kana, Tanaka, Yukari, Chiba, Takeshi, Yukioka, Hideo, Sato, Hiroki, Okuno, Takayuki
Published in Bioorganic & medicinal chemistry letters (01.11.2012)
Published in Bioorganic & medicinal chemistry letters (01.11.2012)
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Journal Article
Hit to lead SAR study on benzoxazole derivatives for an NPY Y5 antagonist
Omori, Naoki, Kouyama, Naoki, Yukimasa, Akira, Watanabe, Kana, Yokota, Yasunori, Tanioka, Hideki, Nambu, Hirohide, Yukioka, Hideo, Sato, Norihito, Tanaka, Yukari, Sekiguchi, Kazutaka, Okuno, Takayuki
Published in Bioorganic & medicinal chemistry letters (01.03.2012)
Published in Bioorganic & medicinal chemistry letters (01.03.2012)
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Journal Article
Identification of a novel benzimidazole derivative as a highly potent NPY Y5 receptor antagonist with an anti-obesity profile
Tamura, Yuusuke, Hayashi, Kyouhei, Omori, Naoki, Nishiura, Yuji, Watanabe, Kana, Tanaka, Nobuyuki, Fujioka, Masahiko, Kouyama, Naoki, Yukimasa, Akira, Tanaka, Yukari, Chiba, Takeshi, Tanioka, Hideki, Nambu, Hirohide, Yukioka, Hideo, Sato, Hiroki, Okuno, Takayuki
Published in Bioorganic & medicinal chemistry letters (01.01.2013)
Published in Bioorganic & medicinal chemistry letters (01.01.2013)
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Journal Article
COMPOUND HAVING NPY Y5 RECEPTOR ANTAGONIST ACTIVITY
YARI HIROSHI, HASHIZUME HIROSHI, TONOGAKI KEISUKE, SAKAGAMI MASAHIRO, TANAKA SATORU, OKUNO TAKAYUKI, KOUYAMA NAOKI
Year of Publication 24.12.2010
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Year of Publication 24.12.2010
Patent
COMPOUND HAVING NPY Y5 RECEPTOR ANTAGONIST ACTIVITY
OKUNO, TAKAYUKI, TANAKA, SATORU, YARI, HIROSHI, KOUYAMA, NAOKI, TONOGAKI, KEISUKE, HASHIZUME, HIROSHI, SAKAGAMI, MASAHIRO
Year of Publication 29.10.2009
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Year of Publication 29.10.2009
Patent