Discovery of E2730, a novel selective uncompetitive GAT1 inhibitor, as a candidate for anti‐seizure medication
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Published in Epilepsia open (01.09.2023)
Published in Epilepsia open (01.09.2023)
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Inhibitory effect of orally administered donepezil hydrochloride (E2020), a novel treatment for Alzheimer's disease, on cholinesterase activity in rats
Kosasa, Takashi, Kuriya, Yuka, Matsui, Kenji, Yamanishi, Yoshiharu
Published in European journal of pharmacology (18.02.2000)
Published in European journal of pharmacology (18.02.2000)
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E2511, a novel small compound TrkA biased positive allosteric modulator, reinnervates cholinergic neuron and activates cholinergic functions in non‐clinical studies
Tomioka, Takeyasu, Hiramatsu, Naoki, Moriyama, Yoshiyuki, Kosasa, Takashi
Published in Alzheimer's & dementia (01.06.2023)
Published in Alzheimer's & dementia (01.06.2023)
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Journal Article
E2511, a novel small compound TrkA allosteric modulator, induces a specific trophic signaling via direct binding to TrkA, and can reverse the loss of choline acetyltransferase (ChAT) positive neurons in transgenic models of AD
Tomioka, Takeyasu, Moriyama, Yoshiyuki, Hiramatsu, Naoki, Kosasa, Takashi, Kondo, Keita, Wakita, Hisashi
Published in Alzheimer's & dementia (01.12.2021)
Published in Alzheimer's & dementia (01.12.2021)
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Journal Article
Donepezil attenuates excitotoxic damage induced by membrane depolarization of cortical neurons exposed to veratridine
Akasofu, Shigeru, Sawada, Kohei, Kosasa, Takashi, Hihara, Hiroe, Ogura, Hiroo, Akaike, Akinori
Published in European journal of pharmacology (07.07.2008)
Published in European journal of pharmacology (07.07.2008)
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Journal Article
NOVEL INDANESULFAMIDE DERIVATIVE
KAZUTA YUJI, SORIMACHI KEIICHI, HIGASHIYAMA HIROYUKI, KOSASA TAKASHI, WATANABE TORU, TERAMOTO TETSUYUKI, ISHIKAWA YUKIO, SAITO MINAKO, KITA YOICHI, HANADA TAKAHISA, TANAKA TOSHIAKI
Year of Publication 30.03.2015
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Year of Publication 30.03.2015
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