Splicing factor SF3b as a target of the antitumor natural product pladienolide
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Published in Nature chemical biology (01.09.2007)
Published in Nature chemical biology (01.09.2007)
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Apratoxin A Shows Novel Pancreas-Targeting Activity through the Binding of Sec 61
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Published in Molecular cancer therapeutics (01.06.2016)
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Total Synthesis of the Potent Antitumor Macrolides Pladienolide B and D
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Published in Angewandte Chemie (International ed.) (01.01.2007)
Published in Angewandte Chemie (International ed.) (01.01.2007)
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Stereochemistry of Pladienolide B
Asai, Naoki, Kotake, Yoshihiko, Niijima, Jun, Fukuda, Yoshio, Uehara, Taisuke, Sakai, Takashi
Published in Journal of antibiotics (01.06.2007)
Published in Journal of antibiotics (01.06.2007)
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Microregional antitumor activity of a small-molecule hypoxia-inducible factor 1 inhibitor
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Published in International journal of molecular medicine (01.04.2012)
Published in International journal of molecular medicine (01.04.2012)
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Synthesis and Evaluation of Novel Pyrimido-Acridone, -Phenoxadine, and -Carbazole as Topoisomerase II Inhibitors
Kamata, Junichi, Okada, Toshimi, Kotake, Yoshihiko, Niijima, Jun, Nakamura, Katsuji, Uenaka, Toshimitsu, Yamaguchi, Atsumi, Tsukahara, Kappei, Nagasu, Takeshi, Koyanagi, Nozomu, Kitoh, Kyosuke, Yoshimatsu, Kentaro, Yoshino, Hiroshi, Sugumi, Hiroyuki
Published in Chemical & Pharmaceutical Bulletin (01.09.2004)
Published in Chemical & Pharmaceutical Bulletin (01.09.2004)
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Total Synthesis of the Potent Antitumor Macrolides Pladienolide B and D
Kanada, Regina M, Itoh, Daisuke, Nagai, Mitsuo, Niijima, Jun, Asai, Naoki, Mizui, Yoshiharu, Abe, Shinya, Kotake, Yoshihiko
Published in Angewandte Chemie (International ed.) (26.11.2007)
Published in Angewandte Chemie (International ed.) (26.11.2007)
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Selective degradation of splicing factor CAPERα by anticancer sulfonamides
Uehara, Taisuke, Minoshima, Yukinori, Sagane, Koji, Sugi, Naoko Hata, Mitsuhashi, Kaoru Ogawa, Yamamoto, Noboru, Kamiyama, Hiroshi, Takahashi, Kentaro, Kotake, Yoshihiko, Uesugi, Mai, Yokoi, Akira, Inoue, Atsushi, Yoshida, Taku, Mabuchi, Miyuki, Tanaka, Akito, Owa, Takashi
Published in Nature chemical biology (01.06.2017)
Published in Nature chemical biology (01.06.2017)
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A novel carbazole topoisomerase II poison, ER‐37328: potent tumoricidal activity against human solid tumors in vitro and in vivo
Nakamura, Katsuji, Uenaka, Toshimitsu, Nagasu, Takeshi, Sugumi, Hiroyuki, Yamaguchi, Atsumi, Kotake, Yoshihiko, Okada, Toshimi, Kamata, Junichi, Niijima, Jun, Taniguchi, Tomoyoshi, Koyanagi, Nozomu, Yoshino, Hiroshi, Kitoh, Kyosuke, Yoshimatsu, Kentaro
Published in Cancer science (01.01.2003)
Published in Cancer science (01.01.2003)
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Antitumor Activity of ER-37328, a Novel Carbazole Topoisomerase II Inhibitor
Nakamura, Katsuji, Sugumi, Hiroyuki, Yamaguchi, Atsumi, Uenaka, Toshimitsu, Kotake, Yoshihiko, Okada, Toshimi, Kamata, Junichi, Niijima, Jun, Nagasu, Takeshi, Koyanagi, Nozomu, Yoshino, Hiroshi, Kitoh, Kyosuke, Yoshimatsu, Kentaro
Published in Molecular cancer therapeutics (01.01.2002)
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Published in Molecular cancer therapeutics (01.01.2002)
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Biological validation that SF3b is a target of the antitumor macrolide pladienolide
Yokoi, Akira, Kotake, Yoshihiko, Takahashi, Kentaro, Kadowaki, Tadashi, Matsumoto, Yoshiko, Minoshima, Yukinori, Sugi, Naoko H., Sagane, Koji, Hamaguchi, Makoto, Iwata, Masao, Mizui, Yoshiharu
Published in The FEBS journal (01.12.2011)
Published in The FEBS journal (01.12.2011)
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Identification of a novel ALDH1A3‐selective inhibitor by a chemical probe with unrelated bioactivity: An approach to affinity‐based drug target discovery
Kamiyama, Hiroshi, Miyano, Masayuki, Ito, Daisuke, Kimura, Takayuki, Hagiwara, Koji, Kogai, Hiroyuki, Kaburagi, Yosuke, Kotake, Yoshihiko, Takase, Yasutaka
