Selective Inhibitors of Protein Methyltransferases
Kaniskan, H. Ümit, Konze, Kyle D, Jin, Jian
Published in Journal of medicinal chemistry (26.02.2015)
Published in Journal of medicinal chemistry (26.02.2015)
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Journal Article
Targeting EZH2 and PRC2 dependence as novel anticancer therapy
Xu, Bowen, Konze, Kyle D, Jin, Jian, Wang, Gang Greg
Published in Experimental hematology (01.08.2015)
Published in Experimental hematology (01.08.2015)
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Reaction-Based Enumeration, Active Learning, and Free Energy Calculations To Rapidly Explore Synthetically Tractable Chemical Space and Optimize Potency of Cyclin-Dependent Kinase 2 Inhibitors
Konze, Kyle D, Bos, Pieter H, Dahlgren, Markus K, Leswing, Karl, Tubert-Brohman, Ivan, Bortolato, Andrea, Robbason, Braxton, Abel, Robert, Bhat, Sathesh
Published in Journal of chemical information and modeling (23.09.2019)
Published in Journal of chemical information and modeling (23.09.2019)
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Selective inhibition of EZH2 and EZH1 enzymatic activity by a small molecule suppresses MLL-rearranged leukemia
Xu, Bowen, On, Doan M., Ma, Anqi, Parton, Trevor, Konze, Kyle D., Pattenden, Samantha G., Allison, David F., Cai, Ling, Rockowitz, Shira, Liu, Shichong, Liu, Ying, Li, Fengling, Vedadi, Masoud, Frye, Stephen V., Garcia, Benjamin A., Zheng, Deyou, Jin, Jian, Wang, Gang Greg
Published in Blood (08.01.2015)
Published in Blood (08.01.2015)
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Combining Cloud-Based Free-Energy Calculations, Synthetically Aware Enumerations, and Goal-Directed Generative Machine Learning for Rapid Large-Scale Chemical Exploration and Optimization
Ghanakota, Phani, Bos, Pieter H, Konze, Kyle D, Staker, Joshua, Marques, Gabriel, Marshall, Kyle, Leswing, Karl, Abel, Robert, Bhat, Sathesh
Published in Journal of chemical information and modeling (28.09.2020)
Published in Journal of chemical information and modeling (28.09.2020)
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An Orally Bioavailable Chemical Probe of the Lysine Methyltransferases EZH2 and EZH1
Konze, Kyle D, Ma, Anqi, Li, Fengling, Barsyte-Lovejoy, Dalia, Parton, Trevor, MacNevin, Christopher J, Liu, Feng, Gao, Cen, Huang, Xi-Ping, Kuznetsova, Ekaterina, Rougie, Marie, Jiang, Alice, Pattenden, Samantha G, Norris, Jacqueline L, James, Lindsey I, Roth, Bryan L, Brown, Peter J, Frye, Stephen V, Arrowsmith, Cheryl H, Hahn, Klaus M, Wang, Gang Greg, Vedadi, Masoud, Jin, Jian
Published in ACS chemical biology (21.06.2013)
Published in ACS chemical biology (21.06.2013)
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Structure–Activity Relationship Studies for Enhancer of Zeste Homologue 2 (EZH2) and Enhancer of Zeste Homologue 1 (EZH1) Inhibitors
Yang, Xiaobao, Li, Fengling, Konze, Kyle D, Meslamani, Jamel, Ma, Anqi, Brown, Peter J, Zhou, Ming-Ming, Arrowsmith, Cheryl H, Kaniskan, H. Ümit, Vedadi, Masoud, Jin, Jian
Published in Journal of medicinal chemistry (25.08.2016)
Published in Journal of medicinal chemistry (25.08.2016)
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A Chemical Tool for In Vitro and In Vivo Precipitation of Lysine Methyltransferase G9a
Konze, Kyle D., Pattenden, Samantha G., Liu, Feng, Barsyte-Lovejoy, Dalia, Li, Fengling, Simon, Jeremy M., Davis, Ian J., Vedadi, Masoud, Jin, Jian
Published in ChemMedChem (01.03.2014)
Published in ChemMedChem (01.03.2014)
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Multi-omic Dissection of Oncogenically Active Epiproteomes Identifies Drivers of Proliferative and Invasive Breast Tumors
