Discovery of 7-Methoxy-6-[4-(4-methyl-1,3-thiazol-2-yl)-1H-imidazol-5-yl]-1,3-benzothiazole (TASP0382088): A Potent and Selective Transforming Growth Factor-β Type I Receptor Inhibitor as a Topical Drug for Alopecia
Amada, Hideaki, Asanuma, Hajime, Koami, Takeshi, Okada, Atsushi, Endo, Mayumi, Ueda, Yasuji, Naruse, Takumi, Ikeda, Akiko
Published in Chemical & pharmaceutical bulletin (01.03.2013)
Published in Chemical & pharmaceutical bulletin (01.03.2013)
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Journal Article
Discovery of 7-Methoxy-6-[4-(4-methyl-1,3-thiazol-2-yl)-1H-imidazol-5-yl]-1,3-benzothiazole (TASP0382088)：A Potent and Selective Transforming Growth Factor-β Type I Receptor Inhibitor as a Topical Drug for Alopecia
Hideaki Amada, Hajime Asanuma, Takeshi Koami, Atsushi Okada, Mayumi Endo, Yasuji Ueda, Takumi Naruse, Akiko Ikeda
Published in Chemical and Pharmaceutical Bulletin (01.03.2013)
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Published in Chemical and Pharmaceutical Bulletin (01.03.2013)
Journal Article
5-(1,3-Benzothiazol-6-yl)-4-(4-methyl-1,3-thiazol-2-yl)-1H-imidazole derivatives as potent and selective transforming growth factor-β type I receptor inhibitors
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Published in Bioorganic & medicinal chemistry (15.12.2012)
Published in Bioorganic & medicinal chemistry (15.12.2012)
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Isoquinoline derivatives as potent CRTH2 antagonists: Design, synthesis and SAR
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Published in Bioorganic & medicinal chemistry (15.12.2013)
Published in Bioorganic & medicinal chemistry (15.12.2013)
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Isoquinoline derivatives as potent CRTH2 receptor antagonists: Synthesis and SAR
Nishikawa-Shimono, Rie, Sekiguchi, Yoshinori, Koami, Takeshi, Kawamura, Madoka, Wakasugi, Daisuke, Watanabe, Kazuhito, Wakahara, Shunichi, Matsumoto, Kayo, Takayama, Tetsuo
Published in Bioorganic & medicinal chemistry letters (01.05.2012)
Published in Bioorganic & medicinal chemistry letters (01.05.2012)
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Design, synthesis, and evaluation of novel 4-thiazolylimidazoles as inhibitors of transforming growth factor-β type I receptor kinase
Amada, Hideaki, Sekiguchi, Yoshinori, Ono, Naoya, Matsunaga, Yuko, Koami, Takeshi, Asanuma, Hajime, Shiozawa, Fumiyasu, Endo, Mayumi, Ikeda, Akiko, Aoki, Mari, Fujimoto, Natsuko, Wada, Reiko, Sato, Masakazu
Published in Bioorganic & medicinal chemistry letters (01.03.2012)
Published in Bioorganic & medicinal chemistry letters (01.03.2012)
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Journal Article
Discovery of 7-Methoxy-6-[4-(4-methyl-1,3-thiazol-2-yl)-1H-imidazol-5-yl]-1,3-benzothiazole (TASP0382088)
Amada, Hideaki, Asanuma, Hajime, Koami, Takeshi, Okada, Atsushi, Endo, Mayumi, Ueda, Yasuji, Naruse, Takumi, Ikeda, Akiko
Published in Chemical & pharmaceutical bulletin (01.03.2013)
Get full text
Published in Chemical & pharmaceutical bulletin (01.03.2013)
Journal Article
5-(1,3-Benzothiazol-6-yl)-4-(4-methyl-1,3-thiazol-2-yl)-1H-imidazo le derivatives as potent and selective transforming growth factor-[beta] type I receptor inhibitors
Amada, Hideaki, Sekiguchi, Yoshinori, Ono, Naoya, Koami, Takeshi, Takayama, Tetsuo, Yabuuchi, Tetsuya, Katakai, Hironori, Ikeda, Akiko, Aoki, Mari, Naruse, Takumi, Wada, Reiko, Nozoe, Akiko, Sato, Masakazu
Published in Bioorganic & medicinal chemistry (15.12.2012)
Published in Bioorganic & medicinal chemistry (15.12.2012)
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Journal Article
Isoquinoline derivatives as potent CRTH2 receptor antagonists: Synthesis andSAR
NISHIKAWA-SHIMONO, Rie, SEKIGUCHI, Yoshinori, KOAMI, Takeshi, KAWAMURA, Madoka, WAKASUGI, Daisuke, WATANABE, Kazuhito, WAKAHARA, Shunichi, MATSUMOTO, Kayo, TAKAYAMA, Tetsuo
Published in Bioorganic & medicinal chemistry letters (2012)
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Published in Bioorganic & medicinal chemistry letters (2012)
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Takayama, Tetsuo, Umemiya, Hiroki, Amada, Hideaki, Yabuuchi, Tetsuya, Koami, Takeshi, Shiozawa, Fumiyasu, Oka, Yusuke, Takaoka, Akiko, Yamaguchi, Akie, Endo, Mayumi, Sato, Masakazu
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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