Establishment of a novel, cell-based autotaxin assay
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Published in Analytical biochemistry (01.10.2021)
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Structure–Permeability Relationship of Semipeptidic MacrocyclesUnderstanding and Optimizing Passive Permeability and Efflux Ratio
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Published in Journal of medicinal chemistry (09.07.2020)
Published in Journal of medicinal chemistry (09.07.2020)
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Predictive Modeling of PROTAC Cell Permeability with Machine Learning
Poongavanam, Vasanthanathan, Kölling, Florian, Giese, Anja, Göller, Andreas H., Lehmann, Lutz, Meibom, Daniel, Kihlberg, Jan
Published in ACS omega (14.02.2023)
Published in ACS omega (14.02.2023)
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Structure-Permeability Relationship of Semi-Peptidic Macrocycles - Understanding and Optimizing Passive Permeability and Efflux Ratio
Le Roux, Antoine, Blaise, Emilie, Boudreault, Pierre-Luc, Comeau, Christian, Doucet, Annie, Giarrusso, Marilena, Collin, Marie-Pierre, Neubauer, Thomas, Koelling, Florian, Göller, Andreas H, Seep, Lea, Tshitenge, Dieudonné T, Wittwer, Matthias, Kullmann, Maximilian, Hillisch, Alexander, Mittendorf, Joachim, Marsault, Éric
Published in Journal of medicinal chemistry (26.05.2020)
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Published in Journal of medicinal chemistry (26.05.2020)
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치환된 5,6,7,8-테트라히드로[1,2,4]트리아졸로[4,3-a]피리딘-3(2H)-온 및 2,5,6,7-테트라히드로-3H-피롤로[2,1-c][1,2,4]트리아졸-3-온, 및 그의 용도
BADOCK VOLKER, MOOSMAYER DIETER, LUSTIG KLEMENS, TIMMERMANN ANDREAS, BIBER NICOLE, TERJUNG CARSTEN, MEIER HEINRICH, NEUBAUER THOMAS, LINDNER NIELS, MOORE STEVEN, ZUBOV DMITRY, KOELLING FLORIAN, MIYATAKE ONDOZABAL HIDEKI, SCHULZ ALEXANDER, BROCKSCHNIEDER DAMIAN, MEDING JOERG, GERICKE KERSTEN MATTHIAS, SCHAEFER MARTINA
Year of Publication 10.01.2019
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Year of Publication 10.01.2019
Patent
HYDROXYALKYL-SUBSTITUTED PHENYLTRIAZOLE DERIVATIVES AND USES THEREOF
LANG DIETER, MONDRITZKI THOMAS, WASNAIRE PIERRE, LUSTIG KLEMENS, POOK ELISABETH, GRIEBENOW NILS, ENGELEN ANNA, GERISCH MICHAEL, SUESSMEIER FRANK, KOELLING FLORIAN, KRETSCHMER AXEL, BECK HARTMUT, SCHMECK CARSTEN, KOLKHOF PETER, VOLLMER SONJA
Year of Publication 11.07.2017
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Year of Publication 11.07.2017
Patent
SUBSTITUTED 5,6,7,8-TETRAHYDRO[1,2,4]TRIAZOLO[4,3-A]PYRIDINE-3(2H)-ONES AND 2,5,6,7-TETRAHYDRO-3H-PYRROLO[2,1-C][1,2,4]TRIAZOL-3-ONES, AND USE THEREOF
NEUBAUER, Thomas, TIMMERMANN, Andreas, LINDNER, Niels, MEDING, Joerg, GERICKE, Kersten Matthias, MEIER, Heinrich, ZUBOV, Dmitry, BIBER, Nicole, SCHULZ, Alexander, MIYATAKE ONDOZABAL, Hideki, MOOSMAYER, Dieter, BADOCK, Volker, BROCKSCHNIEDER, Damian, LUSTIG, Klemens, TERJUNG, Carsten, MOORE, Stephen, SCHÄFER, Martina, KOELLING, Florian
Year of Publication 28.07.2024
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Year of Publication 28.07.2024
Patent
HYDROXYALKYL-SUBSTITUTED PHENYLTRIAZOLE DERIVATIVES AND USES THEREOF
GERISCH, Michael, GRIEBENOW, Nils, KOLKHOF, Peter, WASNAIRE, Pierre, KRETSCHMER, Axel, SCHMECK, Carsten, LUSTIG, Klemens, MONDRITZKI, Thomas, POOK, Elisabeth, BECK, Hartmut, SUESSMEIER, Frank, ENGELEN, Anna, KOELLING, Florian, LANG, Dieter, VOLLMER, Sonja
Year of Publication 28.03.2019
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Year of Publication 28.03.2019
Patent
Substituted 5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyridin-3(2h)-ones and 2,5,6,7-tetrahydro-3h-pyrrolo[2,1-c][1,2,4]triazol-3-ones and use thereof
