Developing lipid nanoparticle-based siRNA therapeutics for hepatocellular carcinoma using an integrated approach
Li, Leiming, Wang, Rongqi, Wilcox, Denise, Sarthy, Aparna, Lin, Xiaoyu, Huang, Xiaoli, Tian, Lu, Dande, Prasad, Hubbard, Robert D, Hansen, Todd M, Wada, Carol, Zhao, Xiaobin, Kohlbrenner, William M, Fesik, Stephen W, Shen, Yu
Published in Molecular cancer therapeutics (01.11.2013)
Published in Molecular cancer therapeutics (01.11.2013)
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Activity of a Potent Hepatitis C Virus Polymerase Inhibitor in the Chimpanzee Model
Chen, Chih-Ming, He, Yupeng, Lu, Liangjun, Lim, Hock Ben, Tripathi, Rakesh L, Middleton, Tim, Hernandez, Lisa E, Beno, David W A, Long, Michelle A, Kati, Warren M, Bosse, Todd D, Larson, Daniel P, Wagner, Rolf, Lanford, Robert E, Kohlbrenner, William E, Kempf, Dale J, Pilot-Matias, Tami J, Molla, Akhteruzzaman
Published in Antimicrobial Agents and Chemotherapy (01.12.2007)
Published in Antimicrobial Agents and Chemotherapy (01.12.2007)
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A robust in vivo positive-readout system for monitoring siRNA delivery to xenograft tumors
Lin, Xiaoyu, Li, Leiming, Wang, Rongqi, Wilcox, Denise, Zhao, Xiaobin, Song, Jingfeng, Huang, Xiaoli, Hansen, T Matthew, Dande, Prasad, Wada, Carol, Hubbard, Robert D, Kohlbrenner, William M, Fesik, Stephen W, Shen, Yu
Published in RNA (Cambridge) (01.04.2011)
Published in RNA (Cambridge) (01.04.2011)
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Small-Sized Human Immunodeficiency Virus Type-1 Protease Inhibitors Containing Allophenylnorstatine to Explore the S2′ Pocket
Hidaka, Koushi, Kimura, Tooru, Abdel-Rahman, Hamdy M, Nguyen, Jeffrey-Tri, McDaniel, Keith F, Kohlbrenner, William E, Molla, Akhteruzzaman, Adachi, Motoyasu, Tamada, Taro, Kuroki, Ryota, Katsuki, Noriko, Tanaka, Yoshiaki, Matsumoto, Hikaru, Wang, Jun, Hayashi, Yoshio, Kempf, Dale J, Kiso, Yoshiaki
Published in Journal of medicinal chemistry (10.12.2009)
Published in Journal of medicinal chemistry (10.12.2009)
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In Vitro Characterization of A-315675, a Highly Potent Inhibitor of A and B Strain Influenza Virus Neuraminidases and Influenza Virus Replication
KATI, Warren M, MONTGOMERY, Debra, KOHLBRENNER, William, CARRICK, Robert, GUBAREVA, Larisa, MARING, Clarence, MCDANIEL, Keith, STEFFY, Kevin, MOLLA, Akhteruzzaman, HAYDEN, Frederick, KEMPF, Dale
Published in Antimicrobial Agents and Chemotherapy (01.04.2002)
Published in Antimicrobial Agents and Chemotherapy (01.04.2002)
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Structure-Based Characterization and Optimization of Novel Hydrophobic Binding Interactions in a Series of Pyrrolidine Influenza Neuraminidase Inhibitors
Maring, Clarence J, Stoll, Vincent S, Zhao, Chen, Sun, Minghua, Krueger, Allan C, Stewart, Kent D, Madigan, Darold L, Kati, Warren M, Xu, Yibo, Carrick, Robert J, Montgomery, Debra A, Kempf-Grote, Anita, Marsh, Kennan C, Molla, Akhteruzzaman, Steffy, Kevin R, Sham, Hing L, Laver, W. Graeme, Gu, Yu-gui, Kempf, Dale J, Kohlbrenner, William E
Published in Journal of medicinal chemistry (16.06.2005)
Published in Journal of medicinal chemistry (16.06.2005)
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Cationic lipids percentage and processing temperature are critical in designing siRNA lipid nanoparticles
Zhao, Xiaobin, Liu, Yemin, Song, Jingfeng, Yong, Hong, Li, Leiming, Shen, Yu, Hubbard, Robert D., Kohlbrenner, William E., Zhou, Ji, Cluff, Kevin D., Skoug, John W.
Published in Journal of drug targeting (01.04.2012)
Published in Journal of drug targeting (01.04.2012)
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Synthesis of potent pyrrolidine influenza neuraminidase inhibitors
Krueger, A. Chris, Xu, Yibo, Kati, Warren M., Kempf, Dale J., Maring, Clarence J., McDaniel, Keith F., Molla, Akhteruzzaman, Montgomery, Debra, Kohlbrenner, William E.
