Discovery and structure-activity relationships study of positive allosteric modulators of the M3 muscarinic acetylcholine receptor
Tanaka, Hiroaki, Negoro, Kenji, Koike, Takanori, Tsukamoto, Issei, Yokoyama, Kazuhiro, Maeda, Jun, Inagaki, Yusuke, Shimoshige, Yukinori, Ino, Katsutoshi, Ishizu, Kenichiro, Takahashi, Taisuke
Published in Bioorganic & medicinal chemistry (01.07.2020)
Published in Bioorganic & medicinal chemistry (01.07.2020)
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Journal Article
Discovery and Biological Evaluation of Potent and Orally Active Human 11β-Hydroxysteroid Dehydrogenase Type 1 Inhibitors for the Treatment of Type 2 Diabetes Mellitus
Koike, Takanori, Shiraki, Ryota, Sasuga, Daisuke, Hosaka, Mitsuru, Kawano, Tomoaki, Fukudome, Hiroki, Kurosawa, Kazuo, Moritomo, Ayako, Mimasu, Shinya, Ishii, Hirofumi, Yoshimura, Seiji
Published in Chemical & pharmaceutical bulletin (01.08.2019)
Published in Chemical & pharmaceutical bulletin (01.08.2019)
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Journal Article
Discovery and Biological Evaluation of Potent and Orally Active Human 11β-Hydroxysteroid Dehydrogenase Type 1 Inhibitors for the Treatment of Type 2 Diabetes Mellitus
Takanori Koike, Ryota Shiraki, Daisuke Sasuga, Mitsuru Hosaka, Tomoaki Kawano, Hiroki Fukudome, Kazuo Kurosawa, Ayako Moritomo, Shinya Mimasu, Hirofumi Ishii, Seiji Yoshimura
Published in Chemical and Pharmaceutical Bulletin (01.08.2019)
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Published in Chemical and Pharmaceutical Bulletin (01.08.2019)
Journal Article
Design, synthesis and biological activity of selective and orally available TF/FVIIa complex inhibitors containing non-amidine P1 ligands
Miura, Masanori, Seki, Norio, Koike, Takanori, Ishihara, Tsukasa, Niimi, Tatsuya, Hirayama, Fukushi, Shigenaga, Takeshi, Sakai-Moritani, Yumiko, Tagawa, Ayako, Kawasaki, Tomihisa, Sakamoto, Shuichi, Okada, Minoru, Ohta, Mitsuaki, Tsukamoto, Shin-ichi
Published in Bioorganic & medicinal chemistry (2007)
Published in Bioorganic & medicinal chemistry (2007)
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Journal Article
Prediction of thermal transport characteristics of microgroove evaporator (Validation of prediction model by measurement of transported heat and capillary-rise length)
SHIRAKASHI, Ryo, KOIKE, Takanori, UEMURA, Mitsuhiro, HAGIYA, Isao, WATANABE, Yuki, FUJITA, Wataru
Published in Kikai Gakkai ronbunshū = Transactions of the Japan Society of Mechanical Engineers (01.01.2014)
Published in Kikai Gakkai ronbunshū = Transactions of the Japan Society of Mechanical Engineers (01.01.2014)
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Journal Article
Lipase-catalyzed preparation of both enantiomers of methyl jasmonate
Kiyota, Hiromasa, Higashi, Emi, Koike, Takanori, Oritani, Takayuki
Published in Tetrahedron: asymmetry (08.05.2001)
Published in Tetrahedron: asymmetry (08.05.2001)
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Journal Article
One-Pot Preparation of Unsymmetrical Biaryls via Suzuki Cross-Coupling Reaction of Aryl Halide using Phase-Transfer Catalyst in a Biphasic Solvent System
Miura, Masanori, Koike, Takanori, Ishihara, Tsukasa, Sakamoto, Shuichi, Okada, Minoru, Ohta, Mitsuaki, Tsukamoto, Shin-ichi
Published in Synthetic communications (01.03.2007)
Published in Synthetic communications (01.03.2007)
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Journal Article
Discovery and biological evaluation of 1-{2,7-diazaspiro[3.5]nonan-2-yl}prop-2-en-1-one derivatives as covalent inhibitors of KRAS G12C with favorable metabolic stability and anti-tumor activity
Imaizumi, Tomoyoshi, Akaiwa, Michinori, Abe, Tomoaki, Nigawara, Takahiro, Koike, Takanori, Satake, Yoshiki, Watanabe, Kazushi, Kaneko, Osamu, Amano, Yasushi, Mori, Kenichi, Yamanaka, Yosuke, Nagashima, Takeyuki, Shimazaki, Masashi, Kuramoto, Kazuyuki
Published in Bioorganic & medicinal chemistry (01.10.2022)
Published in Bioorganic & medicinal chemistry (01.10.2022)
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Journal Article
Discovery of ASP6918, a KRAS G12C inhibitor: Synthesis and structure-activity relationships of 1-{2,7-diazaspiro[3.5]non-2-yl} prop-2-en-1-one derivatives as covalent inhibitors with good potency and oral activity for the treatment of solid tumors
Imaizumi, Tomoyoshi, Shimada, Itsuro, Satake, Yoshiki, Yamaki, Susumu, Koike, Takanori, Nigawara, Takahiro, Kaneko, Osamu, Amano, Yasushi, Mori, Kenichi, Yamanaka, Yosuke, Nakayama, Ayako, Nishizono, Yoshihiro, Shimazaki, Masashi, Nagashima, Takeyuki, Kuramoto, Kazuyuki
Published in Bioorganic & medicinal chemistry (15.01.2024)
Published in Bioorganic & medicinal chemistry (15.01.2024)
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Journal Article
Discovery and structure -activity relationships study of positive allosteric modulators of the M 3 muscarinic acetylcholine receptor
Tanaka, Hiroaki, Negoro, Kenji, Koike, Takanori, Tsukamoto, Issei, Yokoyama, Kazuhiro, Maeda, Jun, Inagaki, Yusuke, Shimoshige, Yukinori, Ino, Katsutoshi, Ishizu, Kenichiro, Takahashi, Taisuke
Published in Bioorganic & medicinal chemistry (01.07.2020)
Published in Bioorganic & medicinal chemistry (01.07.2020)
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Journal Article
AIR CONDITIONER
MIZUNO Yuki, HATOMURA Takeshi, HANYUDA Taku, KOIKE Takanori, ISHIMURA Shohei, WASHIYAMA Hiroki
Year of Publication 18.04.2024
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Year of Publication 18.04.2024
Patent
AIR CONDITIONING DEVICE
NISHIO Jun, MIYAWAKI Kosuke, OKANO Hiroyuki, HATOMURA Takeshi, OGATA Keito, KOIKE Takanori, TAKENAKA Naofumi
Year of Publication 23.11.2023
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Year of Publication 23.11.2023
Patent
REFRIGERATION CYCLE DEVICE
NISHIO Jun, OKANO Hiroyuki, MORIMOTO Osamu, HATOMURA Takeshi, KOIKE Takanori, WAKAMOTO Shinichi, SHINOZAKI Kazuyoshi, TAKENAKA Naofumi
Year of Publication 27.07.2023
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Year of Publication 27.07.2023
Patent