Wrobel, John A., Xie, Ling, Wang, Li, Liu, Cui, Rashid, Naim, Gallagher, Kristalyn K., Xiong, Yan, Konze, Kyle D., Jin, Jian, Gatza, Michael L., Chen, Xian
Published in iScience (26.07.2019)
Published in iScience (26.07.2019)
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Journal Article
Inside Cover: A Chemical Tool for In Vitro and In Vivo Precipitation of Lysine Methyltransferase G9a (ChemMedChem 3/2014)
Konze, Kyle D., Pattenden, Samantha G., Liu, Feng, Barsyte-Lovejoy, Dalia, Li, Fengling, Simon, Jeremy M., Davis, Ian J., Vedadi, Masoud, Jin, Jian
Published in ChemMedChem (01.03.2014)
Published in ChemMedChem (01.03.2014)
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KDM5 억제 활성을 갖는 화합물 및 이의 약학적 용도
KRILOV GORAN, INOYAMA DAIGO, KAKUUCHI AKITO, ZHANG YAN, RUVINSKY ANATOLY, SVENSSON MATS, KONZE KYLE, TAKAHASHI HIDENORI, ASADA MASAKI, UMEMURA SHUHEI
Year of Publication 12.01.2023
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Year of Publication 12.01.2023
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HAHN KRISTOPHER NEIL, LIPPA BLAISE SCOTT, HARRISON BRYCE ALDEN, SVENSSON MATS AKE, GERASYUTO ALEKSEY LGOREVICH, LIN FU YANG, BURSAVICH MATTHEW GREGORY, KONZE KYLE DAVID, ROGERS BRUCE NELSEN, TROAST DAWN MARIE, LUGOVSKOY ALEXEY ALEXANDROVICH, BREWER MARK
Year of Publication 30.11.2023
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Year of Publication 30.11.2023
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CUI DAN, LIN FU YANG, KIM BYUNGCHAN, BURSAVICH MATTHEW G, ROGERS BRUCE N, TROAST DAWN M, HOUANG EVELYNE, KONZE KYLE D, LIPPA BLAISE S, RAFI SALMA, ZAHLER ROBERT, DOWLING JAMES E, HICKEY EUGENE, HARRISON BRYCE A, GERASYUTO ALEKSEY I, DAY TYLER, HAHN KRISTOPHER N, ZHONG CHENG
Year of Publication 19.06.2023
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Year of Publication 19.06.2023
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인간 인테그린 α4β7의 억제
CUI DAN, LIN FU YANG, KIM BYUNGCHAN, BURSAVICH MATTHEW G, ROGERS BRUCE N, TROAST DAWN M, HOUANG EVELYNE, KONZE KYLE D, LIPPA BLAISE S, RAFI SALMA, ZAHLER ROBERT, DOWLING JAMES E, HICKEY EUGENE, HARRISON BRYCE A, GERASYUTO ALEKSEY I, DAY TYLER, HAHN KRISTOPHER N, ZHONG CHENG
Year of Publication 20.07.2022
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Year of Publication 20.07.2022
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αvβ6 인테그린 억제
SOSA BRIAN, LIN FU YANG, BORTOLATO ANDREA, KIM BYUNGCHAN, BURSAVICH MATTHEW G, ROGERS BRUCE N, TROAST DAWN M, KONZE KYLE D, LIPPA BLAISE S, DOWLING JAMES E, HICKEY EUGENE, HARRISON BRYCE A, GERASYUTO ALEKSEY I, QIAO QI, DAY TYLER, SVENSSON MATS A, HAHN KRISTOPHER N, ZHONG CHENG
Year of Publication 04.06.2021
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Year of Publication 04.06.2021
Patent
A chemical tool for chemiprecipitation of the lysine methyltransferase, G9a, in vitro and in vivo
Konze, Kyle D., Pattenden, Samantha G., Liu, Feng, Barsyte-Lovejoy, Dalia, Li, Fengling, Simon, Jeremy M., Davis, Ian J., Vedadi, Masoud, Jin, Jian
Published in ChemMedChem (17.01.2014)
Published in ChemMedChem (17.01.2014)
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αvβ6 인테그린 억제제
HAHN KRISTOPHER NEIL, LIPPA BLAISE SCOTT, HARRISON BRYCE ALDEN, SVENSSON MATS AKE, GERASYUTO ALEKSEY LGOREVICH, LIN FU YANG, BURSAVICH MATTHEW GREGORY, KONZE KYLE DAVID, ROGERS BRUCE NELSEN, TROAST DAWN MARIE, LUGOVSKOY ALEXEY ALEXANDROVICH, BREWER MARK
Year of Publication 03.12.2019
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Year of Publication 03.12.2019
Patent