Published in Bioorganic & medicinal chemistry (01.03.2008)
Published in Bioorganic & medicinal chemistry (01.03.2008)
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Human Serum Attenuates the Activity of Protease Inhibitors toward Wild-Type and Mutant Human Immunodeficiency Virus
Molla, Akhteruzzaman, Vasavanonda, Sudthida, Kumar, Gondi, Sham, Hing L., Johnson, Marianne, Grabowski, Brian, Denissen, Jon F., Kohlbrenner, William, Plattner, Jacob J., Leonard, John M., Norbeck, Daniel W., Kempf, Dale J.
Published in Virology (New York, N.Y.) (25.10.1998)
Published in Virology (New York, N.Y.) (25.10.1998)
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Hepatitis C NS5B polymerase inhibitors: 4,4-Dialkyl-1-hydroxy-3-oxo-3,4-dihydronaphthalene-3-yl benzothiadiazine derivatives
Hutchinson, Douglas K., Rosenberg, Teresa, Klein, Larry L., Bosse, Todd D., Larson, Daniel P., He, Wenping, Jiang, Wen W., Kati, Warren M., Kohlbrenner, William E., Liu, Yaya, Masse, Sherie V., Middleton, Tim, Molla, Akhteruzzaman, Montgomery, Debra A., Beno, David W.A., Stewart, Kent D., Stoll, Vincent S., Kempf, Dale J.
Published in Bioorganic & medicinal chemistry (15.07.2008)
Published in Bioorganic & medicinal chemistry (15.07.2008)
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In Vitro Selection and Characterization of Influenza A (A/N9) Virus Variants Resistant to a Novel Neuraminidase Inhibitor, A-315675
Molla, Akhteruzzaman, Kati, Warren, Carrick, Robert, Steffy, Kevin, Shi, Yan, Montgomery, Debra, Gusick, Nanette, Stoll, Vincent S, Stewart, Kent D, Ng, Teresa I, Maring, Clarence, Kempf, Dale J, Kohlbrenner, William
Published in Journal of Virology (01.06.2002)
Published in Journal of Virology (01.06.2002)
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Novel α- and β-Amino Acid Inhibitors of Influenza Virus Neuraminidase
KATI, Warren M, MONTGOMERY, Debra, MARING, Clarence, STOLL, Vincent S, GIRANDA, Vincent, XIAOQI CHEN, LAVER, W. Graeme, KOHLBRENNER, William, NORBECK, Daniel W
Published in Antimicrobial Agents and Chemotherapy (01.09.2001)
Published in Antimicrobial Agents and Chemotherapy (01.09.2001)
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Inhibition of human immunodeficiency virus type I integrase by naphthamidines and 2-aminobenzimidazoles
Middleton, Tim, Lim, Hock B., Montgomery, Debra, Rockway, Todd, Tang, Hua, Cheng, Xueheng, Lu, Liangjun, Mo, Hongmei, Kohlbrenner, William E., Molla, Akhteruzzaman, Kati, Warren M.
Published in Antiviral research (01.10.2004)
Published in Antiviral research (01.10.2004)
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In Vitro Selection and Characterization of Human Immunodeficiency Virus Type 1 Variants with Increased Resistance to ABT-378, a Novel Protease Inhibitor
Carrillo, A, Stewart, K D, Sham, H L, Norbeck, D W, Kohlbrenner, W E, Leonard, J M, Kempf, D J, Molla, A
Published in Journal of Virology (01.09.1998)
Published in Journal of Virology (01.09.1998)
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Selection and Characterization of Varicella-Zoster Virus Variants Resistant to (R)-9-[4-Hydroxy-2-(Hydroxymethy)Butyl]Guanine
Ng, T I, Shi, Y, Huffaker, H J, Kati, W, Liu, Y, Chen, C M, Lin, Z, Maring, C, Kohlbrenner, W E, Molla, A
Published in Antimicrobial Agents and Chemotherapy (01.06.2001)
Published in Antimicrobial Agents and Chemotherapy (01.06.2001)
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New Quinolone Compounds from Pseudonocardia sp. with Selective and Potent Anti-Helicobacter pylori Activity: Taxonomy of Producing Strain, Fermentation, Isolation, Structural Elucidation and Biological Activities
DEKKER, KOEN A., INAGAKI, TAISUKE, GOOTZ, THOMAS D., HUANG, LIANG H., KOJIMA, YASUHIRO, KOHLBRENNER, WILLIAM E., MATSUNAGA, YASUE, MCGUIRK, PAUL R., NOMURA, ETSUKO, SAKAKIBARA, TATSUO, SAKEMI, SHINICHI, SUZUKI, YUMIKO, YAMAUCHI, YUJI, KOJIMA, NAKAO
Published in Journal of antibiotics (01.02.1998)
Published in Journal of antibiotics (01.02.1998)
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Symmetry-based inhibitors of HIV protease. Structure-activity studies of acylated 2,4-diamino-1,5-diphenyl-3-hydroxypentane and 2,5-diamino-1,6-diphenylhexane-3,4-diol
Kempf, Dale J, Codacovi, Lynnmarie, Wang, Xiu Chun, Kohlbrenner, William E, Wideburg, Norman E, Saldivar, Ayda, Vasavanonda, Sudthida, Marsh, Kennan C, Bryant, Pamela
Published in Journal of medicinal chemistry (01.02.1993)
Published in Journal of medicinal chemistry (01.02.1993)
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