Published in Chemical biology & drug design (01.03.2023)
Published in Chemical biology & drug design (01.03.2023)
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Abstract 1377: Chemical probe-based approach clarifies binding of receptor tyrosine kinases (RTKs) to lenvatinib in preclinical models
Kimura, Takayuki, Yamamoto, Noboru, Kamiyama, Hiroshi, Kawada, Megumi Ikemori, Yamamoto, Akihiko, Kotake, Yoshihiko, Takase, Yasutaka, Funahashi, Yasuhiro, Oda, Yoshiya
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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헤르복시디엔 항체-약물 접합체 및 사용 방법
KOTAKE YOSHIHIKO, OKUBO SHINYA, ARAI KENZO, MIYANO MASAYUKI, PALACINO JAMES, MURAI NORIO, FISHKIN NATHAN, SAMARAKOON THIWANKA
Year of Publication 19.08.2021
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Year of Publication 19.08.2021
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Selective degradation of splicing factor CAPER[alpha] by anticancer sulfonamides
Uehara, Taisuke, Minoshima, Yukinori, Sagane, Koji, Sugi, Naoko Hata, Mitsuhashi, Kaoru Ogawa, Yamamoto, Noboru, Kamiyama, Hiroshi, Takahashi, Kentaro, Kotake, Yoshihiko, Uesugi, Mai, Yokoi, Akira, Inoue, Atsushi, Yoshida, Taku, Mabuchi, Miyuki, Tanaka, Akito, Owa, Takashi
Published in Nature chemical biology (01.06.2017)
Published in Nature chemical biology (01.06.2017)
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Small molecule schweinfurthins selectively inhibit cancer cell proliferation and mTOR/AKT signaling by interfering with trans-Golgi-network trafficking
Bao, Xingfeng, Zheng, Wanjun, Sugi, Naoko Hata, Agarwala, Kishan L, Xu, Qunli, Wang, Zichun, Tendyke, Karen, Lee, Winnie, Parent, Lana, Li, Wei, Cheng, Hongsheng, Shen, Yongchun, Taylor, Noel, Dezso, Zoltan, Du, Hong, Kotake, Yoshihiko, Zhao, Nanding, Wang, John, Postema, Maarten, Woodall-Jappe, Mary, Takase, Yasutaka, Uenaka, Toshimitsu, Kingston, David G I, Nomoto, Kenichi
Published in Cancer biology & therapy (01.01.2015)
Published in Cancer biology & therapy (01.01.2015)
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CERTAIN PLADIENOLIDE COMPOUNDS AND METHODS OF USE
JASON T LOWE, DOMINIC REYNOLDS, LIU XIANG, PARCHAREE TIVITMAHAISOON, ENDO ATSUSHI, WANG JOHN, REGINA MIKIE KANADA SONOBE, ARAI KENZO, GREGG F KEANEY, ZHENG GUO ZHU, LISA A MARCAURELLE, MURAI NORIO, BAUDOUIN GERARD, ANDREW COOK, HAO MING-HONG, MARTA NEVALAINEN, NICHOLAS C GEARHART, LUO TOUPING, SUDEEP PRAJAPATI, JAMES PALACINO, KOTAKE YOSHIHIKO, NAGAO SATOSHI, KIRA KAZUNOBU, MORGAN WELZEL O'SHEA, MIYANO MASAYUKI, SHELBY ELLERY
Year of Publication 24.10.2023
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Year of Publication 24.10.2023
Patent
Synthesis and structure–activity relationships of novel, potent, orally active hypoxia-inducible factor-1 inhibitors
Nagao, Satoshi, Yamane, Yoshinobu, Funasaka, Setsuo, Tanaka, Keigo, Miyazaki, Kazuki, Kotake, Yoshihiko, Kamata, Jun-ichi, Watanabe-Miyano, Saori, Toyama, Osamu, Ozawa, Yoichi, Mizui, Yoshiharu, Okamoto, Kiyoshi, Ito, Daisuke
Published in Bioorganic & medicinal chemistry (01.10.2014)
Published in Bioorganic & medicinal chemistry (01.10.2014)
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플라디에놀리드 화합물 및 그의 용도
HAO MING HONG, KANADA SONOBE REGINA MIKIE, LIU XIANG, NEVALAINEN MARTA, ENDO ATSUSHI, WANG JOHN, ARAI KENZO, REYNOLDS DOMINIC, GEARHART NICHOLAS C, ZHENG GUO ZHU, MURAI NORIO, KEANEY GREGG F, COOK ANDREW, LUO TOUPING, TIVITMAHAISOON PARCHAREE, O'SHEA MORGAN WELZEL, LOWE JASON T, ELLERY SHELBY, GERARD BAUDOUIN, KOTAKE YOSHIHIKO, MARCAURELLE LISA A, NAGAO SATOSHI, KIRA KAZUNOBU, MIYANO MASAYUKI, PRAJAPATI SUDEEP, PALACINO JAMES
Year of Publication 19.01.2021
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Year of Publication 19.01.2021
Patent
2-Alkynyl-8-aryl-9-methyladenines as Novel Adenosine Receptor Antagonists: Their Synthesis and Structure−Activity Relationships toward Hepatic Glucose Production Induced via Agonism of the A2B Receptor
Harada, Hitoshi, Asano, Osamu, Hoshino, Yorihisa, Yoshikawa, Seiji, Matsukura, Masayuki, Kabasawa, Yasuhiro, Niijima, Jun, Kotake, Yoshihiko, Watanabe, Nobuhisa, Kawata, Tsutomu, Inoue, Takashi, Horizoe, Tatsuo, Yasuda, Nobuyuki, Minami, Hiroe, Nagata, Kaya, Murakami, Manabu, Nagaoka, Junsaku, Kobayashi, Seiichi, Tanaka, Isao, Abe, Shinya
Published in Journal of medicinal chemistry (18.01.2001)
Published in Journal of medicinal chemistry (18.01.2001)
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