Identification of Atuveciclib (BAY 1143572), the First Highly Selective, Clinical PTEFb/CDK9 Inhibitor for the Treatment of Cancer
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Published in ChemMedChem (08.11.2017)
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Impact of Isotype-Selective Estrogen Receptor Agonists on Ovarian Function
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Published in Proceedings of the National Academy of Sciences - PNAS (06.04.2004)
Published in Proceedings of the National Academy of Sciences - PNAS (06.04.2004)
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Changing for the Better: Discovery of the Highly Potent and Selective CDK9 Inhibitor VIP152 Suitable for Once Weekly Intravenous Dosing for the Treatment of Cancer
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Published in Journal of medicinal chemistry (12.08.2021)
Published in Journal of medicinal chemistry (12.08.2021)
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Novel Mps1 Kinase Inhibitors with Potent Antitumor Activity
Wengner, Antje M, Siemeister, Gerhard, Koppitz, Marcus, Schulze, Volker, Kosemund, Dirk, Klar, Ulrich, Stoeckigt, Detlef, Neuhaus, Roland, Lienau, Philip, Bader, Benjamin, Prechtl, Stefan, Raschke, Marian, Frisk, Anna-Lena, von Ahsen, Oliver, Michels, Martin, Kreft, Bertolt, von Nussbaum, Franz, Brands, Michael, Mumberg, Dominik, Ziegelbauer, Karl
Published in Molecular cancer therapeutics (01.04.2016)
Published in Molecular cancer therapeutics (01.04.2016)
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Treating Cancer by Spindle Assembly Checkpoint Abrogation: Discovery of Two Clinical Candidates, BAY 1161909 and BAY 1217389, Targeting MPS1 Kinase
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Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
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Abstract 984: Identification of potent and highly selective PTEFb inhibitor BAY 1251152 for the treatment of cancer: from p.o. to i.v. application via scaffold hops
Luecking, Ulrich T., Scholz, Arne, Kosemund, Dirk, Bohlmann, Rolf, Briem, Hans, Lienau, Philip, Siemeister, Gerhard, Terebesi, Ildiko, Meyer, Kirstin, Prelle, Katja, Valencia, Ray, Ince, Stuart, Nussbaum, Franz von, Mumberg, Dominik, Ziegelbauer, Karl, Brands, Michael
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Hillisch, Alexander, Peters, Olaf, Kosemund, Dirk, Müller, Gerd, Walter, Alexander, Schneider, Birgitt, Reddersen, Gudrun, Elger, Walter, Fritzemeier, Karl-Heinrich
Published in Molecular endocrinology (Baltimore, Md.) (01.07.2004)
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면역 활성화를 위한 DGK알파 억제제로서의 치환된 아미노퀴놀론
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Year of Publication 02.09.2022
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DELBECK MARTINA, KOSEMUND DIRK, KALTHOF BERND, SUESSMEIER FRANK, LUSTIG KLEMENS, HAERTER MICHAEL, CANCHO GRANDE YOLANDA
Year of Publication 17.05.2019
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Year of Publication 17.05.2019
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Abstract 3090: Novel Mps1 kinase inhibitors with potent anti-tumor activity
Wengner, Antje Margret, Siemeister, Gerhard, Koppitz, Marcus, Schulze, Volker, Kosemund, Dirk, Klar, Ulrich, Stoeckigt, Detlef, Neuhaus, Roland, Lienau, Philip, Bader, Benjamin, Prechtl, Stefan, Doehr, Olaf, Raschke, Marian, von Ahsen, Oliver, Elbi, Cem, Bruns, Ingmar, Michels, Martin, Kreft, Bertolt, von Nussbaum, Franz, Brands, Michael, Mumberg, Dominik, Ziegelbauer, Karl
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Abstract 2828: Rapid identification of potent and highly selective, oral PTEFb Inhibitor BAY 1143572 with first in class potential
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Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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5-FLUORO-N-(PYRIDIN-2-YL)PYRIDIN-2-AMINE DERIVATIVES CONTAINING A SULFOXIMINE GROUP
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Year of Publication 15.07.2015
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