KOELLING, FLORIAN, SCHAEFER, MARTINA, NEUBAUER, THOMAS, TIMMERMANN, ANDREAS, BADOCK, VOLKER, BROCKSCHNIEDER, DAMIAN, SCHULZ, ALEXANDER, BIBER, NICOLE, MEIER, HEINRICH, MOOSMAYER, DIETER, MIYATAKE ONDOZABAL, HIDEKI, GERICKE, KERSTEN MATTHIAS, ZUBOV, DMITRY, LINDNER, NIELS, MEDING, JOERG, MOORE, STEVEN, LUSTIG, KLEMENS, TERJUNG, CARSTEN
Year of Publication 21.03.2022
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Year of Publication 21.03.2022
Patent
SUBSTITUTED 5,6,7,8-TETRAHYDRO[1,2,4]TRIAZOLO[4,3-a]PYRIDINE-3(2H)-ONE AND 2,5,6,7-TETRAHYDRO-3H-PYRROLO[2,1-c][1,2,4]TRIAZOL-3-ONE, AND USE THEREOF
NEUBAUER, Thomas, TIMMERMANN, Andreas, LINDNER, Niels, MEDING, Joerg, MEIER, Heinrich, ZUBOV, Dmitry, BIBER, Nicole, SCHULZ, Alexander, MIYATAKE ONDOZABAL, Hideki, MOORE, Steven, SCHAEFER, Martina, MOOSMAYER, Dieter, BADOCK, Volker, BROCKSCHNEIDER, Damian, LUSTIG, Klemens, TERJUNG, Carsten, GERICKE, Kersten, Matthias, KOELLING, Florian
Year of Publication 08.04.2021
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Year of Publication 08.04.2021
Patent
Hydroxyalkyl-substituted phenyltriazole derivatives and uses thereof
KOELLING, FLORIAN, ENGELEN, ANNA, SUESSMEIER, FRANK, GRIEBENOW, NILS, MONDRITZKI, THOMAS, VOLLMER, SONJA, WASNAIRE, PIERRE, KRETSCHMER, AXEL, LANG, DIETER, GERISCH, MICHAEL, POOK, ELISABETH, SCHMECK, CARSTEN, LUSTIG, KLEMENS, KOLKHOF, PETER, BECK, HARTMUT
Year of Publication 21.05.2020
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Year of Publication 21.05.2020
Patent
HYDROXYALKYL-SUBSTITUTED PHENYLTRIAZOLE DERIVATIVES AND USES THEREOF
GERISCH, Michael, GRIEBENOW, Nils, KOLKHOF, Peter, WASNAIRE, Pierre, KRETSCHMER, Axel, SCHMECK, Carsten, LUSTIG, Klemens, MONDRITZKI, Thomas, POOK, Elisabeth, BECK, Hartmut, SUESSMEIER, Frank, ENGELEN, Anna, KOELLING, Florian, LANG, Dieter, VOLLMER, Sonja
Year of Publication 30.04.2019
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Year of Publication 30.04.2019
Patent
Substituted 5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-A]pyridin-3(2H)-ones and 2,5,6,7-tetrahydro-3H-pyrrolo[2,1-C][1,2,4]triazol-3-ones and use thereof
KOELLING, FLORIAN, SCHAEFER, MARTINA, NEUBAUER, THOMAS, TIMMERMANN, ANDREAS, BADOCK, VOLKER, BROCKSCHNIEDER, DAMIAN, SCHULZ, ALEXANDER, BIBER, NICOLE, MEIER, HEINRICH, MOOSMAYER, DIETER, MIYATAKE ONDOZABAL, HIDEKI, GERICKE, KERSTEN MATTHIAS, ZUBOV, DMITRY, LINDNER, NIELS, MEDING, JOERG, MOORE, STEVEN, LUSTIG, KLEMENS, TERJUNG, CARSTEN
Year of Publication 01.03.2018
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Year of Publication 01.03.2018
Patent
Hydroxyalkyl-substituted phenyltriazole derivatives and uses thereof
KOELLING, FLORIAN, ENGELEN, ANNA, SUESSMEIER, FRANK, GRIEBENOW, NILS, MONDRITZKI, THOMAS, VOLLMER, SONJA, WASNAIRE, PIERRE, KRETSCHMER, AXEL, LANG, DIETER, GERISCH, MICHAEL, POOK, ELISABETH, SCHMECK, CARSTEN, LUSTIG, KLEMENS, KOLKHOF, PETER, BECK, HARTMUT
Year of Publication 16.08.2016
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Year of Publication 16.08.2016
Patent
SUBSTITUTED 5,6,7,8-TETRAHYDRO[1,2,4]TRIAZOLO[4,3-A]PYRIDINE-3(2H)-ONES AND 2,5,6,7-TETRAHYDRO-3H-PYRROLO[2,1-C][1,2,4]TRIAZOL-3-ONES, AND USE THEREOF
NEUBAUER, Thomas, TIMMERMANN, Andreas, LINDNER, Niels, GERICKE, Kersten Matthias, MEIER, Heinrich, ZUBOV, Dmitry, BIBER, Nicole, SCHULZ, Alexander, MIYATAKE ONDOZABAL, Hideki, MOORE, Steven, KÖLLING, Florian, MOOSMAYER, Dieter, BADOCK, Volker, BROCKSCHNEIDER, Damian, LUSTIG, Klemens, TERJUNG, Carsten, SCHÄFER, Martina, MEDING, Jörg
Year of Publication 16.11.2017
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Year of Publication 16.11.2017
Patent